GT200000220A - Forma de dosificacion de farmaco en capas impulsada por hidrogel. - Google Patents

Forma de dosificacion de farmaco en capas impulsada por hidrogel.

Info

Publication number
GT200000220A
GT200000220A GT200000220A GT200000220A GT200000220A GT 200000220 A GT200000220 A GT 200000220A GT 200000220 A GT200000220 A GT 200000220A GT 200000220 A GT200000220 A GT 200000220A GT 200000220 A GT200000220 A GT 200000220A
Authority
GT
Guatemala
Prior art keywords
dosage form
water
hydrogel
farmaco
sertraline
Prior art date
Application number
GT200000220A
Other languages
English (en)
Inventor
William John Curatolo
Michael Bruce Fergione
Michael Christopher Roy
Avinash Govind Thombre
Kenneth Craig Waterman
Leah Elizabeth Appel
Ronald Arthur Beyerinck
Dwayne Thomas Friesen
Danielle Supplee
Mark Brian Chidlaw
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of GT200000220A publication Critical patent/GT200000220A/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0002Galenical forms characterised by the drug release technique; Application systems commanded by energy
    • A61K9/0004Osmotic delivery systems; Sustained release driven by osmosis, thermal energy or gas
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • A61K31/135Amines having aromatic rings, e.g. ketamine, nortriptyline
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/10Drugs for genital or sexual disorders; Contraceptives for impotence
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/22Anxiolytics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/30Drugs for disorders of the nervous system for treating abuse or dependence
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/04Anorexiants; Antiobesity agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Biomedical Technology (AREA)
  • Epidemiology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Reproductive Health (AREA)
  • Psychiatry (AREA)
  • Endocrinology (AREA)
  • Addiction (AREA)
  • Child & Adolescent Psychology (AREA)
  • Diabetes (AREA)
  • Pain & Pain Management (AREA)
  • Anesthesiology (AREA)
  • Hematology (AREA)
  • Gynecology & Obstetrics (AREA)
  • Obesity (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicinal Preparation (AREA)

Abstract

UNA FORMA DE DOSIFICACION CONTROLADA PARA SERTRALINA EN UNA FORMA HINCHABLE CON AGUA, SEPARADA DEL NUCLEO DE SERTRALINA. UN REVESTIMIENTO EN TORNO AL NUCLEO ES PERMEABLE AL AGUA, INSOLUBLE EN AGUA, Y TIENE AL MENOS UNA ABERTURA DE SUMINISTRO A TRAVES DEL MISMO; EL MECANISMO CONSISTE EN UNA BICAPA OSMOTICA POR HIDROGEL, ESPECIFICAMENTE SE USA POLIOXIDO DE ETILENO MAS UN POLIMERO CELULOSICO HIDROFILO MAS AGLUTINANTE. EN UNA REALIZACION, LA FORMA DE DOSIFICACION LIBERA SERTRALINA HACIA EL ENTORNO DE USO CON UNA VELOCIDAD MEDIA DE 6 A 10% EN PESO POR HORA DESDE LA SEGUNDA HASTA DECIMA HORA DESPUES DE LA INTRODUCCION EN UN ENTORNO DE USO, Y MENOS DE APROXIMADAMENTE25% EN PESO DURANTE LAS DOS PRIMERAS HORAS Y AL MENOS 70% EN PESO AL CABO DE LA DECIMA HORA, EN DONDE LOS PORCENTAJES CORRESPONDEN A LA MASA DEL FARMACO LIBERADO DESDE EL COMPRIMIDO DIVIDIDA POR LA MASA TOTAL DE FARMACO ORIGINALMENTE PRESENTE EN EL COMPRIMIDO.
GT200000220A 1999-12-23 2000-12-21 Forma de dosificacion de farmaco en capas impulsada por hidrogel. GT200000220A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US17210899P 1999-12-23 1999-12-23

Publications (1)

Publication Number Publication Date
GT200000220A true GT200000220A (es) 2002-06-14

Family

ID=22626396

Family Applications (1)

Application Number Title Priority Date Filing Date
GT200000220A GT200000220A (es) 1999-12-23 2000-12-21 Forma de dosificacion de farmaco en capas impulsada por hidrogel.

Country Status (15)

Country Link
US (1) US6899896B2 (es)
EP (1) EP1239839A2 (es)
JP (1) JP2003518487A (es)
AR (1) AR027066A1 (es)
AU (1) AU1724301A (es)
BR (1) BR0016707A (es)
CA (1) CA2395231C (es)
CO (1) CO5271728A1 (es)
GT (1) GT200000220A (es)
MX (1) MXPA02006335A (es)
PA (1) PA8508901A1 (es)
PE (1) PE20010983A1 (es)
TN (1) TNSN00251A1 (es)
UY (1) UY26493A1 (es)
WO (1) WO2001047498A2 (es)

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US20030170309A1 (en) * 2001-06-22 2003-09-11 Babcock Walter C. Pharmaceutical compositions containing polymer and drug assemblies
JP2005529059A (ja) * 2001-09-28 2005-09-29 マクニール−ピーピーシー・インコーポレイテッド 改質した放出用の投薬形態
US20040146559A1 (en) * 2002-09-28 2004-07-29 Sowden Harry S. Dosage forms having an inner core and outer shell with different shapes
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Also Published As

Publication number Publication date
MXPA02006335A (es) 2002-12-13
US20010044474A1 (en) 2001-11-22
UY26493A1 (es) 2001-07-31
AU1724301A (en) 2001-07-09
WO2001047498A2 (en) 2001-07-05
CO5271728A1 (es) 2003-04-30
PE20010983A1 (es) 2001-10-01
JP2003518487A (ja) 2003-06-10
TNSN00251A1 (fr) 2002-05-30
EP1239839A2 (en) 2002-09-18
PA8508901A1 (es) 2003-12-10
CA2395231A1 (en) 2001-07-05
BR0016707A (pt) 2002-09-03
US6899896B2 (en) 2005-05-31
WO2001047498A3 (en) 2001-11-15
AR027066A1 (es) 2003-03-12
CA2395231C (en) 2006-08-15

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