GB1512194A - Benzamides - Google Patents
BenzamidesInfo
- Publication number
- GB1512194A GB1512194A GB6215/77A GB621577A GB1512194A GB 1512194 A GB1512194 A GB 1512194A GB 6215/77 A GB6215/77 A GB 6215/77A GB 621577 A GB621577 A GB 621577A GB 1512194 A GB1512194 A GB 1512194A
- Authority
- GB
- United Kingdom
- Prior art keywords
- benzamides
- halogen
- denotes
- benzoylaziridines
- haloethyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
- 229940054066 benzamide antipsychotics Drugs 0.000 title abstract 3
- 150000003936 benzamides Chemical class 0.000 title abstract 3
- YNAVUWVOSKDBBP-UHFFFAOYSA-N Morpholine Chemical compound C1COCCN1 YNAVUWVOSKDBBP-UHFFFAOYSA-N 0.000 abstract 2
- 229910052736 halogen Inorganic materials 0.000 abstract 2
- 150000002367 halogens Chemical class 0.000 abstract 2
- 208000020401 Depressive disease Diseases 0.000 abstract 1
- 150000001204 N-oxides Chemical class 0.000 abstract 1
- 239000002253 acid Substances 0.000 abstract 1
- HGBCPYMIZWPKMI-UHFFFAOYSA-N aziridin-1-yl(phenyl)methanone Chemical class C=1C=CC=CC=1C(=O)N1CC1 HGBCPYMIZWPKMI-UHFFFAOYSA-N 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 230000005494 condensation Effects 0.000 abstract 1
- 238000009833 condensation Methods 0.000 abstract 1
- 150000002431 hydrogen Chemical class 0.000 abstract 1
- 229910052739 hydrogen Inorganic materials 0.000 abstract 1
- 239000001257 hydrogen Substances 0.000 abstract 1
- 230000002401 inhibitory effect Effects 0.000 abstract 1
- 125000000449 nitro group Chemical group [O-][N+](*)=O 0.000 abstract 1
- 238000007254 oxidation reaction Methods 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 125000002023 trifluoromethyl group Chemical group FC(F)(F)* 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
- C07D295/04—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
- C07D295/12—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms
- C07D295/125—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms with the ring nitrogen atoms and the substituent nitrogen atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings
- C07D295/13—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms with the ring nitrogen atoms and the substituent nitrogen atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings to an acyclic saturated chain
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/26—Psychostimulants, e.g. nicotine, cocaine
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Medicinal Chemistry (AREA)
- Psychiatry (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Biomedical Technology (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pain & Pain Management (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| AT107076A AT345842B (de) | 1976-02-16 | 1976-02-16 | Verfahren zur herstellung von neuen morpholinderivaten, ihren n-oxyden und salzen |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| GB1512194A true GB1512194A (en) | 1978-05-24 |
Family
ID=3505951
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| GB6215/77A Expired GB1512194A (en) | 1976-02-16 | 1977-02-15 | Benzamides |
Country Status (28)
Cited By (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP1716851B1 (en) * | 2004-02-17 | 2012-05-02 | Ishihara Sangyo Kaisha, Ltd. | Thioamides and salts thereof and cytokine production inhibitors containing both |
| RU2570898C2 (ru) * | 2014-03-27 | 2015-12-20 | Федеральное государственное бюджетное образовательное учреждение высшего профессионального образования "Российский химико-технологический университет имени Д.И. Менделеева (РХТУ им. Д.И. Менделеева)" | Способ получения n-[2-(морфолин-4-ил)этил]-4-хлорбензамида (варианты) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US7960391B2 (en) | 2005-05-03 | 2011-06-14 | Bayer Cropscience Ag | Heterocyclylethylbenzamide derivatives |
| RU2414462C1 (ru) * | 2009-11-16 | 2011-03-20 | Федеральное государственное унитарное предприятие "Государственный научный центр "Научно-исследовательский институт органических полупродуктов и красителей" (ФГУП "ГНЦ "НИОПИК") | Способ получения 4-хлор-n-(2-морфолиноэтил)бензамида |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CH451142A (de) * | 1965-01-19 | 1968-05-15 | Sandoz Ag | Verfahren zur Herstellung neuer basisch substituierter Benzoesäureamide |
| FR1501846A (fr) * | 1966-09-26 | 1967-11-18 | Bellon Labor Sa Roger | Procédé amélioré pour la préparation des thioamides |
| US3787419A (en) * | 1971-07-01 | 1974-01-22 | American Home Prod | N-substituted-alpha,alpha,alpha-trifluoro-m-toluamides |
-
1976
- 1976-02-16 AT AT107076A patent/AT345842B/de not_active IP Right Cessation
- 1976-12-16 CH CH1581976A patent/CH623317A5/de not_active IP Right Cessation
-
1977
- 1977-01-06 AU AU21099/77A patent/AU506427B2/en not_active Expired
- 1977-01-12 YU YU60/77A patent/YU39983B/xx unknown
- 1977-01-12 SI SI7710060A patent/SI7710060A8/sl unknown
- 1977-01-27 AR AR266340A patent/AR214307A1/es active
- 1977-02-01 FI FI770356A patent/FI65426C/fi not_active IP Right Cessation
- 1977-02-03 NL NLAANVRAGE7701144,A patent/NL179382C/xx not_active IP Right Cessation
- 1977-02-08 DK DK51677A patent/DK148824C/da not_active IP Right Cessation
- 1977-02-09 ZA ZA770746A patent/ZA77746B/xx unknown
- 1977-02-09 IL IL51406A patent/IL51406A/xx unknown
- 1977-02-11 NZ NZ183316A patent/NZ183316A/xx unknown
- 1977-02-11 CA CA271,635A patent/CA1076112A/en not_active Expired
- 1977-02-11 IE IE296/77A patent/IE44482B1/en not_active IP Right Cessation
- 1977-02-14 FR FR7704087A patent/FR2340940A1/fr active Granted
- 1977-02-14 JP JP1431377A patent/JPS52100476A/ja active Granted
- 1977-02-14 LU LU76771A patent/LU76771A1/xx active Protection Beyond IP Right Term
- 1977-02-14 PH PH19452A patent/PH12847A/en unknown
- 1977-02-14 DE DE2706179A patent/DE2706179C2/de not_active Expired
- 1977-02-14 MC MC771233A patent/MC1136A1/xx unknown
- 1977-02-15 SE SE7701669A patent/SE426822B/xx not_active IP Right Cessation
- 1977-02-15 ES ES455907A patent/ES455907A1/es not_active Expired
- 1977-02-15 GR GR52790A patent/GR62413B/el unknown
- 1977-02-15 NO NO770488A patent/NO148417C/no unknown
- 1977-02-15 GB GB6215/77A patent/GB1512194A/en not_active Expired
- 1977-02-15 BE BE174926A patent/BE851422A/xx not_active IP Right Cessation
- 1977-02-15 PT PT66195A patent/PT66195B/pt unknown
- 1977-08-15 AR AR268800A patent/AR212554A1/es active
-
1978
- 1978-01-13 AT AT25578A patent/AT349479B/de not_active IP Right Cessation
- 1978-01-13 AT AT25678A patent/AT349480B/de not_active IP Right Cessation
- 1978-01-13 AT AT25878A patent/AT349482B/de not_active IP Right Cessation
- 1978-01-13 AT AT25778A patent/AT349481B/de not_active IP Right Cessation
- 1978-03-01 ES ES467449A patent/ES467449A1/es not_active Expired
- 1978-03-01 ES ES467455A patent/ES467455A1/es not_active Expired
- 1978-03-01 ES ES467448A patent/ES467448A1/es not_active Expired
-
1980
- 1980-07-18 CH CH554580A patent/CH623576A5/de not_active IP Right Cessation
- 1980-07-18 CH CH554680A patent/CH623577A5/de not_active IP Right Cessation
- 1980-07-18 CH CH554480A patent/CH622787A5/de not_active IP Right Cessation
- 1980-07-18 CH CH554380A patent/CH622786A5/de not_active IP Right Cessation
-
1993
- 1993-03-24 HR HRP-60/77A patent/HRP930495B1/xx not_active IP Right Cessation
- 1993-06-10 LU LU88300C patent/LU88300I2/de unknown
- 1993-06-17 NL NL930082C patent/NL930082I2/nl unknown
-
1994
- 1994-08-03 NO NO1994008C patent/NO1994008I1/no unknown
Cited By (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP1716851B1 (en) * | 2004-02-17 | 2012-05-02 | Ishihara Sangyo Kaisha, Ltd. | Thioamides and salts thereof and cytokine production inhibitors containing both |
| RU2570898C2 (ru) * | 2014-03-27 | 2015-12-20 | Федеральное государственное бюджетное образовательное учреждение высшего профессионального образования "Российский химико-технологический университет имени Д.И. Менделеева (РХТУ им. Д.И. Менделеева)" | Способ получения n-[2-(морфолин-4-ил)этил]-4-хлорбензамида (варианты) |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| PS | Patent sealed [section 19, patents act 1949] | ||
| 704A | Declaration that licence is not available as of right for an excepted use (par. 4a/1977) | ||
| 732 | Registration of transactions, instruments or events in the register (sect. 32/1977) | ||
| CTFF | Supplementary protection certificate filed |
Free format text: SPC/GB93/082, 930621 |
|
| CTFA | Application for supplementary protection certificate granted |
Free format text: SPC/GB93/082, 930928, EXPIRES:20020214 |
|
| CTFE | Supplementary protection certificate entered into force |
Free format text: SPC/GB93/082, 970215, EXPIRES:20020214 |
|
| PE20 | Patent expired after termination of 20 years |
Effective date: 19970214 |
|
| SPCE | Supplementary protection certificate expired |
Free format text: SPC/GB93/082: 20020214 |