GB0212412D0 - Combination of organic compounds - Google Patents

Combination of organic compounds

Info

Publication number
GB0212412D0
GB0212412D0 GBGB0212412.1A GB0212412A GB0212412D0 GB 0212412 D0 GB0212412 D0 GB 0212412D0 GB 0212412 A GB0212412 A GB 0212412A GB 0212412 D0 GB0212412 D0 GB 0212412D0
Authority
GB
United Kingdom
Prior art keywords
combination
organic compounds
compounds
organic
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
GBGB0212412.1A
Other languages
English (en)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Novartis AG
Original Assignee
Novartis AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novartis AG filed Critical Novartis AG
Priority to GBGB0212412.1A priority Critical patent/GB0212412D0/en
Publication of GB0212412D0 publication Critical patent/GB0212412D0/en
Priority to NZ548971A priority patent/NZ548971A/en
Priority to AU2003242593A priority patent/AU2003242593A1/en
Priority to PL03372571A priority patent/PL372571A1/xx
Priority to CNA2009100075473A priority patent/CN101518650A/zh
Priority to CNA038121840A priority patent/CN1655786A/zh
Priority to CA002487167A priority patent/CA2487167A1/en
Priority to MXPA04011785A priority patent/MXPA04011785A/es
Priority to JP2004506803A priority patent/JP2005532330A/ja
Priority to RU2004139025/15A priority patent/RU2336876C2/ru
Priority to EP03755149A priority patent/EP1511484A1/en
Priority to BR0311397-3A priority patent/BR0311397A/pt
Priority to NZ536758A priority patent/NZ536758A/en
Priority to PCT/EP2003/005639 priority patent/WO2003099279A1/en
Priority to US10/515,864 priority patent/US20060074058A1/en
Priority to ZA200408990A priority patent/ZA200408990B/en
Priority to IL16510104A priority patent/IL165101A0/xx
Priority to CO04124517A priority patent/CO5621286A2/es
Priority to NO20045557A priority patent/NO20045557L/no
Priority to US11/815,536 priority patent/US20070293474A1/en
Priority to RU2008119956/15A priority patent/RU2008119956A/ru
Priority to JP2010010967A priority patent/JP2010090173A/ja
Ceased legal-status Critical Current

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A61K31/454—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. pimozide, domperidone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/16—Amides, e.g. hydroxamic acids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/12—Drugs for disorders of the urinary system of the kidneys
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/10—Drugs for genital or sexual disorders; Contraceptives for impotence
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/04—Drugs for skeletal disorders for non-specific disorders of the connective tissue
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A61P27/06—Antiglaucoma agents or miotics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A61P27/12—Ophthalmic agents for cataracts
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/14—Drugs for disorders of the endocrine system of the thyroid hormones, e.g. T3, T4
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives

Landscapes

  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Diabetes (AREA)
  • Epidemiology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Cardiology (AREA)
  • Hematology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Obesity (AREA)
  • Endocrinology (AREA)
  • Urology & Nephrology (AREA)
  • Hospice & Palliative Care (AREA)
  • Vascular Medicine (AREA)
  • Emergency Medicine (AREA)
  • Child & Adolescent Psychology (AREA)
  • Dermatology (AREA)
  • Gynecology & Obstetrics (AREA)
  • Reproductive Health (AREA)
  • Biomedical Technology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
GBGB0212412.1A 2002-05-29 2002-05-29 Combination of organic compounds Ceased GB0212412D0 (en)

Priority Applications (22)

Application Number Priority Date Filing Date Title
GBGB0212412.1A GB0212412D0 (en) 2002-05-29 2002-05-29 Combination of organic compounds
US10/515,864 US20060074058A1 (en) 2002-05-29 2003-05-28 Combination of dpp iv inhibitor and a cardiovascular compound
EP03755149A EP1511484A1 (en) 2002-05-29 2003-05-28 Combination of a dpp iv inhibitor and a cardiovascular compound
NZ536758A NZ536758A (en) 2002-05-29 2003-05-28 Combination of a DPP IV inhibitor and a cardiovascular compound which is valsartan
PL03372571A PL372571A1 (en) 2002-05-29 2003-05-28 Combination of a dpp iv inhibitor and a cardiovascular compound
CNA2009100075473A CN101518650A (zh) 2002-05-29 2003-05-28 Dpp iv抑制剂和心血管化合物的组合
CNA038121840A CN1655786A (zh) 2002-05-29 2003-05-28 Dpp iv抑制剂和心血管化合物的组合
CA002487167A CA2487167A1 (en) 2002-05-29 2003-05-28 Combination of a dpp iv inhibitor and a cardiovascular compound
MXPA04011785A MXPA04011785A (es) 2002-05-29 2003-05-28 Combinacion de un inhibidor de dpp iv y un compuesto cardiovascular.
JP2004506803A JP2005532330A (ja) 2002-05-29 2003-05-28 Ｄｐｐｉｖ阻害剤および心臓血管化合物の組み合わせ
RU2004139025/15A RU2336876C2 (ru) 2002-05-29 2003-05-28 Комбинация ингибитора дипептидилпептидазы iv (dpp iv) и сердечно-сосудистого вещества
NZ548971A NZ548971A (en) 2002-05-29 2003-05-28 Combination of a DPP IV inhibitor and a cardiovascular compound
BR0311397-3A BR0311397A (pt) 2002-05-29 2003-05-28 Combinação de inibidor de dpp iv e um composto cardiovascular
AU2003242593A AU2003242593A1 (en) 2002-05-29 2003-05-28 Combination of a dpp iv inhibitor and a cardiovascular compound
PCT/EP2003/005639 WO2003099279A1 (en) 2002-05-29 2003-05-28 Combination of a dpp iv inhibitor and a cardiovascular compound
ZA200408990A ZA200408990B (en) 2002-05-29 2004-11-05 Combination of a DPP IV inhibitor and a cardiovascular compound
IL16510104A IL165101A0 (en) 2002-05-29 2004-11-08 Combination of a dpp IV inhibitor and a cardiovas cular compounds
CO04124517A CO5621286A2 (es) 2002-05-29 2004-12-13 Combinacion de un inhibidor de dpp iv y un compuesto cardiovascular
NO20045557A NO20045557L (no) 2002-05-29 2004-12-20 Kombinasjon av en DPP IV inhibitor og en kardiovaskulaer forbindelse
US11/815,536 US20070293474A1 (en) 2002-05-29 2007-08-03 Combination of a DPP IV inhibitor and a cardiovascular compound
RU2008119956/15A RU2008119956A (ru) 2002-05-29 2008-05-21 Комбинация ингибитора дипептидилпептидазы iv (dpp iv) и сердечно-сосудистого вещества
JP2010010967A JP2010090173A (ja) 2002-05-29 2010-01-21 Ｄｐｐｉｖ阻害剤および心臓血管化合物の組み合わせ

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GBGB0212412.1A GB0212412D0 (en) 2002-05-29 2002-05-29 Combination of organic compounds

Publications (1)

Publication Number Publication Date
GB0212412D0 true GB0212412D0 (en) 2002-07-10

Family

ID=9937665

Family Applications (1)

Application Number Title Priority Date Filing Date
GBGB0212412.1A Ceased GB0212412D0 (en) 2002-05-29 2002-05-29 Combination of organic compounds

Country Status (17)

Country Link
US (2) US20060074058A1 (enExample)
EP (1) EP1511484A1 (enExample)
JP (2) JP2005532330A (enExample)
CN (2) CN101518650A (enExample)
AU (1) AU2003242593A1 (enExample)
BR (1) BR0311397A (enExample)
CA (1) CA2487167A1 (enExample)
CO (1) CO5621286A2 (enExample)
GB (1) GB0212412D0 (enExample)
IL (1) IL165101A0 (enExample)
MX (1) MXPA04011785A (enExample)
NO (1) NO20045557L (enExample)
NZ (2) NZ548971A (enExample)
PL (1) PL372571A1 (enExample)
RU (2) RU2336876C2 (enExample)
WO (1) WO2003099279A1 (enExample)
ZA (1) ZA200408990B (enExample)

Families Citing this family (84)

* Cited by examiner, † Cited by third party
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US7407955B2 (en) 2002-08-21 2008-08-05 Boehringer Ingelheim Pharma Gmbh & Co., Kg 8-[3-amino-piperidin-1-yl]-xanthines, the preparation thereof and their use as pharmaceutical compositions
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US20040214804A1 (en) * 2003-04-25 2004-10-28 Pharmacia Corporation Combination of an aldosterone receptor antagonist and an anti-obesity agent
JP2007511467A (ja) 2003-05-14 2007-05-10 タケダ サン ディエゴ インコーポレイテッド ジペプチジルペプチダーゼインヒビター
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US7678909B1 (en) 2003-08-13 2010-03-16 Takeda Pharmaceutical Company Limited Dipeptidyl peptidase inhibitors
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US7501426B2 (en) 2004-02-18 2009-03-10 Boehringer Ingelheim International Gmbh 8-[3-amino-piperidin-1-yl]-xanthines, their preparation and their use as pharmaceutical compositions
US7732446B1 (en) 2004-03-11 2010-06-08 Takeda Pharmaceutical Company Limited Dipeptidyl peptidase inhibitors
CN102079743B (zh) 2004-03-15 2020-08-25 武田药品工业株式会社 二肽基肽酶抑制剂
RU2426532C2 (ru) * 2004-03-17 2011-08-20 Новартис Аг Применение органических соединений
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US7687638B2 (en) 2004-06-04 2010-03-30 Takeda San Diego, Inc. Dipeptidyl peptidase inhibitors
WO2006000564A1 (en) * 2004-06-23 2006-01-05 Solvay Pharmaceuticals Gmbh Pharmaceutical compositions comprising nep-inhibitors, inhibitors of the endogenous endothelin producing system and at1-receptor antagonists
WO2006019965A2 (en) 2004-07-16 2006-02-23 Takeda San Diego, Inc. Dipeptidyl peptidase inhibitors
RU2407523C2 (ru) * 2004-10-08 2010-12-27 Новартис Аг Применение ингибиторов ренина для профилактики или лечения диастолической дисфункции или диастолической сердечной недостаточности
DE102004054054A1 (de) 2004-11-05 2006-05-11 Boehringer Ingelheim Pharma Gmbh & Co. Kg Verfahren zur Herstellung chiraler 8-(3-Amino-piperidin-1-yl)-xanthine
JP2008524331A (ja) 2004-12-21 2008-07-10 武田薬品工業株式会社 ジペプチジルペプチダーゼ阻害剤
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BRPI0711558A2 (pt) 2006-05-04 2011-11-08 Boeringer Ingelheim Internat Gmbh polimorfos
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