GB0112836D0 - Medicaments - Google Patents

Medicaments

Info

Publication number
GB0112836D0
GB0112836D0 GBGB0112836.2A GB0112836A GB0112836D0 GB 0112836 D0 GB0112836 D0 GB 0112836D0 GB 0112836 A GB0112836 A GB 0112836A GB 0112836 D0 GB0112836 D0 GB 0112836D0
Authority
GB
United Kingdom
Prior art keywords
medicaments
derivatives
mammals
useful
treatment
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
GBGB0112836.2A
Other languages
English (en)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
SmithKline Beecham Ltd
Original Assignee
SmithKline Beecham Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by SmithKline Beecham Ltd filed Critical SmithKline Beecham Ltd
Priority to GBGB0112836.2A priority Critical patent/GB0112836D0/en
Publication of GB0112836D0 publication Critical patent/GB0112836D0/en
Priority to DE60215494T priority patent/DE60215494T2/de
Priority to AT02774022T priority patent/ATE342901T1/de
Priority to US10/477,900 priority patent/US7186730B2/en
Priority to ES02774022T priority patent/ES2275006T3/es
Priority to JP2003500086A priority patent/JP2004534780A/ja
Priority to PCT/EP2002/005709 priority patent/WO2002096907A1/en
Priority to EP02774022A priority patent/EP1392686B1/en
Ceased legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
GBGB0112836.2A 2001-05-25 2001-05-25 Medicaments Ceased GB0112836D0 (en)

Priority Applications (8)

Application Number Priority Date Filing Date Title
GBGB0112836.2A GB0112836D0 (en) 2001-05-25 2001-05-25 Medicaments
DE60215494T DE60215494T2 (de) 2001-05-25 2002-05-24 Bicyclische, stickstoffhaltige heterocyclische derivate zur verwendung als antibakterielle mittel
AT02774022T ATE342901T1 (de) 2001-05-25 2002-05-24 Bicyclische, stickstoffhaltige heterocyclische derivate zur verwendung als antibakterielle mittel
US10/477,900 US7186730B2 (en) 2001-05-25 2002-05-24 Bicyclic nitrogen-containing heterocyclic derivatives for use as antibacterials
ES02774022T ES2275006T3 (es) 2001-05-25 2002-05-24 Derivados heterociclicos biciclicos que contienen nitrogeno para usar como antibacterianos.
JP2003500086A JP2004534780A (ja) 2001-05-25 2002-05-24 抗菌剤として用いるための二環式窒素原子含有複素環誘導体
PCT/EP2002/005709 WO2002096907A1 (en) 2001-05-25 2002-05-24 Bicyclic nitrogen-containing heterocyclic derivatives for use as antibacterials
EP02774022A EP1392686B1 (en) 2001-05-25 2002-05-24 Bicyclic nitrogen-containing heterocyclic derivatives for use as antibacterials

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GBGB0112836.2A GB0112836D0 (en) 2001-05-25 2001-05-25 Medicaments

Publications (1)

Publication Number Publication Date
GB0112836D0 true GB0112836D0 (en) 2001-07-18

Family

ID=9915344

Family Applications (1)

Application Number Title Priority Date Filing Date
GBGB0112836.2A Ceased GB0112836D0 (en) 2001-05-25 2001-05-25 Medicaments

Country Status (8)

Country Link
US (1) US7186730B2 (enExample)
EP (1) EP1392686B1 (enExample)
JP (1) JP2004534780A (enExample)
AT (1) ATE342901T1 (enExample)
DE (1) DE60215494T2 (enExample)
ES (1) ES2275006T3 (enExample)
GB (1) GB0112836D0 (enExample)
WO (1) WO2002096907A1 (enExample)

Families Citing this family (46)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6803369B1 (en) 2000-07-25 2004-10-12 Smithkline Beecham Corporation Compounds and methods for the treatment of neoplastic disease
JP2004504397A (ja) 2000-07-26 2004-02-12 スミスクライン ビーチャム パブリック リミテッド カンパニー 抗菌活性を有するアミノピペリジンキノリン類およびそれらのアザイソステリックアナログ類
EP1320529B1 (en) * 2000-09-21 2006-05-24 Smithkline Beecham Plc Quinoline derivatives as antibacterials
GB0031088D0 (en) * 2000-12-20 2001-01-31 Smithkline Beecham Plc Medicaments
GB0031086D0 (en) * 2000-12-20 2001-01-31 Smithkline Beecham Plc Medicaments
GB0101577D0 (en) 2001-01-22 2001-03-07 Smithkline Beecham Plc Compounds
GB0112836D0 (en) 2001-05-25 2001-07-18 Smithkline Beecham Plc Medicaments
GB0112834D0 (en) * 2001-05-25 2001-07-18 Smithkline Beecham Plc Medicaments
GB0118238D0 (en) * 2001-07-26 2001-09-19 Smithkline Beecham Plc Medicaments
JP4445753B2 (ja) * 2002-01-29 2010-04-07 グラクソ グループ リミテッド アミノピペリジン誘導体
WO2003064431A2 (en) 2002-01-29 2003-08-07 Glaxo Group Limited Aminopiperidine compounds, process for their preparation, and pharmaceutical compositions containing them
AR040336A1 (es) * 2002-06-26 2005-03-30 Glaxo Group Ltd Compuesto de piperidina, uso del mismo para la fabricacion de un medicamento, composicion farmaceutica que lo comprende y procedimiento para preparar dicho compuesto
TW200406413A (en) 2002-06-26 2004-05-01 Glaxo Group Ltd Compounds
EP1560488B1 (en) 2002-11-05 2010-09-01 Glaxo Group Limited Antibacterial agents
ES2340484T3 (es) 2002-11-05 2010-06-04 Glaxo Group Limited Agentes antibacterianos.
ES2343127T3 (es) * 2004-10-05 2010-07-23 Actelion Pharmaceuticals Ltd. Nuevos antibioticos de piperidina.
WO2006081289A2 (en) * 2005-01-25 2006-08-03 Glaxo Group Limited Antibacterial agents
US7592334B2 (en) 2005-01-25 2009-09-22 Glaxo Group Limited Antibacterial agents
WO2006081179A1 (en) * 2005-01-25 2006-08-03 Glaxo Group Limited Antibacterial agents
JP2008528586A (ja) * 2005-01-25 2008-07-31 グラクソ グループ リミテッド 抗菌剤
WO2006081264A1 (en) 2005-01-25 2006-08-03 Glaxo Group Limited Antibacterial agents
MY150958A (en) 2005-06-16 2014-03-31 Astrazeneca Ab Compounds for the treatment of multi-drug resistant bacterial infections
DE602006012535D1 (de) * 2005-10-21 2010-04-08 Glaxo Group Ltd Peri-kondensierte tricyclische verbindungen verwendbar als antibakterielle mittel
US20070185153A1 (en) * 2005-12-22 2007-08-09 Nathalie Cailleau Compounds
MX2008010671A (es) * 2006-02-21 2008-10-01 Amgen Inc Derivados de cinolina como inhibidores de fosfodiesterasa 10.
WO2007100880A1 (en) * 2006-02-28 2007-09-07 Amgen Inc. Cinnoline and quinazoline derivates as phosphodiesterase 10 inhibitors
MX2008011257A (es) * 2006-03-08 2008-09-25 Amgen Inc Derivados de quinolina e isoquinolina como inhibidores de fosfodiesterasa 10.
EP2007377A4 (en) 2006-04-06 2011-08-17 Glaxo Group Ltd ANTIBACTERIAL ACTIVE SUBSTANCES
DE602007009205D1 (de) 2006-04-06 2010-10-28 Glaxo Group Ltd Pyrrolochinoxalinonderivate als antibakterielle mittel
GB0608263D0 (en) 2006-04-26 2006-06-07 Glaxo Group Ltd Compounds
AU2007268749B2 (en) 2006-05-26 2012-07-26 Taisho Pharmaceutical Co., Ltd. Novel heterocyclic compound or salt thereof and intermediate thereof
GB0613208D0 (en) 2006-07-03 2006-08-09 Glaxo Group Ltd Compounds
EP1992628A1 (en) 2007-05-18 2008-11-19 Glaxo Group Limited Derivatives and analogs of N-ethylquinolones and N-ethylazaquinolones
CL2008001003A1 (es) * 2007-04-11 2008-10-17 Actelion Pharmaceuticals Ltd Compuestos derivados de oxazolidinona; composicion farmaceutica que comprende a dichos compuestos; y su uso para preparar un medicamento para tratar una infeccion bacteriana.
CL2008001002A1 (es) * 2007-04-11 2008-10-17 Actelion Pharmaceuticals Ltd Compuestos derivados de oxazolidinona; composicion farmaceutica que comprende a dichos compuestos; y su uso para preparar un medicamento para tratar una infeccion bacteriana.
WO2008128942A1 (en) * 2007-04-20 2008-10-30 Glaxo Group Limited Tricyclic nitrogen containing compounds as antibacterial agents
CA2685888A1 (en) 2007-05-09 2008-11-20 Pfizer Inc. Substituted heterocyclic derivatives and their pharmaceutical use and compositions
BRPI0820985A2 (pt) 2007-12-18 2015-06-16 Actelion Pharmaceuticals Ltd Composto derivado de 5-aminociclometil-oxazondin-2-ona, medicamento e composição farmacêutica que os contém e uso dos mesmos
EP2080761A1 (en) 2008-01-18 2009-07-22 Glaxo Group Limited Compounds
US8466168B2 (en) * 2008-08-04 2013-06-18 Actellon Pharmaceuticals Ltd. Tricyclic alkylaminomethyloxazolidinone derivatives
JP2012505866A (ja) 2008-10-17 2012-03-08 グラクソ グループ リミテッド 抗菌剤として使用される三環式窒素化合物
JP5653935B2 (ja) 2009-01-15 2015-01-14 グラクソ グループ リミテッドGlaxo Group Limited 抗菌薬として有用なナフチリジン―2(1h)−オン化合物
AR089929A1 (es) 2012-02-10 2014-10-01 Actelion Pharmaceuticals Ltd Proceso para manufacturar un derivado de naftiridina
AR101674A1 (es) 2014-08-22 2017-01-04 Glaxosmithkline Ip Dev Ltd Uso de un compuesto tricíclico que contiene nitrógeno
UY36851A (es) 2015-08-16 2017-03-31 Glaxosmithkline Ip Dev Ltd Compuestos para uso en aplicaciones antibacterianas
CN114793434A (zh) 2019-10-18 2022-07-26 加利福尼亚大学董事会 作为用于治疗病原性血管病症的药剂的3-苯基磺酰基-喹啉衍生物

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JP4445753B2 (ja) 2002-01-29 2010-04-07 グラクソ グループ リミテッド アミノピペリジン誘導体
WO2003064431A2 (en) 2002-01-29 2003-08-07 Glaxo Group Limited Aminopiperidine compounds, process for their preparation, and pharmaceutical compositions containing them

Also Published As

Publication number Publication date
ATE342901T1 (de) 2006-11-15
WO2002096907A1 (en) 2002-12-05
ES2275006T3 (es) 2007-06-01
DE60215494D1 (de) 2006-11-30
EP1392686B1 (en) 2006-10-18
DE60215494T2 (de) 2007-03-15
JP2004534780A (ja) 2004-11-18
US7186730B2 (en) 2007-03-06
US20040198755A1 (en) 2004-10-07
EP1392686A1 (en) 2004-03-03

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Legal Events

Date Code Title Description
AT Applications terminated before publication under section 16(1)