GB0030710D0 - Piperazine derivatives - Google Patents
Piperazine derivativesInfo
- Publication number
- GB0030710D0 GB0030710D0 GBGB0030710.8A GB0030710A GB0030710D0 GB 0030710 D0 GB0030710 D0 GB 0030710D0 GB 0030710 A GB0030710 A GB 0030710A GB 0030710 D0 GB0030710 D0 GB 0030710D0
- Authority
- GB
- United Kingdom
- Prior art keywords
- piperazine derivatives
- piperazine
- derivatives
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Ceased
Links
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/30—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
- C07D207/32—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
- C07D207/325—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms with substituted hydrocarbon radicals directly attached to the ring nitrogen atom
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
- C07D295/16—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
- C07D295/20—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carbonic acid, or sulfur or nitrogen analogues thereof
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- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
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- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D213/28—Radicals substituted by singly-bound oxygen or sulphur atoms
- C07D213/30—Oxygen atoms
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
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- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/62—Oxygen or sulfur atoms
- C07D213/63—One oxygen atom
- C07D213/64—One oxygen atom attached in position 2 or 6
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- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
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- C07D213/62—Oxygen or sulfur atoms
- C07D213/63—One oxygen atom
- C07D213/64—One oxygen atom attached in position 2 or 6
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- C07D295/21—Radicals derived from sulfur analogues of carbonic acid
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Priority Applications (20)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GBGB0030710.8A GB0030710D0 (en) | 2000-12-15 | 2000-12-15 | Piperazine derivatives |
| JP2002549655A JP4047724B2 (ja) | 2000-12-15 | 2001-12-06 | ピペラジン誘導体 |
| EP01990522A EP1343775B1 (en) | 2000-12-15 | 2001-12-06 | Piperazine derivatives |
| DE60134338T DE60134338D1 (de) | 2000-12-15 | 2001-12-06 | Piperazin-derivate |
| PCT/EP2001/014343 WO2002048124A2 (en) | 2000-12-15 | 2001-12-06 | Piperazine derivatives |
| AU2962602A AU2962602A (en) | 2000-12-15 | 2001-12-06 | Piperazine derivatives |
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- 2001-12-12 PA PA20018534801A patent/PA8534801A1/es unknown
- 2001-12-12 AR ARP010105788A patent/AR035517A1/es not_active Application Discontinuation
- 2001-12-13 PE PE2001001247A patent/PE20020667A1/es not_active Application Discontinuation
- 2001-12-14 UY UY27075A patent/UY27075A1/es not_active Application Discontinuation
-
2003
- 2003-06-03 ZA ZA200304346A patent/ZA200304346B/en unknown
-
2004
- 2004-06-23 US US10/874,662 patent/US7022707B2/en not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| UY27075A1 (es) | 2002-07-31 |
| ZA200304346B (en) | 2004-09-03 |
| ATE397595T1 (de) | 2008-06-15 |
| CN1277824C (zh) | 2006-10-04 |
| PA8534801A1 (es) | 2002-08-26 |
| WO2002048124A3 (en) | 2003-06-05 |
| JP2004519438A (ja) | 2004-07-02 |
| JP4047724B2 (ja) | 2008-02-13 |
| CN1533382A (zh) | 2004-09-29 |
| CA2430601C (en) | 2008-05-06 |
| ES2306736T3 (es) | 2008-11-16 |
| US20020143020A1 (en) | 2002-10-03 |
| DE60134338D1 (de) | 2008-07-17 |
| US7022707B2 (en) | 2006-04-04 |
| AR035517A1 (es) | 2004-06-02 |
| CA2430601A1 (en) | 2002-06-20 |
| KR20030072563A (ko) | 2003-09-15 |
| BR0116201A (pt) | 2004-03-02 |
| EP1343775A2 (en) | 2003-09-17 |
| AU2962602A (en) | 2002-06-24 |
| EP1343775B1 (en) | 2008-06-04 |
| KR100623833B1 (ko) | 2006-09-18 |
| MXPA03005270A (es) | 2003-09-25 |
| WO2002048124A2 (en) | 2002-06-20 |
| US20040235859A1 (en) | 2004-11-25 |
| PE20020667A1 (es) | 2002-07-27 |
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| AT | Applications terminated before publication under section 16(1) |