GB0021421D0 - Compounds - Google Patents
CompoundsInfo
- Publication number
- GB0021421D0 GB0021421D0 GBGB0021421.3A GB0021421A GB0021421D0 GB 0021421 D0 GB0021421 D0 GB 0021421D0 GB 0021421 A GB0021421 A GB 0021421A GB 0021421 D0 GB0021421 D0 GB 0021421D0
- Authority
- GB
- United Kingdom
- Prior art keywords
- sub
- hydrogen
- specific substituents
- compounds
- independently
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Ceased
Links
- 150000001875 compounds Chemical class 0.000 title abstract 2
- 229910052739 hydrogen Inorganic materials 0.000 abstract 3
- 239000001257 hydrogen Substances 0.000 abstract 3
- 150000002431 hydrogen Chemical group 0.000 abstract 2
- 125000001424 substituent group Chemical group 0.000 abstract 2
- 101100516572 Caenorhabditis elegans nhr-8 gene Proteins 0.000 abstract 1
- 206010017533 Fungal infection Diseases 0.000 abstract 1
- UFHFLCQGNIYNRP-UHFFFAOYSA-N Hydrogen Chemical compound [H][H] UFHFLCQGNIYNRP-UHFFFAOYSA-N 0.000 abstract 1
- 208000031888 Mycoses Diseases 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 125000000547 substituted alkyl group Chemical group 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/10—Antimycotics
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Communicable Diseases (AREA)
- Animal Behavior & Ethology (AREA)
- Oncology (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Thiazole And Isothizaole Compounds (AREA)
Priority Applications (9)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GBGB0021421.3A GB0021421D0 (en) | 2000-08-31 | 2000-08-31 | Compounds |
| JP2002522888A JP2004507501A (ja) | 2000-08-31 | 2001-08-30 | ベンジリデンチアゾリジンジオンおよび抗真菌剤としてのそれらの使用 |
| ES01963157T ES2282283T3 (es) | 2000-08-31 | 2001-08-30 | Derivados de bencilideno tiazolidinadionas y su uso como agentes antifungicos. |
| EP01963157A EP1313471B1 (en) | 2000-08-31 | 2001-08-30 | Benzylidene thiazolidinediones and their use as antimycotic agents |
| AT01963157T ATE359073T1 (de) | 2000-08-31 | 2001-08-30 | Benzylidenthiazolidindione und ihre verwendung als antimykotische mittel |
| PCT/GB2001/003862 WO2002017915A1 (en) | 2000-08-31 | 2001-08-30 | Benzylidene thiazolidinediones and their use as antimycotic agents |
| AU2001284190A AU2001284190A1 (en) | 2000-08-31 | 2001-08-30 | Benzylidene thiazolidinediones and their use as antimycotic agents |
| DE60127845T DE60127845T2 (de) | 2000-08-31 | 2001-08-30 | Benzylidenthiazolidindione und ihre verwendung als antimykotische mittel |
| US10/371,964 US7105554B2 (en) | 2000-08-31 | 2003-02-21 | Benzylidene thiazolidinediones and their use as antimycotic agents |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GBGB0021421.3A GB0021421D0 (en) | 2000-08-31 | 2000-08-31 | Compounds |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| GB0021421D0 true GB0021421D0 (en) | 2000-10-18 |
Family
ID=9898616
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| GBGB0021421.3A Ceased GB0021421D0 (en) | 2000-08-31 | 2000-08-31 | Compounds |
Country Status (9)
| Country | Link |
|---|---|
| US (1) | US7105554B2 (enExample) |
| EP (1) | EP1313471B1 (enExample) |
| JP (1) | JP2004507501A (enExample) |
| AT (1) | ATE359073T1 (enExample) |
| AU (1) | AU2001284190A1 (enExample) |
| DE (1) | DE60127845T2 (enExample) |
| ES (1) | ES2282283T3 (enExample) |
| GB (1) | GB0021421D0 (enExample) |
| WO (1) | WO2002017915A1 (enExample) |
Families Citing this family (23)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB0204252D0 (en) * | 2002-02-23 | 2002-04-10 | Oxford Glycosciences Uk Ltd | Novel compounds |
| WO2003070238A1 (en) * | 2002-02-23 | 2003-08-28 | Oxford Glycosciences (Uk) Ltd | Thiazolidine antifungal agents |
| WO2005092840A1 (en) | 2004-03-23 | 2005-10-06 | Pfizer Limited | Formamide derivatives useful as adrenoceptor |
| CA2628725A1 (en) | 2005-11-15 | 2007-05-31 | Glycofi, Inc. | Production of glycoproteins with reduced o-glycosylation |
| WO2007079466A2 (en) * | 2006-01-04 | 2007-07-12 | Nano Mist International, Llc | Air driven delivery system for sprayable media |
| US8637435B2 (en) * | 2007-11-16 | 2014-01-28 | Merck Sharp & Dohme Corp. | Eukaryotic cell display systems |
| JP5731827B2 (ja) * | 2008-03-03 | 2015-06-10 | グライコフィ, インコーポレイテッド | 下等真核生物中での組換えタンパク質の表面ディスプレイ |
| AU2009249314A1 (en) | 2008-05-20 | 2009-11-26 | Merck Sharp & Dohme Corp. | Efficient production of heterologous proteins using mannosyl transferase inhibitors |
| US8067339B2 (en) | 2008-07-09 | 2011-11-29 | Merck Sharp & Dohme Corp. | Surface display of whole antibodies in eukaryotes |
| EP2324121B1 (en) | 2008-08-12 | 2012-11-07 | GlycoFi, Inc. | Improved vectors and yeast strains for protein production: ca2+ atpase overexpression |
| EP2678440B1 (en) | 2011-02-25 | 2018-05-23 | Merck Sharp & Dohme Corp. | Yeast strain for the production of proteins with modified o-glycosylation |
| WO2013018735A1 (ja) | 2011-07-29 | 2013-02-07 | 大正製薬株式会社 | アミジン化合物又はその塩 |
| WO2014024897A1 (ja) * | 2012-08-06 | 2014-02-13 | Meiji Seikaファルマ株式会社 | チアゾリジンジオンおよびピロリジンジオン誘導体、並びにそれらを有効成分としてなる殺菌剤 |
| WO2014062811A2 (en) * | 2012-10-16 | 2014-04-24 | New York University | METHOD OF TREATING CANCER WITH MODULATORS OF SCFSkp2 |
| MX364532B (es) | 2013-07-04 | 2019-04-29 | Glykos Finland Oy | Celulas de hongos filamentosos deficientes de o-manosiltransferasa y metodos de uso de las mismas. |
| SG11201700446XA (en) | 2014-07-21 | 2017-02-27 | Glykos Finland Oy | Production of glycoproteins with mammalian-like n-glycans in filamentous fungi |
| EP3468555B1 (en) * | 2016-06-14 | 2023-08-09 | Versitech Limited | Compositions for use in treating bacterial infections |
| CN109476656A (zh) * | 2016-06-24 | 2019-03-15 | 俄亥俄州大学 | 葡萄糖转运抑制剂及使用其的方法 |
| RU2662153C1 (ru) * | 2017-04-20 | 2018-07-24 | Общество С Ограниченной Ответственностью "Дермавитал Групп" | Гибридные эфиры на основе производных тиазолидин-2,4-диона и азолов (1н-1,3-имидазола и 1н-1,3,4-триазола) и их применение |
| RU2690161C1 (ru) * | 2018-06-28 | 2019-05-31 | Общество С Ограниченной Ответственностью "Дермавитал Групп" | 3,5-Замещенные производные тиазолидин-2,4-диона, обладающие противомикробной активностью |
| RU2703997C1 (ru) * | 2018-12-13 | 2019-10-23 | Общество с ограниченной ответственностью "Л-Био" | Гибридные амиды на основе триазола и тиазолидина, обладающие антимикробной активностью |
| CN112521382A (zh) * | 2020-12-14 | 2021-03-19 | 西南大学 | 芦荟大黄素噻唑烷二酮类化合物及其制备方法和应用 |
| WO2024258316A1 (ru) * | 2023-06-16 | 2024-12-19 | Общество с ограниченной ответственностью "Л-Био" | Новые потенциальные противогрибковые средства на основе тиазолидин-2,4-диона и триазола |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS6156175A (ja) * | 1984-08-24 | 1986-03-20 | Yamanouchi Pharmaceut Co Ltd | ロダニン誘導体およびその製造法 |
| IL106877A (en) * | 1992-09-10 | 1998-03-10 | Lilly Co Eli | Rhodanine derivatives for use as medicaments for the treatment of alzheimer's disease |
| DE4318550A1 (de) * | 1993-06-04 | 1994-12-08 | Boehringer Mannheim Gmbh | Aryliden-4-oxo-2-thioxo-3- thiazolidincarbonsäuren, Verfahren zu ihrer Herstellung und diese Verbindungen enthaltende Arzneimittel |
| JPH08109175A (ja) * | 1994-10-07 | 1996-04-30 | Torii Yakuhin Kk | チアゾリジン−2−オンエステル誘導体 |
| JPH08109174A (ja) * | 1994-10-07 | 1996-04-30 | Torii Yakuhin Kk | チアゾリジン−2−オン誘導体 |
| EP1117655A1 (en) * | 1998-09-30 | 2001-07-25 | Angelika Esswein | Rhodanine carboxylic acid derivatives for the treatment and prevention of metabolic bone disorders |
| WO2000018746A1 (en) * | 1998-09-30 | 2000-04-06 | Roche Diagnostics Gmbh | Thiazolidine derivatives for the treatment and prevention of metabolic bone disorders |
| US6506755B2 (en) * | 2000-02-03 | 2003-01-14 | Hoffmann-La Roche Inc. | Thiazolidinecarboxyl acids |
-
2000
- 2000-08-31 GB GBGB0021421.3A patent/GB0021421D0/en not_active Ceased
-
2001
- 2001-08-30 JP JP2002522888A patent/JP2004507501A/ja active Pending
- 2001-08-30 DE DE60127845T patent/DE60127845T2/de not_active Expired - Lifetime
- 2001-08-30 EP EP01963157A patent/EP1313471B1/en not_active Expired - Lifetime
- 2001-08-30 ES ES01963157T patent/ES2282283T3/es not_active Expired - Lifetime
- 2001-08-30 AU AU2001284190A patent/AU2001284190A1/en not_active Abandoned
- 2001-08-30 AT AT01963157T patent/ATE359073T1/de not_active IP Right Cessation
- 2001-08-30 WO PCT/GB2001/003862 patent/WO2002017915A1/en not_active Ceased
-
2003
- 2003-02-21 US US10/371,964 patent/US7105554B2/en not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| DE60127845D1 (de) | 2007-05-24 |
| US20040006112A1 (en) | 2004-01-08 |
| JP2004507501A (ja) | 2004-03-11 |
| ES2282283T3 (es) | 2007-10-16 |
| EP1313471B1 (en) | 2007-04-11 |
| ATE359073T1 (de) | 2007-05-15 |
| EP1313471A1 (en) | 2003-05-28 |
| WO2002017915A1 (en) | 2002-03-07 |
| AU2001284190A1 (en) | 2002-03-13 |
| US7105554B2 (en) | 2006-09-12 |
| DE60127845T2 (de) | 2007-12-20 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| AT | Applications terminated before publication under section 16(1) |