ATE359073T1 - Benzylidenthiazolidindione und ihre verwendung als antimykotische mittel - Google Patents

Benzylidenthiazolidindione und ihre verwendung als antimykotische mittel

Info

Publication number
ATE359073T1
ATE359073T1 AT01963157T AT01963157T ATE359073T1 AT E359073 T1 ATE359073 T1 AT E359073T1 AT 01963157 T AT01963157 T AT 01963157T AT 01963157 T AT01963157 T AT 01963157T AT E359073 T1 ATE359073 T1 AT E359073T1
Authority
AT
Austria
Prior art keywords
sub
benzylidenthiazolidindiones
antifungal agents
hydrogen
specific substituents
Prior art date
Application number
AT01963157T
Other languages
German (de)
English (en)
Inventor
Michael Glen Orchard
Judi Charlotte Neuss
Carl Maurice Swedler Galley
Original Assignee
Ucb Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ucb Sa filed Critical Ucb Sa
Application granted granted Critical
Publication of ATE359073T1 publication Critical patent/ATE359073T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10—Antimycotics
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Communicable Diseases (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
AT01963157T 2000-08-31 2001-08-30 Benzylidenthiazolidindione und ihre verwendung als antimykotische mittel ATE359073T1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GBGB0021421.3A GB0021421D0 (en) 2000-08-31 2000-08-31 Compounds

Publications (1)

Publication Number Publication Date
ATE359073T1 true ATE359073T1 (de) 2007-05-15

Family

ID=9898616

Family Applications (1)

Application Number Title Priority Date Filing Date
AT01963157T ATE359073T1 (de) 2000-08-31 2001-08-30 Benzylidenthiazolidindione und ihre verwendung als antimykotische mittel

Country Status (9)

Country Link
US (1) US7105554B2 (enExample)
EP (1) EP1313471B1 (enExample)
JP (1) JP2004507501A (enExample)
AT (1) ATE359073T1 (enExample)
AU (1) AU2001284190A1 (enExample)
DE (1) DE60127845T2 (enExample)
ES (1) ES2282283T3 (enExample)
GB (1) GB0021421D0 (enExample)
WO (1) WO2002017915A1 (enExample)

Families Citing this family (23)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB0204252D0 (en) * 2002-02-23 2002-04-10 Oxford Glycosciences Uk Ltd Novel compounds
WO2003070238A1 (en) * 2002-02-23 2003-08-28 Oxford Glycosciences (Uk) Ltd Thiazolidine antifungal agents
AU2005225632B2 (en) 2004-03-23 2011-08-04 Pfizer Inc. Formamide derivatives useful as adrenoceptor
EP1954815B1 (en) * 2005-11-15 2015-02-25 GlycoFi, Inc. Production of glycoproteins with reduced o-glycosylation
WO2007079466A2 (en) * 2006-01-04 2007-07-12 Nano Mist International, Llc Air driven delivery system for sprayable media
US8637435B2 (en) * 2007-11-16 2014-01-28 Merck Sharp & Dohme Corp. Eukaryotic cell display systems
WO2009111183A1 (en) * 2008-03-03 2009-09-11 Glycofi, Inc. Surface display of recombinant proteins in lower eukaryotes
ATE536347T1 (de) * 2008-05-20 2011-12-15 Merck Sharp & Dohme Effiziente herstellung heterologer proteine unter verwendung von mannosyltransferaseinhibitoren
US8067339B2 (en) 2008-07-09 2011-11-29 Merck Sharp & Dohme Corp. Surface display of whole antibodies in eukaryotes
JP2011530311A (ja) 2008-08-12 2011-12-22 グライコフィ， インコーポレイテッド タンパク質製造のための改良されたベクターおよび酵母株：Ｃａ２＋ＡＴＰアーゼ過剰発現
US8936918B2 (en) 2011-02-25 2015-01-20 Merck Sharp & Dohme Corp. Yeast strain for the production of proteins with modified O-glycosylation
MX336268B (es) * 2011-07-29 2016-01-13 Toyama Chemical Co Ltd Compuesto de amidina o sal del mismo.
WO2014024897A1 (ja) * 2012-08-06 2014-02-13 Ｍｅｉｊｉ Ｓｅｉｋａファルマ株式会社 チアゾリジンジオンおよびピロリジンジオン誘導体、並びにそれらを有効成分としてなる殺菌剤
US9261497B2 (en) 2012-10-16 2016-02-16 New York University Method of treating cancer with modulators of SCFSkp2
WO2015001049A1 (en) 2013-07-04 2015-01-08 Novartis Ag O-mannosyltransferase deficient filamentous fungal cells and methods of use thereof
CN108064266A (zh) 2014-07-21 2018-05-22 格利科斯芬兰公司 在丝状真菌中具有哺乳动物样n-聚糖的糖蛋白的制备
JP2019523229A (ja) * 2016-06-14 2019-08-22 ヴェルシテック リミテッド 抗微生物化合物及びその使用方法
WO2017223473A1 (en) * 2016-06-24 2017-12-28 Ohio University Glucose transport inhibitors and methods of using same
RU2662153C1 (ru) * 2017-04-20 2018-07-24 Общество С Ограниченной Ответственностью "Дермавитал Групп" Гибридные эфиры на основе производных тиазолидин-2,4-диона и азолов (1н-1,3-имидазола и 1н-1,3,4-триазола) и их применение
RU2690161C1 (ru) * 2018-06-28 2019-05-31 Общество С Ограниченной Ответственностью "Дермавитал Групп" 3,5-Замещенные производные тиазолидин-2,4-диона, обладающие противомикробной активностью
RU2703997C1 (ru) * 2018-12-13 2019-10-23 Общество с ограниченной ответственностью "Л-Био" Гибридные амиды на основе триазола и тиазолидина, обладающие антимикробной активностью
CN112521382A (zh) * 2020-12-14 2021-03-19 西南大学 芦荟大黄素噻唑烷二酮类化合物及其制备方法和应用
WO2024258316A1 (ru) * 2023-06-16 2024-12-19 Общество с ограниченной ответственностью "Л-Био" Новые потенциальные противогрибковые средства на основе тиазолидин-2,4-диона и триазола

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS6156175A (ja) * 1984-08-24 1986-03-20 Yamanouchi Pharmaceut Co Ltd ロダニン誘導体およびその製造法
EP0915090A1 (en) * 1992-09-10 1999-05-12 Eli Lilly And Company Compounds useful as hypoglycemic agents and for treating Alzheimer's disease
DE4318550A1 (de) * 1993-06-04 1994-12-08 Boehringer Mannheim Gmbh Aryliden-4-oxo-2-thioxo-3- thiazolidincarbonsäuren, Verfahren zu ihrer Herstellung und diese Verbindungen enthaltende Arzneimittel
JPH08109174A (ja) * 1994-10-07 1996-04-30 Torii Yakuhin Kk チアゾリジン−２−オン誘導体
JPH08109175A (ja) * 1994-10-07 1996-04-30 Torii Yakuhin Kk チアゾリジン−２−オンエステル誘導体
AU6331099A (en) * 1998-09-30 2000-04-17 Roche Diagnostics Gmbh Thiazolidine derivatives for the treatment and prevention of metabolic bone disorders
AU6330799A (en) * 1998-09-30 2000-04-17 Roche Diagnostics Gmbh Rhodanine carboxylic acid derivatives for the treatment and prevention of metabolic bone disorders
US6506755B2 (en) * 2000-02-03 2003-01-14 Hoffmann-La Roche Inc. Thiazolidinecarboxyl acids

Also Published As

Publication number Publication date
JP2004507501A (ja) 2004-03-11
AU2001284190A1 (en) 2002-03-13
DE60127845T2 (de) 2007-12-20
GB0021421D0 (en) 2000-10-18
WO2002017915A1 (en) 2002-03-07
US20040006112A1 (en) 2004-01-08
ES2282283T3 (es) 2007-10-16
EP1313471B1 (en) 2007-04-11
US7105554B2 (en) 2006-09-12
EP1313471A1 (en) 2003-05-28
DE60127845D1 (de) 2007-05-24

Similar Documents

Publication Publication Date Title
ATE359073T1 (de) Benzylidenthiazolidindione und ihre verwendung als antimykotische mittel
DK1377593T3 (da) 2-Amino-propanolderivater
DE69910831D1 (de) Epothilonderivate und ihre verwendung als antitumormittel
DE60012188D1 (de) Fungizide
MXPA05010652A (es) Pirazoles sustituidos.
ATE469892T1 (de) Substituierte 1h-dihydropyrazole, ihre herstellung und verwendung
SE0004245D0 (sv) Novel compounds and their use
BR0213140A (pt) Fungicidas de pirazol-pirimidina
GEP20074198B (en) N-aryl-2-oxazolidinone-5-carboxamides and their derivates and their use as antibacterials
IS4425A (is) Arylþíósambönd sem varnarefni gegn bakteríum og veirum
TW200510405A (en) Bridged n-arylsulfonylpiperidines as gamma-secretase inhibitors
EA200301100A1 (ru) Новые фталазиноны
DE69821530D1 (de) Dihydrobenzifurane
ATE245642T1 (de) Benzamide mit tetrahydrofuranyloxy-substituenten als inhibitoren der phosphodiesterase 4
ATE399168T1 (de) Imidazopyridin-derivate und ihre verwendung als induzierbare no-synthase inhibitoren
TR200201128T2 (tr) PDE4 inhibitörleri olarak tetrahidrotiyopiranfitalazinon türevleri.
MXPA05010651A (es) Compuestos de pirazol.
DE60202669D1 (de) 6-phenylbenzonaphthyidine
SE9903290D0 (sv) Novel compounds
MXPA05010650A (es) Pirazoles sustituidos.
DE602004008633D1 (de) Siliziumverbindungen und deren verwendung
ATE266026T1 (de) Benzofurancarboxamide und deren therapeutische verwendung
CA2206125A1 (en) N-substituted hydrazinophenylsulphonylureas, as herbicides and plant growth regulators
BRPI0412360A (pt) compostos de organossilìcio e seu uso
ATE401329T1 (de) Neue antivirale makrocyclische derivate und metallkomplexe, in die verbrückte makrocyclen eingebaut sind

Legal Events

Date Code Title Description
RER Ceased as to paragraph 5 lit. 3 law introducing patent treaties