ATE359073T1 - Benzylidenthiazolidindione und ihre verwendung als antimykotische mittel - Google Patents

Benzylidenthiazolidindione und ihre verwendung als antimykotische mittel

Info

Publication number
ATE359073T1
ATE359073T1 AT01963157T AT01963157T ATE359073T1 AT E359073 T1 ATE359073 T1 AT E359073T1 AT 01963157 T AT01963157 T AT 01963157T AT 01963157 T AT01963157 T AT 01963157T AT E359073 T1 ATE359073 T1 AT E359073T1
Authority
AT
Austria
Prior art keywords
sub
benzylidenthiazolidindiones
antifungal agents
hydrogen
specific substituents
Prior art date
Application number
AT01963157T
Other languages
German (de)
English (en)
Inventor
Michael Glen Orchard
Judi Charlotte Neuss
Carl Maurice Swedler Galley
Original Assignee
Ucb Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ucb Sa filed Critical Ucb Sa
Application granted granted Critical
Publication of ATE359073T1 publication Critical patent/ATE359073T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10—Antimycotics
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Communicable Diseases (AREA)
  • Animal Behavior & Ethology (AREA)
  • Oncology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
AT01963157T 2000-08-31 2001-08-30 Benzylidenthiazolidindione und ihre verwendung als antimykotische mittel ATE359073T1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GBGB0021421.3A GB0021421D0 (en) 2000-08-31 2000-08-31 Compounds

Publications (1)

Publication Number Publication Date
ATE359073T1 true ATE359073T1 (de) 2007-05-15

Family

ID=9898616

Family Applications (1)

Application Number Title Priority Date Filing Date
AT01963157T ATE359073T1 (de) 2000-08-31 2001-08-30 Benzylidenthiazolidindione und ihre verwendung als antimykotische mittel

Country Status (9)

Country Link
US (1) US7105554B2 (enExample)
EP (1) EP1313471B1 (enExample)
JP (1) JP2004507501A (enExample)
AT (1) ATE359073T1 (enExample)
AU (1) AU2001284190A1 (enExample)
DE (1) DE60127845T2 (enExample)
ES (1) ES2282283T3 (enExample)
GB (1) GB0021421D0 (enExample)
WO (1) WO2002017915A1 (enExample)

Families Citing this family (23)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2003205907A1 (en) * 2002-02-23 2003-09-09 Oxford Glycosciences (Uk) Ltd Thiazolidine antifungal agents
GB0204252D0 (en) * 2002-02-23 2002-04-10 Oxford Glycosciences Uk Ltd Novel compounds
PL1730103T3 (pl) 2004-03-23 2010-10-29 Pfizer Pochodne formamidu użyteczne jako adrenoreceptor
AU2006316838B2 (en) 2005-11-15 2012-04-12 Glycofi, Inc Production of glycoproteins with reduced O-glycosylation
US7731106B2 (en) * 2006-01-04 2010-06-08 Nano Mist International, Llc Air driven delivery system for sprayable media
US8637435B2 (en) * 2007-11-16 2014-01-28 Merck Sharp & Dohme Corp. Eukaryotic cell display systems
EP2263089B1 (en) * 2008-03-03 2015-01-28 GlycoFi, Inc. Surface display of recombinant proteins in lower eukaryotes
CN102036974B (zh) * 2008-05-20 2014-07-23 默沙东公司 利用甘露糖基转移酶抑制剂有效生产异源蛋白质
US8067339B2 (en) 2008-07-09 2011-11-29 Merck Sharp & Dohme Corp. Surface display of whole antibodies in eukaryotes
MX2011001706A (es) 2008-08-12 2011-03-24 Glycofi Inc Vectores mejorados y cepas de levadura para produccion de proteina: sobreexpresion de ca2+ atpasa.
JP2014518608A (ja) 2011-02-25 2014-08-07 メルク・シャープ・アンド・ドーム・コーポレーション 修飾ｏ−グリコシル化を有するタンパク質の製造のための酵母株
AU2012291133A1 (en) * 2011-07-29 2014-02-20 Taisho Pharmaceutical Co., Ltd. Amidine compound or salt thereof
WO2014024897A1 (ja) * 2012-08-06 2014-02-13 Ｍｅｉｊｉ Ｓｅｉｋａファルマ株式会社 チアゾリジンジオンおよびピロリジンジオン誘導体、並びにそれらを有効成分としてなる殺菌剤
WO2014062811A2 (en) * 2012-10-16 2014-04-24 New York University METHOD OF TREATING CANCER WITH MODULATORS OF SCFSkp2
WO2015001049A1 (en) 2013-07-04 2015-01-08 Novartis Ag O-mannosyltransferase deficient filamentous fungal cells and methods of use thereof
AU2015293949B2 (en) 2014-07-21 2019-07-25 Teknologian Tutkimuskeskus Vtt Oy Production of glycoproteins with mammalian-like N-glycans in filamentous fungi
KR20190017981A (ko) * 2016-06-14 2019-02-20 벌시테크 리미티드 항균성 화합물 및 이의 사용 방법
US10647654B2 (en) 2016-06-24 2020-05-12 Ohio University Glucose transport inhibitors and methods of using same
RU2662153C1 (ru) * 2017-04-20 2018-07-24 Общество С Ограниченной Ответственностью "Дермавитал Групп" Гибридные эфиры на основе производных тиазолидин-2,4-диона и азолов (1н-1,3-имидазола и 1н-1,3,4-триазола) и их применение
RU2690161C1 (ru) * 2018-06-28 2019-05-31 Общество С Ограниченной Ответственностью "Дермавитал Групп" 3,5-Замещенные производные тиазолидин-2,4-диона, обладающие противомикробной активностью
RU2703997C1 (ru) * 2018-12-13 2019-10-23 Общество с ограниченной ответственностью "Л-Био" Гибридные амиды на основе триазола и тиазолидина, обладающие антимикробной активностью
CN112521382A (zh) * 2020-12-14 2021-03-19 西南大学 芦荟大黄素噻唑烷二酮类化合物及其制备方法和应用
WO2024258316A1 (ru) * 2023-06-16 2024-12-19 Общество с ограниченной ответственностью "Л-Био" Новые потенциальные противогрибковые средства на основе тиазолидин-2,4-диона и триазола

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS6156175A (ja) * 1984-08-24 1986-03-20 Yamanouchi Pharmaceut Co Ltd ロダニン誘導体およびその製造法
NZ248573A (en) * 1992-09-10 1996-02-27 Lilly Co Eli 5-arylmethyl (and methylidene) thiazolidin-4-one derivatives; their preparation and pharmaceutical compositions
DE4318550A1 (de) * 1993-06-04 1994-12-08 Boehringer Mannheim Gmbh Aryliden-4-oxo-2-thioxo-3- thiazolidincarbonsäuren, Verfahren zu ihrer Herstellung und diese Verbindungen enthaltende Arzneimittel
JPH08109175A (ja) * 1994-10-07 1996-04-30 Torii Yakuhin Kk チアゾリジン−２−オンエステル誘導体
JPH08109174A (ja) * 1994-10-07 1996-04-30 Torii Yakuhin Kk チアゾリジン−２−オン誘導体
US6673816B1 (en) * 1998-09-30 2004-01-06 Angelika Esswein Rhodanine carboxylic acid derivatives for the treatment and prevention of metabolic bone disorders
AU6331099A (en) * 1998-09-30 2000-04-17 Roche Diagnostics Gmbh Thiazolidine derivatives for the treatment and prevention of metabolic bone disorders
US6506755B2 (en) * 2000-02-03 2003-01-14 Hoffmann-La Roche Inc. Thiazolidinecarboxyl acids

Also Published As

Publication number Publication date
WO2002017915A1 (en) 2002-03-07
EP1313471A1 (en) 2003-05-28
EP1313471B1 (en) 2007-04-11
AU2001284190A1 (en) 2002-03-13
JP2004507501A (ja) 2004-03-11
US7105554B2 (en) 2006-09-12
ES2282283T3 (es) 2007-10-16
GB0021421D0 (en) 2000-10-18
DE60127845T2 (de) 2007-12-20
US20040006112A1 (en) 2004-01-08
DE60127845D1 (de) 2007-05-24

Similar Documents

Publication Publication Date Title
ATE359073T1 (de) Benzylidenthiazolidindione und ihre verwendung als antimykotische mittel
DK1377593T3 (da) 2-Amino-propanolderivater
DE69910831D1 (de) Epothilonderivate und ihre verwendung als antitumormittel
DE60012188D1 (de) Fungizide
MXPA05010652A (es) Pirazoles sustituidos.
DE60236600D1 (de) Substituierte 1h-dihydropyrazole, ihre herstellung und verwendung
SE0004245D0 (sv) Novel compounds and their use
BR0213140A (pt) Fungicidas de pirazol-pirimidina
GEP20074198B (en) N-aryl-2-oxazolidinone-5-carboxamides and their derivates and their use as antibacterials
IS4425A (is) Arylþíósambönd sem varnarefni gegn bakteríum og veirum
TW200510405A (en) Bridged n-arylsulfonylpiperidines as gamma-secretase inhibitors
EA200301100A1 (ru) Новые фталазиноны
ATE258930T1 (de) Dihydrobenzifurane
ATE245642T1 (de) Benzamide mit tetrahydrofuranyloxy-substituenten als inhibitoren der phosphodiesterase 4
ATE399168T1 (de) Imidazopyridin-derivate und ihre verwendung als induzierbare no-synthase inhibitoren
NO20062629L (no) Oksazolderivater av tetrackliner
MXPA05010651A (es) Compuestos de pirazol.
ATE287403T1 (de) 6-phenylbenzonaphthyidine
SE9903290D0 (sv) Novel compounds
MXPA05010650A (es) Pirazoles sustituidos.
DE602004008633D1 (de) Siliziumverbindungen und deren verwendung
ATE266026T1 (de) Benzofurancarboxamide und deren therapeutische verwendung
CA2206125A1 (en) N-substituted hydrazinophenylsulphonylureas, as herbicides and plant growth regulators
BRPI0412360A (pt) compostos de organossilìcio e seu uso
ATE401329T1 (de) Neue antivirale makrocyclische derivate und metallkomplexe, in die verbrückte makrocyclen eingebaut sind

Legal Events

Date Code Title Description
RER Ceased as to paragraph 5 lit. 3 law introducing patent treaties