FR2949468B1 - Derives de 2-pyridin-2-yl-pyrazol-3(2h)-one, leur preparation et leur application en therapeutique - Google Patents
Derives de 2-pyridin-2-yl-pyrazol-3(2h)-one, leur preparation et leur application en therapeutiqueInfo
- Publication number
- FR2949468B1 FR2949468B1 FR0904091A FR0904091A FR2949468B1 FR 2949468 B1 FR2949468 B1 FR 2949468B1 FR 0904091 A FR0904091 A FR 0904091A FR 0904091 A FR0904091 A FR 0904091A FR 2949468 B1 FR2949468 B1 FR 2949468B1
- Authority
- FR
- France
- Prior art keywords
- pyrazol
- pyridin
- derivatives
- preparation
- therapeutic use
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Fee Related
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Engineering & Computer Science (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Priority Applications (36)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR0904091A FR2949468B1 (fr) | 2009-08-28 | 2009-08-28 | Derives de 2-pyridin-2-yl-pyrazol-3(2h)-one, leur preparation et leur application en therapeutique |
MA34029A MA32978B1 (fr) | 2008-12-29 | 2009-12-24 | Derives de 2-pyridin-2-yl-pyrazol-3(2h)-one, leur preparation et leur application en therapeutique |
SI200931025T SI2382215T1 (sl) | 2008-12-29 | 2009-12-24 | Derivati 2-piridin-2-il-pirazol-3(2H)-ona, njihova priprava in njihova terapevtska uporaba |
PE2011001291A PE20120338A1 (es) | 2008-12-29 | 2009-12-24 | Derivados de 2-piridin-2-il-pirazol-3(2h)-ona, su preparacion y su aplicacion en terapeutica |
NZ593797A NZ593797A (en) | 2008-12-29 | 2009-12-24 | Derivatives of 2-pyridin-2-yl-pyrazol-3(2h)-one, preparation and therapeutic use thereof |
PL09805790T PL2382215T3 (pl) | 2008-12-29 | 2009-12-24 | Pochodne 2-pirydyny-2-ylo-pirazol-3(2H)-onu, ich wytwarzanie i zastosowanie terapeutyczne |
KR1020117017677A KR101630475B1 (ko) | 2008-12-29 | 2009-12-24 | 2-피리딘-2-일-피라졸-3(2h)-온의 유도체, 그의 제조법 및 치료 용도 |
PT98057904T PT2382215E (pt) | 2008-12-29 | 2009-12-24 | Derivados de 2-piridin-2-il-pirazol-3(2h)-ona, sua preparação e sua aplicação terapêutica |
EA201170900A EA019774B1 (ru) | 2008-12-29 | 2009-12-24 | Производные 2-пиридин-2-ил-пиразол-3(2h)-она, их получение и применение в терапии |
CA2748413A CA2748413A1 (fr) | 2008-12-29 | 2009-12-24 | Derives de 2-pyridin-2-yl-pyrazol-3(2h)-one, leur preparation et leur application en therapeutique |
MX2011007061A MX2011007061A (es) | 2008-12-29 | 2009-12-24 | Derivados de 2 piridin- 2-il-pirazol-3 (2h)-ona, su preparacion y aplicacion terapeutica. |
DK09805790.4T DK2382215T3 (da) | 2008-12-29 | 2009-12-24 | Derivater af 2-pyridin-2-yl-pyrazol-3(2h)-on, fremstilling og terapeutisk anvendelse heraf |
PCT/FR2009/052692 WO2010076525A1 (fr) | 2008-12-29 | 2009-12-24 | Dérivés de 2-pyridin-2-yl-pyrazol-3(2h)-one, leur préparation et leur application en thérapeutique |
AU2009334570A AU2009334570B2 (en) | 2008-12-29 | 2009-12-24 | Derivatives of 2-pyridin-2-yl-pyrazol-3(2h)-one, preparation and therapeutic use thereof |
JP2011542887A JP5865704B2 (ja) | 2008-12-29 | 2009-12-24 | 2−ピリジン−2−イル−ピラゾール−3(2h)−オンの誘導体、この調製および治療的使用 |
BRPI0923875-1A BRPI0923875A2 (pt) | 2008-12-29 | 2009-12-24 | Derivados de 2-piridin-2-il-pirazol-3 (2h)-ona, o respectivo preparo e a respectiva aplicação terapêutica. |
SG2011047529A SG172422A1 (en) | 2008-12-29 | 2009-12-24 | Derivatives of 2-pyridin-2-yl-pyrazol-3(2h)-one, preparation and therapeutic use thereof |
EP09805790.4A EP2382215B1 (fr) | 2008-12-29 | 2009-12-24 | Dérivés de 2-pyridin-2-yl-pyrazol-3(2h)-one, leur préparation et leur application en thérapeutique |
MYPI2011003011A MY155244A (en) | 2008-12-29 | 2009-12-24 | Derivatives of 2-pyridin-2-yl-pyrazol-3(2h)-one, preparation and therapeutic use thereof |
ES09805790.4T ES2511917T3 (es) | 2008-12-29 | 2009-12-24 | Derivados de 2-piridin-2-il-pirazol-3(2H)-ona, su preparación y su aplicación en terapéutica |
CN200980157589.3A CN102333776B (zh) | 2008-12-29 | 2009-12-24 | 2-吡啶-2-基-吡唑-3(2h)-酮的衍生物、其制备和治疗用途 |
TW098145333A TWI441828B (zh) | 2008-12-29 | 2009-12-28 | 2-吡啶-2-基-吡唑-3(2h)-酮衍生物、其製備及治療用途 |
PA20098856101A PA8856101A1 (es) | 2008-12-29 | 2009-12-28 | Derivados de 2-piridin-2-il-pirazol-3(2h)-ona, su preparcion y su aplicacion en terapeutica |
ARP090105127A AR074916A1 (es) | 2008-12-29 | 2009-12-28 | Derivados de 2-piridin-2-il-pirazol-3(2h)-ona, su preparacion, composiciones farmaceuticas y su uso en enfermedades cardiovasculares. |
TN2011000308A TN2011000308A1 (fr) | 2008-12-29 | 2011-06-17 | Derives de 2-pyridin-2-yl-pyrazol-3(2h)-one, leur preparation et leur application en therapeutique |
CR20110360A CR20110360A (es) | 2008-12-29 | 2011-06-23 | Derivados de 2-piridin-2-il-pirazol-3-(2h)-ona, su preparacion y su aplicacion en terapeutica |
EC2011011164A ECSP11011164A (es) | 2008-12-29 | 2011-06-27 | Derivados de 2-piridin-2-il-pirazol-3(2h)-ona, su preparación y su aplicación en terapéutica |
IL213790A IL213790A (en) | 2008-12-29 | 2011-06-27 | 2-Pyridine-2-Ill-Pyrazole-3 (2 h) History - On, Preparation and Medical Use |
NI201100132A NI201100132A (es) | 2008-12-29 | 2011-06-28 | Derivados de 2 - piridin - 2 - il - pirazol - 3 (2h) - ona, su preparación y su aplicación en terapéutica. |
ZA2011/04785A ZA201104785B (en) | 2008-12-29 | 2011-06-28 | Derivatives of 2-pyridin-2-yl-pyrazol-3(2h)-one,preparation and therapeutic use thereof |
CO11081313A CO6400145A2 (es) | 2008-12-29 | 2011-06-29 | Derivados de 2-piridin-2-il pirazol-3(2h) -ona, su preparción y su aplicación terapeútica |
US13/172,321 US8697731B2 (en) | 2008-12-29 | 2011-06-29 | Derivatives of 2-pyridin-2-yl-pyrazol-3(2H)-one, preparation and therapeutic use thereof |
HK12104300.3A HK1163679A1 (en) | 2008-12-29 | 2012-05-02 | Derivatives of 2-pyridin-2-yl-pyrazol-3(2h)-one, preparation and therapeutic use thereof 2--2---3(2h)- |
US14/200,698 US9359329B2 (en) | 2008-12-29 | 2014-03-07 | Derivatives of 2-pyridin-2-yl-pyrazol-3(2H)-one, preparation and therapeutic use thereof |
CY20141100849T CY1115635T1 (el) | 2008-12-29 | 2014-10-16 | Παραγωγα 2-πυριδιν-2-υλο-πυραζολ-3(2η)-ονης, η παρασκευη τους και η εφαρμογη τους στη θεραπευτικη |
SM201400157T SMT201400157B (it) | 2008-12-29 | 2014-10-29 | Derivati di 2-piridin-2-il-pirazol-3(2H)-one, loropreparazione e loro uso terapeutico |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR0904091A FR2949468B1 (fr) | 2009-08-28 | 2009-08-28 | Derives de 2-pyridin-2-yl-pyrazol-3(2h)-one, leur preparation et leur application en therapeutique |
Publications (2)
Publication Number | Publication Date |
---|---|
FR2949468A1 FR2949468A1 (fr) | 2011-03-04 |
FR2949468B1 true FR2949468B1 (fr) | 2011-09-30 |
Family
ID=41820704
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
FR0904091A Expired - Fee Related FR2949468B1 (fr) | 2008-12-29 | 2009-08-28 | Derives de 2-pyridin-2-yl-pyrazol-3(2h)-one, leur preparation et leur application en therapeutique |
Country Status (1)
Country | Link |
---|---|
FR (1) | FR2949468B1 (fr) |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5750088A (en) * | 1993-03-30 | 1998-05-12 | The Dupont Merck Pharmaceutical Company | Stable hydrazones linked to a peptide moiety as reagents for the preparation of radiopharmaceuticals |
EP2074128B1 (fr) * | 2006-10-16 | 2013-08-14 | Medicis Pharmaceutical Corporation | Pyrazolyl thienopyridines therapeutiques |
WO2008137060A1 (fr) * | 2007-05-04 | 2008-11-13 | Amgen Inc. | Dérivés de la thienopyridine et de la thiazolopyridine qui inhibent l'activité prolyle hydroxylase |
-
2009
- 2009-08-28 FR FR0904091A patent/FR2949468B1/fr not_active Expired - Fee Related
Also Published As
Publication number | Publication date |
---|---|
FR2949468A1 (fr) | 2011-03-04 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
FR2949470B1 (fr) | Derives anticancereux, leur preparation et leur application therapeutique | |
FR2945534B1 (fr) | DERIVES DE CYCLOPENTAL[c]PYRROLE-2-CARBOXYLATES, LEUR PREPARATION ET LEUR APPLICATION EN THERAPEUTIQUE | |
FR2953520B1 (fr) | Derives de diphenyl-pyrazolopyridines, leur preparation et leur application en therapeutique | |
FR2933700B1 (fr) | Derives de pyridino-pyridinones, leur preparation et leur application en therapeutique | |
FR2915198B1 (fr) | Derives de triazolopyridine-carboxamides et triazolopyridine -carboxamides, leur preparation et leur application en therapeutique. | |
FR2963007B1 (fr) | Derives anticancereux, leur preparation et leur application therapeutique | |
FR2952934B1 (fr) | Derives de pyridino-pyridinones, leur preparation et leur application en therapeutique | |
FR2943669B1 (fr) | Derives de nicotinamide,leur preparation et leur application en therapeutique | |
FR2915199B1 (fr) | Derives de triazolopyridine-carboxamides et triazolopyrimidine-carboxamides, leur preparation et leur application en therapeutique. | |
FR2941696B1 (fr) | Derives d'azaspiranyl-alkylcarbamates d'heterocycles a 5 chainons, leur preparation et leur application en therapeutique | |
FR2948939B1 (fr) | Derives de 2h pyridazin-3-ones, leur preparation et leur application en therapeutique humaine | |
FR2945533B1 (fr) | Derives de cyclopenta°c!pyrrolyl-alkylcarbamates d'heterocycles a 5 chainons, leur preparation et leur application en therapeutique | |
IL213790A (en) | 2-Pyridine-2-Ill-Pyrazole-3 (2 h) History - On, Preparation and Medical Use | |
FR2917413B1 (fr) | Derives de 7-alkynyl-1,8-naphthyridones, leur preparation et leur application en therapeutique | |
FR2927625B1 (fr) | Nouveaux derives de 3-aminoalkyl-1,3-dihydro-2h-indol-2-one, leur preparation et leur application en therapeutique | |
FR2947546B1 (fr) | Derives de pyrazoles, leur preparation et leur application en therapeutique | |
FR2940284B1 (fr) | Derives de 6-cycloamino-2,3-di-pyridinyl-imidazo°1,2-b!- pyridazine,leur preparation et leur application en therapeutique | |
FR2963005B1 (fr) | Derives d'oxadiazoles et de pyridazines, leur preparation et leur application en therapeutique | |
FR2925901B1 (fr) | DERIVES DE N-HETEROCYCLIQUE-IMIDAZO°1,2-a!PYRIDINE-2- CARBOXAMIDES, LEUR PREPARATION ET LEUR APPLICATION EN THERAPEUTIQUE | |
FR2932481B1 (fr) | Derives de 4-{2-°4-phenyl-3,6-dihydro-2h-pyridin-1-yl!-2- oxo-alkyl}-1-piperazin-2-one, leur preparation et leur application en therapeutique. | |
FR2911605B1 (fr) | Derives de pyrrolopyridine-2-carbowamides, leur preparation et leur application en therapeutique | |
FR2919610B1 (fr) | Derives de n-heteroaryl-carboxamides tricycliques,leur preparation et leur application en therapeutique | |
FR2934594B1 (fr) | Derives de thiophene-2-carboxamide, leur preparation et leur application en therapeutique. | |
FR2925903B1 (fr) | DERIVES 6-HETEROCYCLIQUE-IMIDAZO°1,2-a!PYRIDINE-2- CARBOXAMIDES, LEUR PREPARATION ET LEUR APPLICATION EN THERAPEUTIQUE | |
FR2930939B1 (fr) | Derives de pyrrole, leur preparation et leur application en therapeutique |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
PLFP | Fee payment |
Year of fee payment: 7 |
|
ST | Notification of lapse |
Effective date: 20170428 |