FR2658822A1 - N-cycloalkylalkylamines, leur procede de preparation, leur utilisation comme medicament et leurs intermediaires de synthese. - Google Patents

N-cycloalkylalkylamines, leur procede de preparation, leur utilisation comme medicament et leurs intermediaires de synthese. Download PDF

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Publication number
FR2658822A1
FR2658822A1 FR9002494A FR9002494A FR2658822A1 FR 2658822 A1 FR2658822 A1 FR 2658822A1 FR 9002494 A FR9002494 A FR 9002494A FR 9002494 A FR9002494 A FR 9002494A FR 2658822 A1 FR2658822 A1 FR 2658822A1
Authority
FR
France
Prior art keywords
sep
cycloalkylalkylamines
compounds
phenyl
compound
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
FR9002494A
Other languages
English (en)
French (fr)
Other versions
FR2658822B1 (enrdf_load_stackoverflow
Inventor
Gilbert Aubard
Alain Calvet
Jean-Pierre Defaux
Claude-Jean Gouret
Agnes Grouhel
James Hudspeth
Henri Jacobelli
Jean-Louis Junien
Xavier Pascaud
Francois Roman
Lin Yuan
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Jouveinal SA
Original Assignee
Jouveinal SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority to FR9002494A priority Critical patent/FR2658822A1/fr
Application filed by Jouveinal SA filed Critical Jouveinal SA
Priority to HU9803012A priority patent/HU217873B/hu
Priority to CA002037114A priority patent/CA2037114C/en
Priority to KR1019910003016A priority patent/KR0166084B1/ko
Priority to IL9735491A priority patent/IL97354A/en
Priority to AU71340/91A priority patent/AU633695B2/en
Priority to DK91400497.3T priority patent/DK0445013T3/da
Priority to AT91400497T priority patent/ATE106879T1/de
Priority to EP91400497A priority patent/EP0445013B1/fr
Priority to HU91625A priority patent/HU215430B/hu
Priority to ES91400497T priority patent/ES2054452T3/es
Priority to DE69102309T priority patent/DE69102309T2/de
Priority to FI910894A priority patent/FI97384C/fi
Priority to IE62091A priority patent/IE66180B1/en
Priority to PT96885A priority patent/PT96885B/pt
Priority to NZ237224A priority patent/NZ237224A/en
Priority to JP3031059A priority patent/JP2899429B2/ja
Publication of FR2658822A1 publication Critical patent/FR2658822A1/fr
Application granted granted Critical
Publication of FR2658822B1 publication Critical patent/FR2658822B1/fr
Granted legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/06—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to the ring carbon atoms
    • C07D333/08—Hydrogen atoms or radicals containing only hydrogen and carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/02—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings
    • C07D307/34—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D307/38—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D307/52—Radicals substituted by nitrogen atoms not forming part of a nitro radical
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/06—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to the ring carbon atoms
    • C07D333/14—Radicals substituted by singly bound hetero atoms other than halogen
    • C07D333/20—Radicals substituted by singly bound hetero atoms other than halogen by nitrogen atoms

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
FR9002494A 1990-02-26 1990-02-28 N-cycloalkylalkylamines, leur procede de preparation, leur utilisation comme medicament et leurs intermediaires de synthese. Granted FR2658822A1 (fr)

Priority Applications (17)

Application Number Priority Date Filing Date Title
FR9002494A FR2658822A1 (fr) 1990-02-28 1990-02-28 N-cycloalkylalkylamines, leur procede de preparation, leur utilisation comme medicament et leurs intermediaires de synthese.
ES91400497T ES2054452T3 (es) 1990-02-26 1991-02-25 N-cicloalquilalquilaminas, su procedimiento de preparacion, su utilizacion como medicamento y sus intermedios de sintesis.
KR1019910003016A KR0166084B1 (ko) 1990-02-26 1991-02-25 N-시클로알킬알킬아민, 그의 제조 방법, 약제로서 그의 용도 및 그의 합성 중간체
IL9735491A IL97354A (en) 1990-02-26 1991-02-25 Furyl or thienyl-n-cycloalkylalkylamines and pharmaceutical compositions containing them
AU71340/91A AU633695B2 (en) 1990-02-26 1991-02-25 N-cycloalkylalkylamines, their process of preparation, their use as a medicament and their synthesis intermediates
DK91400497.3T DK0445013T3 (da) 1990-02-26 1991-02-25 N-Cycloalkylalkylaminer, fremgangsmåde til fremstilling deraf, deres anvendelse som lægemiddel og deres syntese-mellemprodukter
AT91400497T ATE106879T1 (de) 1990-02-26 1991-02-25 N-cycloalkyl-alkylamine, verfahren zu ihrer herstellung, ihre verwendung als arzneimittel und zwischenprodukte zu ihrer synthese.
EP91400497A EP0445013B1 (fr) 1990-02-26 1991-02-25 N-Cycloalkylalkylamines, leur procédé de préparation, leur utilisation comme médicament et leurs intermédiaires de synthèse
HU9803012A HU217873B (hu) 1990-02-26 1991-02-25 N-cikloalkil-amin-származékok, valamint hatóanyagként e vegyületeket tartalmazó gyógyászati készítmények
CA002037114A CA2037114C (en) 1990-02-26 1991-02-25 N-cycloalkylalkylamines, their process of preparation, their use as medication and their synthetic intermediates
DE69102309T DE69102309T2 (de) 1990-02-26 1991-02-25 N-cycloalkyl-Alkylamine, Verfahren zu ihrer Herstellung, ihre Verwendung als Arzneimittel und Zwischenprodukte zu ihrer Synthese.
FI910894A FI97384C (fi) 1990-02-26 1991-02-25 Menetelmä terapeuttisesti käyttökelpoisten N-sykloalkyylialkyyliamiinien valmistamiseksi
IE62091A IE66180B1 (en) 1990-02-26 1991-02-25 N-Cycloalkylalkylamines their process of preparation their use as a medicament and their synthesis intermediates
HU91625A HU215430B (hu) 1990-02-26 1991-02-25 Eljárás N-cikloalkil-alkil-amin-származékok, valamint hatóanyagként e vegyületeket tartalmazó gyógyászati készítmények előállítására
PT96885A PT96885B (pt) 1990-02-26 1991-02-26 Processo para a preparacao de n-cicloalquilalquilaminas e de composicoes farmaceuticas que os contem
NZ237224A NZ237224A (en) 1990-02-26 1991-02-26 N-cycloalkylalkylamine derivatives and pharmaceutical formulations thereof
JP3031059A JP2899429B2 (ja) 1990-02-26 1991-02-26 Ｎ−シクロアルキルアルキルアミン、その製造法、薬物としてのその使用、ならびにその合成中間体

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR9002494A FR2658822A1 (fr) 1990-02-28 1990-02-28 N-cycloalkylalkylamines, leur procede de preparation, leur utilisation comme medicament et leurs intermediaires de synthese.

Publications (2)

Publication Number Publication Date
FR2658822A1 true FR2658822A1 (fr) 1991-08-30
FR2658822B1 FR2658822B1 (enrdf_load_stackoverflow) 1994-08-19

Family

ID=9394221

Family Applications (1)

Application Number Title Priority Date Filing Date
FR9002494A Granted FR2658822A1 (fr) 1990-02-26 1990-02-28 N-cycloalkylalkylamines, leur procede de preparation, leur utilisation comme medicament et leurs intermediaires de synthese.

Country Status (2)

Country Link
KR (1) KR0166084B1 (enrdf_load_stackoverflow)
FR (1) FR2658822A1 (enrdf_load_stackoverflow)

Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0297782A1 (en) * 1987-06-30 1989-01-04 Tanabe Seiyaku Co., Ltd. A thiophene derivative and process for preparing the same
EP0298703A1 (en) * 1987-07-09 1989-01-11 Tanabe Seiyaku Co., Ltd. A thiophene derivative and process for preparing the same

Patent Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0297782A1 (en) * 1987-06-30 1989-01-04 Tanabe Seiyaku Co., Ltd. A thiophene derivative and process for preparing the same
EP0298703A1 (en) * 1987-07-09 1989-01-11 Tanabe Seiyaku Co., Ltd. A thiophene derivative and process for preparing the same

Also Published As

Publication number Publication date
KR910021396A (ko) 1991-12-20
KR0166084B1 (ko) 1999-01-15
FR2658822B1 (enrdf_load_stackoverflow) 1994-08-19

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