FR2509311A1 - Derives de beta-lactame, les compositions pharmaceutiques les contenant et leur procede de preparation - Google Patents

Derives de beta-lactame, les compositions pharmaceutiques les contenant et leur procede de preparation Download PDF

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Publication number
FR2509311A1
FR2509311A1 FR8207659A FR8207659A FR2509311A1 FR 2509311 A1 FR2509311 A1 FR 2509311A1 FR 8207659 A FR8207659 A FR 8207659A FR 8207659 A FR8207659 A FR 8207659A FR 2509311 A1 FR2509311 A1 FR 2509311A1
Authority
FR
France
Prior art keywords
group
compound
general formula
alkyl
ester
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
FR8207659A
Other languages
English (en)
French (fr)
Inventor
Rezso Bognar
Csaba Jaszberenyi
Erzsebet Farkas
Maria Punyiczky
Ferenc Hernadi
Katalin Eke
Ilona Petrikovics
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Chinoin Private Co Ltd
Original Assignee
Chinoin Gyogyszer es Vegyeszeti Termekek Gyara Zrt
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Chinoin Gyogyszer es Vegyeszeti Termekek Gyara Zrt filed Critical Chinoin Gyogyszer es Vegyeszeti Termekek Gyara Zrt
Publication of FR2509311A1 publication Critical patent/FR2509311A1/fr
Withdrawn legal-status Critical Current

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14—Compounds having a nitrogen atom directly attached in position 7
    • C07D501/16—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
    • C07D501/20—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D499/21—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with a nitrogen atom directly attached in position 6 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
    • C07D499/44—Compounds with an amino radical acylated by carboxylic acids, attached in position 6
    • C07D499/48—Compounds with an amino radical acylated by carboxylic acids, attached in position 6 with a carbon chain, substituted by hetero atoms or by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, attached to the carboxamido radical
    • C07D499/58—Compounds with an amino radical acylated by carboxylic acids, attached in position 6 with a carbon chain, substituted by hetero atoms or by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, attached to the carboxamido radical substituted in alpha-position to the carboxamido radical
    • C07D499/64—Compounds with an amino radical acylated by carboxylic acids, attached in position 6 with a carbon chain, substituted by hetero atoms or by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, attached to the carboxamido radical substituted in alpha-position to the carboxamido radical by nitrogen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Cephalosporin Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
FR8207659A 1981-05-04 1982-05-03 Derives de beta-lactame, les compositions pharmaceutiques les contenant et leur procede de preparation Withdrawn FR2509311A1 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
HU115481 1981-05-04

Publications (1)

Publication Number Publication Date
FR2509311A1 true FR2509311A1 (fr) 1983-01-14

Family

ID=10953073

Family Applications (1)

Application Number Title Priority Date Filing Date
FR8207659A Withdrawn FR2509311A1 (fr) 1981-05-04 1982-05-03 Derives de beta-lactame, les compositions pharmaceutiques les contenant et leur procede de preparation

Country Status (17)

Country Link
JP (1) JPS5813590A (enrdf_load_stackoverflow)
AU (1) AU8321282A (enrdf_load_stackoverflow)
BE (1) BE893057A (enrdf_load_stackoverflow)
BG (1) BG37227A1 (enrdf_load_stackoverflow)
DE (1) DE3215941A1 (enrdf_load_stackoverflow)
DK (1) DK198282A (enrdf_load_stackoverflow)
ES (1) ES8307814A1 (enrdf_load_stackoverflow)
FI (1) FI821551A7 (enrdf_load_stackoverflow)
FR (1) FR2509311A1 (enrdf_load_stackoverflow)
GB (1) GB2101586A (enrdf_load_stackoverflow)
GR (1) GR78166B (enrdf_load_stackoverflow)
IL (1) IL65602A0 (enrdf_load_stackoverflow)
IT (1) IT1156467B (enrdf_load_stackoverflow)
NL (1) NL8201810A (enrdf_load_stackoverflow)
NO (1) NO821456L (enrdf_load_stackoverflow)
PL (1) PL236277A1 (enrdf_load_stackoverflow)
SE (1) SE8202674L (enrdf_load_stackoverflow)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3137376C2 (de) * 1981-09-19 1986-02-27 Degussa Ag, 6000 Frankfurt Verfahren zur Herstellung von 1,5-Alkylen-3-aryl-hydantoin-Derivaten
AU577105B2 (en) * 1985-04-02 1988-09-15 T.P.O. :Pharmachim: Acylaminic penicillin derivatives

Citations (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2285135A1 (fr) * 1974-09-20 1976-04-16 Squibb & Sons Inc 3-heterothio-7-ureido cephalosporines et leur procede de preparation
FR2319366A1 (fr) * 1975-07-30 1977-02-25 3-heterothio-7-thio-ureidocephalosporines
GB1476312A (en) * 1974-06-03 1977-06-10 Beecham Group Ltd Penicillins and cephalosporins
FR2346356A1 (fr) * 1976-03-30 1977-10-28 Squibb & Sons Inc Nouveaux derives de ((((2,4-dioxo-1-imidazolinyl) amino) carbonyl) amino) acetylcephalosporine
FR2370052A1 (fr) * 1976-11-06 1978-06-02 Merck Patent Gmbh Lactames utiles notamment comme medicaments et leur procede de preparation
GB1517098A (en) * 1975-08-29 1978-07-12 Toyama Chemical Co Ltd Process for producing penicillins and cephalosporins
EP0003814A2 (de) * 1978-02-25 1979-09-05 Dr. Karl Thomae GmbH Neue Penicilline, ihre Salze, Verfahren zu ihrer Herstellung und diese Verbindungen enthaltende Arzneimittel
EP0006532A1 (de) * 1978-06-28 1980-01-09 Dr. Karl Thomae GmbH Neue Lactame, Verfahren zu ihrer Herstellung und diese Verbindungen enthaltende Arzneimittel

Patent Citations (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1476312A (en) * 1974-06-03 1977-06-10 Beecham Group Ltd Penicillins and cephalosporins
FR2285135A1 (fr) * 1974-09-20 1976-04-16 Squibb & Sons Inc 3-heterothio-7-ureido cephalosporines et leur procede de preparation
FR2319366A1 (fr) * 1975-07-30 1977-02-25 3-heterothio-7-thio-ureidocephalosporines
GB1517098A (en) * 1975-08-29 1978-07-12 Toyama Chemical Co Ltd Process for producing penicillins and cephalosporins
FR2346356A1 (fr) * 1976-03-30 1977-10-28 Squibb & Sons Inc Nouveaux derives de ((((2,4-dioxo-1-imidazolinyl) amino) carbonyl) amino) acetylcephalosporine
FR2370052A1 (fr) * 1976-11-06 1978-06-02 Merck Patent Gmbh Lactames utiles notamment comme medicaments et leur procede de preparation
EP0003814A2 (de) * 1978-02-25 1979-09-05 Dr. Karl Thomae GmbH Neue Penicilline, ihre Salze, Verfahren zu ihrer Herstellung und diese Verbindungen enthaltende Arzneimittel
EP0006532A1 (de) * 1978-06-28 1980-01-09 Dr. Karl Thomae GmbH Neue Lactame, Verfahren zu ihrer Herstellung und diese Verbindungen enthaltende Arzneimittel

Also Published As

Publication number Publication date
AU8321282A (en) 1982-11-11
SE8202674L (sv) 1982-11-05
IL65602A0 (en) 1982-07-30
ES511884A0 (es) 1983-08-16
GR78166B (enrdf_load_stackoverflow) 1984-09-26
PL236277A1 (en) 1983-08-15
DE3215941A1 (de) 1983-05-05
FI821551A0 (fi) 1982-05-03
NO821456L (no) 1982-11-05
NL8201810A (nl) 1982-12-01
GB2101586A (en) 1983-01-19
DK198282A (da) 1982-11-05
FI821551L (fi) 1982-11-05
ES8307814A1 (es) 1983-08-16
FI821551A7 (fi) 1982-11-05
BG37227A1 (en) 1985-04-15
JPS5813590A (ja) 1983-01-26
IT8267577A0 (it) 1982-05-03
BE893057A (fr) 1982-08-30
IT1156467B (it) 1987-02-04

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