ES8307814A1 - "procedimiento de preparar compuestos beta-lactamicos". - Google Patents

"procedimiento de preparar compuestos beta-lactamicos".

Info

Publication number
ES8307814A1
ES8307814A1 ES511884A ES511884A ES8307814A1 ES 8307814 A1 ES8307814 A1 ES 8307814A1 ES 511884 A ES511884 A ES 511884A ES 511884 A ES511884 A ES 511884A ES 8307814 A1 ES8307814 A1 ES 8307814A1
Authority
ES
Spain
Prior art keywords
group
optionally
alkyl
hydroxy
substituent
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES511884A
Other languages
English (en)
Other versions
ES511884A0 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Chinoin Private Co Ltd
Original Assignee
Chinoin Gyogyszer es Vegyeszeti Termekek Gyara Zrt
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Chinoin Gyogyszer es Vegyeszeti Termekek Gyara Zrt filed Critical Chinoin Gyogyszer es Vegyeszeti Termekek Gyara Zrt
Publication of ES8307814A1 publication Critical patent/ES8307814A1/es
Publication of ES511884A0 publication Critical patent/ES511884A0/es
Granted legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14—Compounds having a nitrogen atom directly attached in position 7
    • C07D501/16—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
    • C07D501/20—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D499/21—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with a nitrogen atom directly attached in position 6 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
    • C07D499/44—Compounds with an amino radical acylated by carboxylic acids, attached in position 6
    • C07D499/48—Compounds with an amino radical acylated by carboxylic acids, attached in position 6 with a carbon chain, substituted by hetero atoms or by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, attached to the carboxamido radical
    • C07D499/58—Compounds with an amino radical acylated by carboxylic acids, attached in position 6 with a carbon chain, substituted by hetero atoms or by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, attached to the carboxamido radical substituted in alpha-position to the carboxamido radical
    • C07D499/64—Compounds with an amino radical acylated by carboxylic acids, attached in position 6 with a carbon chain, substituted by hetero atoms or by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, attached to the carboxamido radical substituted in alpha-position to the carboxamido radical by nitrogen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Cephalosporin Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)

Abstract

PROCEDIMIENTO DE PREPARAR COMPUESTOS ~J-LACTAMICOS. SE EMPLEA ALGUNO DE LOS SIGUIENTES PROCEDIMIENTOS: 1 ) REACCION DEL COMPUESTO (II) CON EL COMPUESTO (III). 2 ) REACCION DEL COMPUESTO (V) CON EL (IV), O BIEN. 3 ) REACCION DEL COMPUESTO (II) CON EL (VI). CUANDO SE EMPLEAN COMO SUBSTANCIAS DE PARTIDA CEFALEXINA Y 4-FLAVANILISOTIOCIANATO, LA REACCION PUEDE EFECTUARSE SEGUN EL PRIMER METODO. SEGUN EL CARACTER DE LAS SUBSTANCIAS DE PARTIDAS, PUEDEN APLICARSE COMO MEDIO DE REACCION HIDROCARBUROS ALIFATICOS CLORADOS, ETERES ALIFATICOS O BIEN OTROS DISOLVENTES APROTICOS, PREFERENTEMENTE ACETONIHILO O ACETATO DE ETILO O SUS MEZCLAS.
ES511884A 1981-05-04 1982-05-03 "procedimiento de preparar compuestos beta-lactamicos". Granted ES511884A0 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
HU115481 1981-05-04

Publications (2)

Publication Number Publication Date
ES8307814A1 true ES8307814A1 (es) 1983-08-16
ES511884A0 ES511884A0 (es) 1983-08-16

Family

ID=10953073

Family Applications (1)

Application Number Title Priority Date Filing Date
ES511884A Granted ES511884A0 (es) 1981-05-04 1982-05-03 "procedimiento de preparar compuestos beta-lactamicos".

Country Status (17)

Country Link
JP (1) JPS5813590A (es)
AU (1) AU8321282A (es)
BE (1) BE893057A (es)
BG (1) BG37227A1 (es)
DE (1) DE3215941A1 (es)
DK (1) DK198282A (es)
ES (1) ES511884A0 (es)
FI (1) FI821551L (es)
FR (1) FR2509311A1 (es)
GB (1) GB2101586A (es)
GR (1) GR78166B (es)
IL (1) IL65602A0 (es)
IT (1) IT1156467B (es)
NL (1) NL8201810A (es)
NO (1) NO821456L (es)
PL (1) PL236277A1 (es)
SE (1) SE8202674L (es)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3137376C2 (de) * 1981-09-19 1986-02-27 Degussa Ag, 6000 Frankfurt Verfahren zur Herstellung von 1,5-Alkylen-3-aryl-hydantoin-Derivaten
AU577105B2 (en) * 1985-04-02 1988-09-15 T.P.O. :Pharmachim: Acylaminic penicillin derivatives

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1476312A (en) * 1974-06-03 1977-06-10 Beecham Group Ltd Penicillins and cephalosporins
CA1074298A (en) * 1974-09-20 1980-03-25 E.R. Squibb And Sons 3-heterothio-7-ureido cephalosporins
CA1075679A (en) * 1975-07-30 1980-04-15 E.R. Squibb And Sons 3-heterothio-7-thioureido cephalosporins
JPS5239694A (en) * 1975-08-29 1977-03-28 Toyama Chem Co Ltd Producing novel penicillins and cephalosporins
US4063019A (en) * 1976-03-30 1977-12-13 E. R. Squibb & Sons, Inc. [[[(2,4-Dioxo-1-imidazolidinyl)amino]carbonyl]amino]-acetylcephalosporin derivatives
PT67170B (de) * 1976-11-06 1979-03-21 Merck Patent Gmbh Lactame verfahren zu ihrer herstellung und diese verbindungen enthaltende mittel
ES477520A1 (es) * 1978-02-25 1979-06-01 Thomae Gmbh Dr K Procedimiento para la preparacion de nuevas penicilinas.
DE2828261A1 (de) * 1978-06-28 1980-01-10 Thomae Gmbh Dr K Neue penicilline, ihre salze, verfahren zu ihrer herstellung und diese verbindungen enthaltende arzneimittel

Also Published As

Publication number Publication date
BG37227A1 (en) 1985-04-15
FI821551A0 (fi) 1982-05-03
FR2509311A1 (fr) 1983-01-14
JPS5813590A (ja) 1983-01-26
NL8201810A (nl) 1982-12-01
DE3215941A1 (de) 1983-05-05
NO821456L (no) 1982-11-05
IT8267577A0 (it) 1982-05-03
FI821551L (fi) 1982-11-05
BE893057A (fr) 1982-08-30
SE8202674L (sv) 1982-11-05
DK198282A (da) 1982-11-05
PL236277A1 (en) 1983-08-15
GR78166B (es) 1984-09-26
AU8321282A (en) 1982-11-11
IT1156467B (it) 1987-02-04
IL65602A0 (en) 1982-07-30
GB2101586A (en) 1983-01-19
ES511884A0 (es) 1983-08-16

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Legal Events

Date Code Title Description
FD1A Patent lapsed

Effective date: 19980302