FR2389622A1 - - Google Patents

Info

Publication number
FR2389622A1
FR2389622A1 FR7812084A FR7812084A FR2389622A1 FR 2389622 A1 FR2389622 A1 FR 2389622A1 FR 7812084 A FR7812084 A FR 7812084A FR 7812084 A FR7812084 A FR 7812084A FR 2389622 A1 FR2389622 A1 FR 2389622A1
Authority
FR
France
Prior art keywords
piperidinyl
phenyl
pharmaceutically acceptable
disclosed
following formula
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
FR7812084A
Other languages
English (en)
French (fr)
Other versions
FR2389622B1 (ru
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Janssen Pharmaceutica NV
Original Assignee
Janssen Pharmaceutica NV
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Pharmaceutica NV filed Critical Janssen Pharmaceutica NV
Publication of FR2389622A1 publication Critical patent/FR2389622A1/fr
Application granted granted Critical
Publication of FR2389622B1 publication Critical patent/FR2389622B1/fr
Expired legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D257/00Heterocyclic compounds containing rings having four nitrogen atoms as the only ring hetero atoms
    • C07D257/02Heterocyclic compounds containing rings having four nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D257/04Five-membered rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D211/00Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/36Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D211/56Nitrogen atoms
    • C07D211/58Nitrogen atoms attached in position 4
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pain & Pain Management (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biomedical Technology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
FR7812084A 1977-05-05 1978-04-24 Expired FR2389622B1 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US79381477A 1977-05-05 1977-05-05
US88618878A 1978-03-13 1978-03-13

Publications (2)

Publication Number Publication Date
FR2389622A1 true FR2389622A1 (ru) 1978-12-01
FR2389622B1 FR2389622B1 (ru) 1982-05-21

Family

ID=27121432

Family Applications (1)

Application Number Title Priority Date Filing Date
FR7812084A Expired FR2389622B1 (ru) 1977-05-05 1978-04-24

Country Status (26)

Country Link
JP (1) JPS53149980A (ru)
AT (1) AT368994B (ru)
AU (1) AU514360B2 (ru)
CA (1) CA1105464A (ru)
CH (1) CH635585A5 (ru)
CY (1) CY1253A (ru)
DE (1) DE2819873A1 (ru)
DK (1) DK152211C (ru)
ES (1) ES469473A1 (ru)
FI (1) FI64364C (ru)
FR (1) FR2389622B1 (ru)
GB (1) GB1598872A (ru)
HK (1) HK72585A (ru)
HU (1) HU179204B (ru)
IE (1) IE46836B1 (ru)
IL (1) IL54639A (ru)
IT (1) IT1105288B (ru)
KE (1) KE3429A (ru)
LU (1) LU79575A1 (ru)
NL (1) NL186861C (ru)
NO (1) NO148747C (ru)
NZ (1) NZ187164A (ru)
PH (1) PH12831A (ru)
SE (1) SE437516B (ru)
SU (1) SU867304A3 (ru)
YU (1) YU40703B (ru)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS6144294A (ja) * 1984-08-07 1986-03-03 Nippon Denso Co Ltd 熱交換器
US5053411A (en) * 1989-04-20 1991-10-01 Anaquest, Inc. N-aryl-N-[4-(1-heterocyclicalkyl)piperidinyl]amides and pharmaceutical compositions and methods employing such compounds
USRE34201E (en) * 1989-04-20 1993-03-23 Anaquest, Inc. N-aryl-N-[4-(1-heterocyclicalkyl)piperidinyl]amides and pharmaceutical compositions and methods employing such compounds
JPH08193074A (ja) * 1994-11-18 1996-07-30 Nippon Bayeragrochem Kk 除草性1−シクロプロピルテトラゾリノン類
JP2000327668A (ja) 1999-05-21 2000-11-28 Nippon Bayer Agrochem Co Ltd テトラゾリノン誘導体
BR0016063A (pt) * 1999-12-06 2002-08-06 Mallinckrodt Inc Métodos para a sìntese de alfentanila, sufentanila e remifentanila
JPWO2006030931A1 (ja) * 2004-09-14 2008-05-15 日本ケミファ株式会社 N−置換−n−(4−ピペリジニル)アミド誘導体

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3998834A (en) * 1975-03-14 1976-12-21 Janssen Pharmaceutica N.V. N-(4-piperidinyl)-n-phenylamides and -carbamates

Also Published As

Publication number Publication date
AU3552278A (en) 1979-11-01
YU108578A (en) 1983-01-21
AU514360B2 (en) 1981-02-05
JPS6324995B2 (ru) 1988-05-23
FR2389622B1 (ru) 1982-05-21
KE3429A (en) 1984-08-10
DE2819873A1 (de) 1978-11-09
IE780901L (en) 1978-11-05
FI781398A (fi) 1978-11-06
DK152211C (da) 1988-08-08
NL186861B (nl) 1990-10-16
NL186861C (nl) 1991-03-18
FI64364C (fi) 1983-11-10
IT1105288B (it) 1985-10-28
NO781559L (no) 1978-11-07
IL54639A0 (en) 1978-07-31
ES469473A1 (es) 1979-09-16
DK152211B (da) 1988-02-08
IL54639A (en) 1982-02-28
NO148747C (no) 1983-12-07
NO148747B (no) 1983-08-29
IE46836B1 (en) 1983-10-05
HK72585A (en) 1985-10-04
SU867304A3 (ru) 1981-09-23
ATA322078A (de) 1982-04-15
SE7805110L (sv) 1978-11-06
IT7849203A0 (it) 1978-05-04
SE437516B (sv) 1985-03-04
JPS53149980A (en) 1978-12-27
HU179204B (en) 1982-09-28
PH12831A (en) 1979-09-05
CA1105464A (en) 1981-07-21
DE2819873C2 (ru) 1989-05-03
YU40703B (en) 1986-04-30
CH635585A5 (en) 1983-04-15
LU79575A1 (fr) 1978-11-03
FI64364B (fi) 1983-07-29
DK193778A (da) 1978-11-06
CY1253A (en) 1984-08-31
NL7804844A (nl) 1978-11-07
AT368994B (de) 1982-11-25
GB1598872A (en) 1981-09-23
NZ187164A (en) 1981-03-16

Similar Documents

Publication Publication Date Title
ES469567A1 (es) Un procedimiento para la produccion de derivados de ciclos- porina
ES2044836T3 (es) Derivado de la piperidina, su utilizacion y compuesto farmaceutico que lo contiene.
FR2369297A1 (fr) Nouveaux esters d'acides androstadiene-17-carboxyliques
LU90317I2 (fr) Tacrolimus et ses sels et dérivés pharmaceutiquement acceptables
ES2001341A6 (es) Un procedimiento de producir un derivado de acido guanidinometilbenzoico.
FR2385713A1 (fr) Derives de 5-(4-(diarylmethyl)-1-piperazinylalkyl)benzimidazole ayant une activite antihistaminique, anti-allergique et anti-asthmatique
FR2372817A1 (fr) Derives d'acides thiazolidinecarboxyliques et d'acides apparentes, utiles comme agents anti-hypertension
CA2126118A1 (en) 5-Amino-8-Methyl-7-Pyrrolidinylquinoline-3-Carboxylic Acid Derivative
FR2389622A1 (ru)
FR2398745A1 (fr) Acides dithietane-1,3-carboxylique-2 et leur procede de preparation
FR2380278A1 (fr) Nouvelles 1-((diarylmethyl)aminoalkyl) piperidines
PT87277A (pt) Process for the preparation of new bicyclic compounds and pharmaceutical compositions comprising same
FR2395272A1 (fr) Nouveaux medicaments derives de l'acide amidinopenicillanique
GR3015475T3 (en) Sulfonylamino substituted bicyclyl hydroxamic acid derivatives.
FR2450837A1 (fr) Acides penicillaniques 6-b-substitues inhibiteurs de b-lactamase, leur procede de production et composition pharmaceutique les contenant
ES8501763A1 (es) "procedimiento para la fabricacion de derivados de la tetrahidro-5.6.7.7. 4h-tieno (3, 2-c) piridinona-2
FR2394514A1 (fr) Nouvel acide cyclohexanecarboxylique et ses derives
SE7702130L (sv) Forfarande for framstellning av n-(merkaptoacyl)-histidiner
FR2389631A1 (ru)
FR2390958A1 (fr) Association de substances actives utile au traitement du paludisme
FR2357527A1 (fr) Nouveau procede de synthese du chlorhydrate de derives particuliers de catecholamine
FR2430230A1 (fr) Medicaments a base de derives de l'acide anthranilique
FR2380271A1 (fr) Acides halogene-benzofuranone-carboxyliques utiles comme intermediaires de synthese
FR2398738A1 (fr) Preparation de benzoylurees
FR2370038A1 (fr) Derives de l'oxime de l'acide 4-(d-3-amino-3-carboxypropoxy) phenylglyoxylique, constituant la chaine laterale de l'antibiotique nocardicine

Legal Events

Date Code Title Description
CC Supplementary protection certificate (spc) laid open to the public (law of 25 june 1990)

Free format text: 92C0449, 920618

CB Supplementary protection certificate (spc) granted (law of 25 june 1990)

Free format text: 92C0449, 780424

CL Concession to grant licences