FIC20230025I1 - neratinibi - Google Patents

neratinibi

Info

Publication number
FIC20230025I1
FIC20230025I1 FIC20230025C FIC20230025C FIC20230025I1 FI C20230025 I1 FIC20230025 I1 FI C20230025I1 FI C20230025 C FIC20230025 C FI C20230025C FI C20230025 C FIC20230025 C FI C20230025C FI C20230025 I1 FIC20230025 I1 FI C20230025I1
Authority
FI
Finland
Prior art keywords
neratinib
Prior art date
Application number
FIC20230025C
Other languages
English (en)
Original Assignee
Wyeth Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=42313339&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=FIC20230025(I1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Wyeth Llc filed Critical Wyeth Llc
Publication of FIC20230025I1 publication Critical patent/FIC20230025I1/fi

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • A61K31/4709Non-condensed quinolines and containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • A61K31/47064-Aminoquinolines; 8-Aminoquinolines, e.g. chloroquine, primaquine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K39/00Medicinal preparations containing antigens or antibodies
    • A61K39/395Antibodies; Immunoglobulins; Immune serum, e.g. antilymphocytic serum
    • A61K39/39533Antibodies; Immunoglobulins; Immune serum, e.g. antilymphocytic serum against materials from animals
    • A61K39/39558Antibodies; Immunoglobulins; Immune serum, e.g. antilymphocytic serum against materials from animals against tumor tissues, cells, antigens
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/08Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
    • A61P19/10Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K39/00Medicinal preparations containing antigens or antibodies
    • A61K2039/505Medicinal preparations containing antigens or antibodies comprising antibodies
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2300/00Mixtures or combinations of active ingredients, wherein at least one active ingredient is fully defined in groups A61K31/00 - A61K41/00
FIC20230025C 2009-04-06 2023-07-19 neratinibi FIC20230025I1 (fi)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US16679609P 2009-04-06 2009-04-06

Publications (1)

Publication Number Publication Date
FIC20230025I1 true FIC20230025I1 (fi) 2023-07-19

Family

ID=42313339

Family Applications (2)

Application Number Title Priority Date Filing Date
FIEP15188350.1T FI3000467T3 (fi) 2009-04-06 2010-03-24 Rintasyöpähoitokuuri, jossa käytetään neratinibia
FIC20230025C FIC20230025I1 (fi) 2009-04-06 2023-07-19 neratinibi

Family Applications Before (1)

Application Number Title Priority Date Filing Date
FIEP15188350.1T FI3000467T3 (fi) 2009-04-06 2010-03-24 Rintasyöpähoitokuuri, jossa käytetään neratinibia

Country Status (30)

Country Link
US (1) US9211291B2 (fi)
EP (3) EP2416774B1 (fi)
JP (7) JP5992325B2 (fi)
KR (6) KR20140036332A (fi)
CN (3) CN105999264A (fi)
AR (1) AR076197A1 (fi)
AU (1) AU2010234968B2 (fi)
BR (1) BRPI1012699A2 (fi)
CA (1) CA2755789C (fi)
DK (1) DK3000467T3 (fi)
ES (2) ES2561495T3 (fi)
FI (2) FI3000467T3 (fi)
FR (1) FR23C1027I1 (fi)
HK (2) HK1167313A1 (fi)
HR (1) HRP20230315T1 (fi)
HU (2) HUE061640T2 (fi)
IL (4) IL264349B2 (fi)
LT (2) LT3000467T (fi)
MX (1) MX356593B (fi)
NL (1) NL301237I2 (fi)
NO (1) NO2023028I1 (fi)
NZ (1) NZ595143A (fi)
PL (1) PL3000467T3 (fi)
PT (1) PT3000467T (fi)
RU (2) RU2011139363A (fi)
SG (1) SG174382A1 (fi)
SI (1) SI3000467T1 (fi)
TW (2) TWI557108B (fi)
WO (1) WO2010117633A1 (fi)
ZA (1) ZA201108118B (fi)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
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RU2451524C2 (ru) 2005-11-04 2012-05-27 Вайет Противоопухолевые комбинации с ингибиторами mtor, герцептином и/или hki-272
US8022216B2 (en) 2007-10-17 2011-09-20 Wyeth Llc Maleate salts of (E)-N-{4-[3-chloro-4-(2-pyridinylmethoxy)anilino]-3-cyano-7-ethoxy-6-quinolinyl}-4-(dimethylamino)-2-butenamide and crystalline forms thereof
CA2725598C (en) 2008-06-17 2013-10-08 Wyeth Llc Antineoplastic combinations containing hki-272 and vinorelbine
NZ590464A (en) 2008-08-04 2012-10-26 Wyeth Llc Antineoplastic combinations of the 4-anilino-3-cyanoquinoline neratinib and capecitabine
DK3000467T3 (da) 2009-04-06 2023-03-27 Wyeth Llc Behandling med neratinib mod brystkræft
EP2498751B1 (en) 2009-11-09 2019-04-03 Wyeth LLC Coated drug spheroids and uses thereof for eliminating or reducing conditions such as emesis and diarrhea
KR20200022187A (ko) 2018-08-22 2020-03-03 울산대학교 산학협력단 Nono의 발현 또는 활성 억제제를 유효성분으로 포함하는 방사선 민감성 증진용 조성물
AU2020379734A1 (en) 2019-11-04 2022-05-05 Revolution Medicines, Inc. Ras inhibitors

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