FI962754A - Uusia mahdollisesti substituoituja fenyyli-imidatsolidiineja, menetelmä niiden valmistamiseksi sekä valmistuksen välituotteita, niiden käyttö lääkkeinä ja niitä käsittävät farmaseuttiset koostumukset - Google Patents

Uusia mahdollisesti substituoituja fenyyli-imidatsolidiineja, menetelmä niiden valmistamiseksi sekä valmistuksen välituotteita, niiden käyttö lääkkeinä ja niitä käsittävät farmaseuttiset koostumukset Download PDF

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Publication number
FI962754A
FI962754A FI962754A FI962754A FI962754A FI 962754 A FI962754 A FI 962754A FI 962754 A FI962754 A FI 962754A FI 962754 A FI962754 A FI 962754A FI 962754 A FI962754 A FI 962754A
Authority
FI
Finland
Prior art keywords
preparation
optionally substituted
pct
imidazolidines
pharmaceuticals
Prior art date
Application number
FI962754A
Other languages
English (en)
Swedish (sv)
Other versions
FI962754A0 (fi
FI112475B (fi
Inventor
Andre Claussner
Francois Goubet
Jean-Georges Teutsch
Original Assignee
Roussel Uclaf
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from FR9400042A external-priority patent/FR2715402B1/fr
Priority claimed from FR9410660A external-priority patent/FR2724169B1/fr
Application filed by Roussel Uclaf filed Critical Roussel Uclaf
Publication of FI962754A publication Critical patent/FI962754A/fi
Publication of FI962754A0 publication Critical patent/FI962754A0/fi
Application granted granted Critical
Publication of FI112475B publication Critical patent/FI112475B/fi

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
    • A61P5/26—Androgens
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D233/72—Two oxygen atoms, e.g. hydantoin
    • C07D233/76—Two oxygen atoms, e.g. hydantoin with substituted hydrocarbon radicals attached to the third ring carbon atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D233/72—Two oxygen atoms, e.g. hydantoin
    • C07D233/76—Two oxygen atoms, e.g. hydantoin with substituted hydrocarbon radicals attached to the third ring carbon atom
    • C07D233/78—Radicals substituted by oxygen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D233/86—Oxygen and sulfur atoms, e.g. thiohydantoin
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D233/88—Nitrogen atoms, e.g. allantoin
FI962754A 1994-01-05 1996-07-04 Uusia, mahdollisesti substituoituja fenyyli-imidatsolidiineja, menetelmä niiden valmistamiseksi, niiden käyttö lääkkeinä ja niitä käsittävät farmaseuttiset koostumukset FI112475B (fi)

Applications Claiming Priority (6)

Application Number Priority Date Filing Date Title
FR9400042A FR2715402B1 (fr) 1994-01-05 1994-01-05 Nouvelles phénylimidazolines éventuellement substituées, leur procédé et des intermédiaires de préparation, leur application comme médicaments et les compositions pharmaceutiques les renfermant.
FR9400042 1994-01-05
FR9410660 1994-09-06
FR9410660A FR2724169B1 (fr) 1994-09-06 1994-09-06 Nouvelles phenylimidazolidines eventuellement substituees, leur procede et des intermediaires de preparation, leur application comme medicaments et les compositions pharmaceutiques les renfermant
FR9500004 1995-01-04
PCT/FR1995/000004 WO1995018794A1 (fr) 1994-01-05 1995-01-04 Nouvelles phenylimidazolidines eventuellement substituees, leur procede et des intermediaires de preparation, leur application comme medicaments et les compositions pharmaceutiques les renfermant

Publications (3)

Publication Number Publication Date
FI962754A true FI962754A (fi) 1996-07-04
FI962754A0 FI962754A0 (fi) 1996-07-04
FI112475B FI112475B (fi) 2003-12-15

Family

ID=26230882

Family Applications (1)

Application Number Title Priority Date Filing Date
FI962754A FI112475B (fi) 1994-01-05 1996-07-04 Uusia, mahdollisesti substituoituja fenyyli-imidatsolidiineja, menetelmä niiden valmistamiseksi, niiden käyttö lääkkeinä ja niitä käsittävät farmaseuttiset koostumukset

Country Status (20)

Country Link
US (1) US5750553A (fi)
EP (1) EP0738263B1 (fi)
JP (1) JPH09507241A (fi)
KR (1) KR100372065B1 (fi)
CN (1) CN1113873C (fi)
AT (1) ATE200281T1 (fi)
AU (1) AU687152B2 (fi)
BR (1) BR9506457A (fi)
CA (1) CA2180379A1 (fi)
DE (1) DE69520560T2 (fi)
DK (1) DK0738263T3 (fi)
ES (1) ES2156204T3 (fi)
FI (1) FI112475B (fi)
GR (1) GR3035853T3 (fi)
HU (1) HUT76299A (fi)
IL (1) IL111908A (fi)
MA (1) MA23423A1 (fi)
PT (1) PT738263E (fi)
TW (1) TW521073B (fi)
WO (1) WO1995018794A1 (fi)

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Also Published As

Publication number Publication date
DE69520560D1 (de) 2001-05-10
EP0738263B1 (fr) 2001-04-04
DK0738263T3 (da) 2001-06-18
CN1113873C (zh) 2003-07-09
KR100372065B1 (ko) 2003-05-12
CA2180379A1 (fr) 1995-07-13
EP0738263A1 (fr) 1996-10-23
ATE200281T1 (de) 2001-04-15
HUT76299A (en) 1997-07-28
IL111908A (en) 2003-05-29
CN1141631A (zh) 1997-01-29
DE69520560T2 (de) 2001-09-13
FI962754A0 (fi) 1996-07-04
HU9601836D0 (en) 1996-09-30
US5750553A (en) 1998-05-12
JPH09507241A (ja) 1997-07-22
WO1995018794A1 (fr) 1995-07-13
PT738263E (pt) 2001-08-30
BR9506457A (pt) 1997-10-07
FI112475B (fi) 2003-12-15
GR3035853T3 (en) 2001-08-31
MA23423A1 (fr) 1995-10-01
AU687152B2 (en) 1998-02-19
IL111908A0 (en) 1995-03-15
ES2156204T3 (es) 2001-06-16
AU1457395A (en) 1995-08-01
TW521073B (en) 2003-02-21

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