FI962639A0 - Diaryyli-5,6-fuusioituneita heterosyklisiä happoja leukotrieeniantagonisteina - Google Patents
Diaryyli-5,6-fuusioituneita heterosyklisiä happoja leukotrieeniantagonisteinaInfo
- Publication number
- FI962639A0 FI962639A0 FI962639A FI962639A FI962639A0 FI 962639 A0 FI962639 A0 FI 962639A0 FI 962639 A FI962639 A FI 962639A FI 962639 A FI962639 A FI 962639A FI 962639 A0 FI962639 A0 FI 962639A0
- Authority
- FI
- Finland
- Prior art keywords
- diaryl
- fused heterocyclic
- leukotriene antagonists
- heterocyclic acids
- acids
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
- C07D491/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pulmonology (AREA)
- Immunology (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Ophthalmology & Optometry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US17493793A | 1993-12-28 | 1993-12-28 | |
US08/260,592 US5472964A (en) | 1992-12-22 | 1994-06-16 | Diaryl 5,6-fused heterocyclic acids as leukotriene antagonists |
PCT/CA1994/000716 WO1995018132A1 (en) | 1993-12-28 | 1994-12-22 | Diaryl 5,6-fused heterocyclic acids as leukotriene antagonists |
Publications (2)
Publication Number | Publication Date |
---|---|
FI962639A FI962639A (fi) | 1996-06-26 |
FI962639A0 true FI962639A0 (fi) | 1996-06-26 |
Family
ID=26870689
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
FI962639A FI962639A0 (fi) | 1993-12-28 | 1996-06-26 | Diaryyli-5,6-fuusioituneita heterosyklisiä happoja leukotrieeniantagonisteina |
Country Status (12)
Country | Link |
---|---|
US (1) | US5472964A (fi) |
EP (1) | EP0737196A1 (fi) |
JP (1) | JP3594603B2 (fi) |
CN (1) | CN1148389A (fi) |
AU (1) | AU684884B2 (fi) |
CA (1) | CA2180014A1 (fi) |
CZ (1) | CZ187996A3 (fi) |
FI (1) | FI962639A0 (fi) |
HU (1) | HUT76544A (fi) |
NO (1) | NO962717D0 (fi) |
SK (1) | SK83896A3 (fi) |
WO (1) | WO1995018132A1 (fi) |
Families Citing this family (15)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5656638A (en) * | 1995-04-18 | 1997-08-12 | Geron Corporation | Telomerase inhibitors |
AU732671B2 (en) * | 1996-02-08 | 2001-04-26 | Merck & Co., Inc. | Method of treatment and pharmaceutical composition |
US6262066B1 (en) | 1998-07-27 | 2001-07-17 | Schering Corporation | High affinity ligands for nociceptin receptor ORL-1 |
EP1321169A1 (en) * | 2001-12-18 | 2003-06-25 | Biofrontera Pharmaceuticals AG | Combination of a serotonin receptor antagonist with a histidine decarboxylase inhibitor as a medicament |
CA2371048C (en) | 2002-02-06 | 2011-01-04 | Delmar Chemicals Inc. | Process for the preparation of 1-(mercaptomethyl)-cyclopropaneacetic acid |
WO2006017505A2 (en) * | 2004-08-04 | 2006-02-16 | Schering Corporation | Pharmaceutical formulations comprising pleconaril for the treatment of airway diseases |
US20060110449A1 (en) | 2004-10-25 | 2006-05-25 | Lorber Richard R | Pharmaceutical composition |
WO2007101841A2 (en) * | 2006-03-06 | 2007-09-13 | Farmaprojects, S. A. | Process for preparing a leukotriene antagonist |
BRPI0712915A2 (pt) * | 2006-07-11 | 2012-10-09 | Schering Corp | sal de xinafoato de um composto de 5-oxazal-2-il-quinolina substituìdo |
US20110040095A1 (en) * | 2008-03-17 | 2011-02-17 | Dr. Reddy's Laboratories Ltd. | Preparation of montelukast and its salts |
MX2010011154A (es) * | 2008-04-11 | 2010-12-21 | Janssen Pharmaceutica Nv | Tiazolopiridin-2-iloxi-fenilo y tiazolopirazin-2-iloxifenilaminas como moduladores de la leucotrieno a4 hidrolasa. |
US9532717B2 (en) * | 2008-10-28 | 2017-01-03 | The Procter & Gamble Company | Method for diagnosing vulvovaginal disorders |
CN102834406A (zh) | 2009-06-16 | 2012-12-19 | 默沙东公司 | 作为糖皮质激素受体激动剂的新的[3.2-c]杂芳基甾体、其组合物和用途 |
CN110386888A (zh) * | 2019-07-30 | 2019-10-29 | 上海红蓝医药科技有限公司 | 一种低成本、高收率的1-(巯甲基)环丙基乙酸生产工艺 |
WO2023218023A1 (en) | 2022-05-13 | 2023-11-16 | Idorsia Pharmaceuticals Ltd | Thiazoloaryl-methyl substituted cyclic hydrazine-n-carboxamide derivatives |
Family Cites Families (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4794188A (en) * | 1982-12-01 | 1988-12-27 | Usv Pharmaceutical Corporation | Certain unsymmetrical quinolinyl ethers having anti-inflammatory and anti-allergic activity |
CA1322005C (en) * | 1987-11-25 | 1993-09-07 | Robert N. Young | Benzoheterazoles |
US5026698A (en) * | 1988-11-02 | 1991-06-25 | Nissan Chemical Industries, Ltd. | Thienopyridine type mevalonolactones |
DE19875039I2 (de) * | 1990-10-12 | 2003-05-22 | Merck Frosst Canada Inc | Ungesaettigte Hydroxyalkylchinolinsaeuren als Leukotrien-Antagonisten |
CA2053216C (en) * | 1990-10-12 | 2003-04-08 | Michel L. Belley | Saturated hydroxyalkylquinoline acids as leukotriene antagonists |
US5308850A (en) * | 1991-09-30 | 1994-05-03 | Merck Frosst Canada, Inc. | (Bicyclic-hetero-arylmethoxy)indoles as inhibitors of leukotriene biosynthesis |
US5506227A (en) * | 1992-04-13 | 1996-04-09 | Merck Frosst Canada, Inc. | Pyridine-substituted benzyl alcohols as leukotriene antagonists |
CA2111372C (en) * | 1992-12-22 | 2007-01-16 | Robert N. Young | Diaryl 5,6-fusedheterocyclic acids as leukotriene antagonists |
-
1994
- 1994-06-16 US US08/260,592 patent/US5472964A/en not_active Expired - Lifetime
- 1994-12-22 AU AU13781/95A patent/AU684884B2/en not_active Ceased
- 1994-12-22 CZ CZ961879A patent/CZ187996A3/cs unknown
- 1994-12-22 JP JP51764995A patent/JP3594603B2/ja not_active Expired - Fee Related
- 1994-12-22 CA CA002180014A patent/CA2180014A1/en not_active Abandoned
- 1994-12-22 EP EP95904990A patent/EP0737196A1/en not_active Withdrawn
- 1994-12-22 CN CN94194674A patent/CN1148389A/zh active Pending
- 1994-12-22 WO PCT/CA1994/000716 patent/WO1995018132A1/en not_active Application Discontinuation
- 1994-12-22 HU HU9601772A patent/HUT76544A/hu unknown
- 1994-12-22 SK SK838-96A patent/SK83896A3/sk unknown
-
1996
- 1996-06-26 FI FI962639A patent/FI962639A0/fi unknown
- 1996-06-27 NO NO962717A patent/NO962717D0/no unknown
Also Published As
Publication number | Publication date |
---|---|
HU9601772D0 (en) | 1996-09-30 |
NO962717L (no) | 1996-06-27 |
JPH09507080A (ja) | 1997-07-15 |
SK83896A3 (en) | 1997-02-05 |
JP3594603B2 (ja) | 2004-12-02 |
CZ187996A3 (en) | 1997-01-15 |
HUT76544A (en) | 1997-09-29 |
US5472964A (en) | 1995-12-05 |
CN1148389A (zh) | 1997-04-23 |
WO1995018132A1 (en) | 1995-07-06 |
CA2180014A1 (en) | 1995-07-06 |
FI962639A (fi) | 1996-06-26 |
EP0737196A1 (en) | 1996-10-16 |
AU1378195A (en) | 1995-07-17 |
AU684884B2 (en) | 1998-01-08 |
NO962717D0 (no) | 1996-06-27 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
ATE226578T1 (de) | Benzofuranderivate als tachykininantagonisten | |
DE59501802D1 (de) | Substituierte 1H-3-Aryl-pyrrolidin-2,4-dion-Derivate | |
BR9711262A (pt) | Derivados 6,6 substituido hetero biciclicos | |
MX20359A (es) | Derivados de 2-oxindol 3-substituidos. | |
NL300035I2 (nl) | Gesubstitueerde thiazolidinedionderivaten. | |
MX9201823A (es) | Derivados de quinolina. | |
KR950700304A (ko) | 5ht4-수용체 길항질로서 축합 인돌 유도체(condensed indole derivatives as 5ht4-receptor antagonists) | |
FI962639A0 (fi) | Diaryyli-5,6-fuusioituneita heterosyklisiä happoja leukotrieeniantagonisteina | |
FI961628A0 (fi) | Indolijohdannaisia NMDA-antagonisteina | |
MX9204190A (es) | Derivdos de 2-(4-hidroxipiperidino)-1-alcanol como agentes antiisquemicos. | |
FI955164A0 (fi) | Heterosykliset johdannaiset | |
MA26543A1 (fr) | Derives de pyrrolopyrrolone comme inhibiteurs d'elastase de neutrophiles. | |
ID22838A (id) | Oksazolidina sebagai antagonis 5-ht2a | |
FI970110A (fi) | Helico-bakteerin vastaisia heterosyklisiä atsolonijohdannaisia | |
DE68923913D1 (de) | Neplanocinderivate. | |
DE69106545D1 (de) | Verbesserungen an Leukotrien-Antagonieten. | |
DE69006142D1 (de) | Substituierte Glutaramidsäuren und Derivate. | |
ATE218564T1 (de) | Pyrazol-4-yl-hetaroylderivate als herbizide | |
ATE325118T1 (de) | Piperazinoderivate als neurokinin-antagonisten | |
DE69514315T2 (de) | AZABICYCLOALKYLDERIVATE VON IMIDAZO[1,5-a]INDOL-3-ONE ALS 5HT3 ANTAGONISTEN | |
NO950684D0 (no) | Nye imidazopyridinderivater som angiotensinII-antagonister | |
DE69013131D1 (de) | 2-(2-Cyclopropylpyrrolidin-4-ylthio)carbapenemderivate. | |
AU7379794A (en) | Aza-5,5-fused heterocyclic acids as leukotriene antagonists | |
FI940607A0 (fi) | Imidatso(5,1-C)(1,4)bentsoksatsin-1-onijohdannaiset 5HT3-antagonisteina | |
DE69710921T2 (de) | Heterocyclische substituierte pyrrolidinamid-derivate |