FI940607A0 - Imidatso(5,1-C)(1,4)bentsoksatsin-1-onijohdannaiset 5HT3-antagonisteina - Google Patents

Imidatso(5,1-C)(1,4)bentsoksatsin-1-onijohdannaiset 5HT3-antagonisteina

Info

Publication number
FI940607A0
FI940607A0 FI940607A FI940607A FI940607A0 FI 940607 A0 FI940607 A0 FI 940607A0 FI 940607 A FI940607 A FI 940607A FI 940607 A FI940607 A FI 940607A FI 940607 A0 FI940607 A0 FI 940607A0
Authority
FI
Finland
Prior art keywords
benzoxazin
imidazo
antagonists
derivatives
Prior art date
Application number
FI940607A
Other languages
English (en)
Swedish (sv)
Other versions
FI940607A (fi
Inventor
Mario Varasi
Franco Heidempergher
Claudio Arrigoni
Carla Caccia
Original Assignee
Erba Carlo Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Erba Carlo Spa filed Critical Erba Carlo Spa
Publication of FI940607A publication Critical patent/FI940607A/fi
Publication of FI940607A0 publication Critical patent/FI940607A0/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D519/00Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/26Psychostimulants, e.g. nicotine, cocaine

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Psychiatry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
FI940607A 1992-06-12 1994-02-09 Imidatso(5,1-C)(1,4)bentsoksatsin-1-onijohdannaiset 5HT3-antagonisteina FI940607A0 (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB929212486A GB9212486D0 (en) 1992-06-12 1992-06-12 Derivatives of substituted imidazo benzoxazin-1-one and process for their preparation
PCT/EP1993/001498 WO1993025555A1 (en) 1992-06-12 1993-06-14 Derivatives of imidazo [5,1-c][1, 4]benzoxazin-1-one as 5 ht3 antagonists

Publications (2)

Publication Number Publication Date
FI940607A FI940607A (fi) 1994-02-09
FI940607A0 true FI940607A0 (fi) 1994-02-09

Family

ID=10716979

Family Applications (1)

Application Number Title Priority Date Filing Date
FI940607A FI940607A0 (fi) 1992-06-12 1994-02-09 Imidatso(5,1-C)(1,4)bentsoksatsin-1-onijohdannaiset 5HT3-antagonisteina

Country Status (15)

Country Link
US (1) US5364854A (fi)
EP (1) EP0606421A1 (fi)
JP (1) JPH06510064A (fi)
CN (1) CN1081679A (fi)
AU (1) AU661784B2 (fi)
CA (1) CA2114643A1 (fi)
FI (1) FI940607A0 (fi)
GB (1) GB9212486D0 (fi)
HU (1) HUT70415A (fi)
IL (1) IL105867A0 (fi)
MX (1) MX9303392A (fi)
NZ (1) NZ253132A (fi)
PL (1) PL302373A1 (fi)
WO (1) WO1993025555A1 (fi)
ZA (1) ZA934107B (fi)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9410441D0 (en) * 1994-05-25 1994-07-13 Erba Carlo Spa Azabicycloakyl derivatives of imidazo (1,5-a) indol-3-one and process for their preparation
GB9410469D0 (en) * 1994-05-25 1994-07-13 Erba Farmitalia Imidazolylalkyl derivatives of imidazo (5,1-c) (1,4) benzoxazin-1-one and process for their preparation
US6451771B1 (en) * 1999-02-12 2002-09-17 Nutramax Laboratories, Inc. Use of anabolic agents anti-catabolic agents and antioxidant agents for protection treatment and repair of connective tissues in humans and animals
WO2002092606A1 (fr) * 2001-05-15 2002-11-21 Takeda Chemical Industries, Ltd. Derives d'imidazolidine fusionnes, leur procede de preparation et d'utilisation
CN110028521B (zh) * 2019-05-27 2020-07-14 湖南科技大学 11-芳基-1,4-苯并恶嗪酮并咪唑啉类化合物及其制备方法和用途

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1052009B (it) * 1975-12-30 1981-06-20 Erba Carlo Spa Imidazo 4.3 c 1.4 benzossazino imidazo 4.3 c 1.4 benzotiazino pirazo 2.1 c 1.4 benzossazino e pirazo 2.1 c 1.4 benzotiazino derivati
GB1538479A (en) * 1976-05-21 1979-01-17 Roussel Labor Ltd Imidazobenzoxazines
SE444319B (sv) * 1977-11-18 1986-04-07 Roussel Uclaf Nya imidazobensoxazinderivat, forfarande for framstellning derav och farmaceutiska kompositioner innehallande dessa foreningar
SE441449B (sv) * 1979-02-09 1985-10-07 Roussel Uclaf Heterocykliska derivat och farmaceutiska kompositioner innehallande dessa derivat
DK476885D0 (da) * 1985-10-17 1985-10-17 Ferrosan As Heterocycliske forbindelser og fremgangsmaader til fremstilling heraf
EP0235878A3 (en) * 1986-01-16 1989-06-14 Beecham Group Plc Novel compounds
GB9106571D0 (en) * 1991-03-27 1991-05-15 Erba Carlo Spa Derivatives of substituted imidazol-2-one and process for their preparation

Also Published As

Publication number Publication date
CA2114643A1 (en) 1993-12-23
NZ253132A (en) 1996-02-27
US5364854A (en) 1994-11-15
HUT70415A (en) 1995-10-30
HU9400404D0 (en) 1994-05-30
GB9212486D0 (en) 1992-07-22
AU661784B2 (en) 1995-08-03
CN1081679A (zh) 1994-02-09
PL302373A1 (en) 1994-07-25
ZA934107B (en) 1994-01-12
FI940607A (fi) 1994-02-09
EP0606421A1 (en) 1994-07-20
JPH06510064A (ja) 1994-11-10
WO1993025555A1 (en) 1993-12-23
AU4325793A (en) 1994-01-04
IL105867A0 (en) 1993-10-20
MX9303392A (es) 1994-06-30

Similar Documents

Publication Publication Date Title
DE69409503T2 (de) 1,6-diaminopurin-derivate
NL300035I1 (nl) Gesubstitueerde thiahzolidinedionderivaten.
DK0533268T3 (da) Benzanilidderivater som 5HT-1D antagonister
LV10099A (lv) Bicikliski heterocikliski atvasinajumi
DK0447891T3 (da) Thieno(2,3-d)pyrimidinderivater
MX9100717A (es) Antagonistas de la bradiquinina
NO932146D0 (no) Benzimidazolderivater
FI961628A0 (fi) Indolijohdannaisia NMDA-antagonisteina
FI930429A0 (fi) Nya 1,4-dihyropyridinderivat
KR950703530A (ko) 5-HT4 길항제(5-HT4 Antagonists)
TR26336A (tr) SüBSTITüE EDILMIS PIRAZOLIN TüREVLERI
DK301789D0 (da) Neplanocin-derivater
ATE116980T1 (de) Verbesserungen an leukotrien-antagonieten.
FI923290A (fi) Imidazo(2,1-b)bensotiazol-3-acetamidderivat
DK0432275T3 (da) Substituerede bicykloheptandionderivater
FI951798A0 (fi) Bentsofuraanijohdannaiset 5-HT1-kaltaisina reseptoriantagonisteina
DE69514315D1 (de) AZABICYCLOALKYLDERIVATE VON IMIDAZO[1,5-a]INDOL-3-ONE ALS 5HT3 ANTAGONISTEN
FI940607A0 (fi) Imidatso(5,1-C)(1,4)bentsoksatsin-1-onijohdannaiset 5HT3-antagonisteina
ZA93144B (en) Substituted benzimidazole derivatives
DE69122555T2 (de) 2,4-Dihydroxyadipinsäurederivate
KR950700297A (ko) 5-HT3-수용체 길항제로서의 2,6-메타노-2H-퀴놀리진 유도체(2,6-Methano-2H-quinolizin derivative as 5-HT3-receptor antagonist)
FI922980A (fi) 2-piperidinylpyrimidin-4-karboxamidderivat, framstaellning av dessa ochterapeutisk anvaendning av dessa
NO931897D0 (no) Fremgangsmaate for fremstilling av dibeskyttet 2,3-hydroksymetyl-cyklobutanol
MX9201931A (es) Nuevos derivados de tiazol.
FI840088A0 (fi) Foerfarande foer framstaellning av substituerade karboxi-tiazolo (3,2-a)pyrimidinderivat

Legal Events

Date Code Title Description
FD Application lapsed