FI935658A0 - Nya selektiva aromatasinhiberande 4(5)-imidazoler - Google Patents

Nya selektiva aromatasinhiberande 4(5)-imidazoler

Info

Publication number
FI935658A0
FI935658A0 FI935658A FI935658A FI935658A0 FI 935658 A0 FI935658 A0 FI 935658A0 FI 935658 A FI935658 A FI 935658A FI 935658 A FI935658 A FI 935658A FI 935658 A0 FI935658 A0 FI 935658A0
Authority
FI
Finland
Prior art keywords
aromatazinic
imidazole
selective
acid
selective aromatazinic
Prior art date
Application number
FI935658A
Other languages
English (en)
Finnish (fi)
Other versions
FI935658A7 (fi
Inventor
Arto Johannes Karjalainen
Marja-Liisa Soedervall
Arja Marketta Kalapudas
Reino Olavi Pelkonen
Aire Marja Laine
Risto Arvo Sakari Lammintausta
Jarmo Sakari Salonen
Original Assignee
Orion Yhtymae Oy
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB919113142A external-priority patent/GB9113142D0/en
Application filed by Orion Yhtymae Oy filed Critical Orion Yhtymae Oy
Publication of FI935658A7 publication Critical patent/FI935658A7/fi
Publication of FI935658A0 publication Critical patent/FI935658A0/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/64Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms, e.g. histidine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • A61P35/02Antineoplastic agents specific for leukemia

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Hematology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)
FI935658A 1991-06-18 1993-12-16 Nya selektiva aromatasinhiberande 4(5)-imidazoler FI935658A0 (fi)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB919113142A GB9113142D0 (en) 1991-06-18 1991-06-18 New selective aromatase inhibiting 4(5)-imidazoles
GB919125924A GB9125924D0 (en) 1991-06-18 1991-12-05 Stereoisomers of an imidazole derivative
PCT/FI1992/000184 WO1992022537A1 (en) 1991-06-18 1992-06-12 New selective aromatase inhibiting 4(5)-imidazoles

Publications (2)

Publication Number Publication Date
FI935658A7 FI935658A7 (fi) 1993-12-16
FI935658A0 true FI935658A0 (fi) 1993-12-16

Family

ID=26299089

Family Applications (1)

Application Number Title Priority Date Filing Date
FI935658A FI935658A0 (fi) 1991-06-18 1993-12-16 Nya selektiva aromatasinhiberande 4(5)-imidazoler

Country Status (25)

Country Link
US (1) US5559141A (cs)
EP (1) EP0589975A1 (cs)
JP (1) JPH06508119A (cs)
KR (1) KR940701386A (cs)
CN (1) CN1068819A (cs)
AU (1) AU665002B2 (cs)
BG (1) BG98306A (cs)
CA (1) CA2111469A1 (cs)
CZ (1) CZ280293A3 (cs)
FI (1) FI935658A0 (cs)
GB (1) GB9125924D0 (cs)
HR (1) HRP920170A2 (cs)
HU (1) HUT67325A (cs)
IE (1) IE921963A1 (cs)
IL (2) IL102216A (cs)
LT (1) LT3164B (cs)
LV (1) LV10093B (cs)
MX (1) MX9203000A (cs)
NO (1) NO934688D0 (cs)
NZ (1) NZ243139A (cs)
PT (1) PT100604A (cs)
SI (1) SI9200113A (cs)
SK (1) SK144393A3 (cs)
TW (1) TW206217B (cs)
WO (1) WO1992022537A1 (cs)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB2273704B (en) * 1992-12-16 1997-01-22 Orion Yhtymae Oy Triazolyl diaryl selective aromatase inhibiting compounds
SE9302333D0 (sv) * 1993-07-06 1993-07-06 Ab Astra New compounds
US6063930A (en) * 1996-04-03 2000-05-16 Merck & Co., Inc. Substituted imidazole compounds useful as farnesyl-protein transferase inhibitors
US6080870A (en) * 1996-04-03 2000-06-27 Merck & Co., Inc. Biaryl substituted imidazole compounds useful as farnesyl-protein transferase inhibitors
EP0891333A1 (en) * 1996-04-03 1999-01-20 Merck & Co., Inc. Inhibitors of farnesyl-protein transferase
US6297239B1 (en) * 1997-10-08 2001-10-02 Merck & Co., Inc. Inhibitors of prenyl-protein transferase
CN1466572A (zh) 2000-07-28 2004-01-07 ס����ҩ��ʽ���� 吡咯衍生物
MXPA06003951A (es) 2003-10-07 2006-06-27 Renovis Inc Derivados de amida como ligandos del canal de ion y composiciones farmaceuticas y sus metodos de uso.
EA200701835A1 (ru) * 2005-02-28 2008-02-28 Реновис, Инк. Амидные производные в качестве лигандов ионных каналов, их фармацевтические композиции и способы их применения
US7576099B2 (en) 2005-02-28 2009-08-18 Renovis, Inc. Amide derivatives as ion-channel ligands and pharmaceutical compositions and methods of using the same
US7902247B2 (en) * 2008-01-09 2011-03-08 Allergan, Inc. Substituted-aryl-2-phenylethyl-1H-imidazole compounds as subtype selective modulators of alpha 2B and/or alpha 2C adrenergic receptors
WO2024226608A2 (en) * 2023-04-25 2024-10-31 Aglaeapharma Inc. Imidazole containing compounds, derivatives therefore, and uses thereof

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4605661A (en) * 1984-06-18 1986-08-12 Eli Lilly And Company Aromastase inhibiting α,α-diarylimidazole-4(5)-propionitriles, α,α-diarylimidazole-4(5)-propionamides, and 4(5)-(2,2-diarylethyl)imidazoles
GB2210875B (en) * 1987-10-09 1991-05-29 Farmos Oy Aromatase inhibiting 4(5)-imidazoles
AU627559B2 (en) * 1989-03-30 1992-08-27 Farmos-Yhtyma Oy Novel aromatase inhibiting 4(5)-imidazoles
US5439928A (en) * 1989-03-30 1995-08-08 Orion-Yhtyma Oy Aromatase inhibiting 4(5)-imidazoles
GB2248058B (en) * 1990-09-21 1994-09-14 Orion Yhtymae Oy Aromatase inhibiting 4(5)-imidazoles

Also Published As

Publication number Publication date
BG98306A (bg) 1994-08-30
IL115439A0 (en) 1995-12-31
IL102216A (en) 1996-06-18
CZ280293A3 (en) 1994-05-18
FI935658A7 (fi) 1993-12-16
MX9203000A (es) 1993-02-01
CN1068819A (zh) 1993-02-10
PT100604A (pt) 1993-10-29
LTIP175A (lt) 1994-08-25
CA2111469A1 (en) 1992-12-23
LT3164B (en) 1995-02-27
LV10093A (lv) 1994-05-10
IL102216A0 (en) 1993-01-14
NO934688L (no) 1993-12-17
NO934688D0 (no) 1993-12-17
SK144393A3 (en) 1994-11-09
US5559141A (en) 1996-09-24
TW206217B (cs) 1993-05-21
AU665002B2 (en) 1995-12-14
KR940701386A (ko) 1994-05-28
HRP920170A2 (en) 1994-08-31
HUT67325A (en) 1995-03-28
EP0589975A1 (en) 1994-04-06
WO1992022537A1 (en) 1992-12-23
AU1978392A (en) 1993-01-12
IE921963A1 (en) 1992-12-30
LV10093B (en) 1995-02-20
HU9303653D0 (en) 1994-04-28
NZ243139A (en) 1994-08-26
GB9125924D0 (en) 1992-02-05
SI9200113A (en) 1992-12-31
JPH06508119A (ja) 1994-09-14

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Legal Events

Date Code Title Description
FD Application lapsed