FI924756A7 - 1,5-Bentsotiasepinonin johdannaiset, niiden valmistukset ja farmaseutt inen käyttö - Google Patents

1,5-Bentsotiasepinonin johdannaiset, niiden valmistukset ja farmaseutt inen käyttö Download PDF

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Publication number
FI924756A7
FI924756A7 FI924756A FI924756A FI924756A7 FI 924756 A7 FI924756 A7 FI 924756A7 FI 924756 A FI924756 A FI 924756A FI 924756 A FI924756 A FI 924756A FI 924756 A7 FI924756 A7 FI 924756A7
Authority
FI
Finland
Prior art keywords
preparations
pharmaceutical use
benzothiazepinone
derivatives
benzothiazepinone derivatives
Prior art date
Application number
FI924756A
Other languages
English (en)
Finnish (fi)
Swedish (sv)
Other versions
FI924756L (fi
FI924756A0 (fi
Inventor
Aldo Salimbeni
Saturnino Caliari
Francesco Fici
Elso Manghisi
Original Assignee
St Luso Farmaco Ditalia S P A
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by St Luso Farmaco Ditalia S P A filed Critical St Luso Farmaco Ditalia S P A
Publication of FI924756L publication Critical patent/FI924756L/fi
Publication of FI924756A0 publication Critical patent/FI924756A0/fi
Publication of FI924756A7 publication Critical patent/FI924756A7/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D281/00Heterocyclic compounds containing rings of more than six members having one nitrogen atom and one sulfur atom as the only ring hetero atoms
    • C07D281/02Seven-membered rings
    • C07D281/04Seven-membered rings having the hetero atoms in positions 1 and 4
    • C07D281/08Seven-membered rings having the hetero atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D281/10Seven-membered rings having the hetero atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems condensed with one six-membered ring
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/12Drugs for disorders of the metabolism for electrolyte homeostasis
    • A61P3/14Drugs for disorders of the metabolism for electrolyte homeostasis for calcium homeostasis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/08Vasodilators for multiple indications
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Endocrinology (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
FI924756A 1990-04-27 1991-04-18 1,5-Bentsotiasepinonin johdannaiset, niiden valmistukset ja farmaseutt inen käyttö FI924756A7 (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IT20160A IT1240686B (it) 1990-04-27 1990-04-27 Derivati 1,5-benzotiazepinonici, loro preparazione e uso farmaceutico
PCT/EP1991/000742 WO1991017153A1 (en) 1990-04-27 1991-04-18 1,5-benzothiazepinone derivatives, their preparations and pharmaceutical use

Publications (3)

Publication Number Publication Date
FI924756L FI924756L (fi) 1992-10-20
FI924756A0 FI924756A0 (fi) 1992-10-20
FI924756A7 true FI924756A7 (fi) 1992-10-20

Family

ID=11164306

Family Applications (1)

Application Number Title Priority Date Filing Date
FI924756A FI924756A7 (fi) 1990-04-27 1991-04-18 1,5-Bentsotiasepinonin johdannaiset, niiden valmistukset ja farmaseutt inen käyttö

Country Status (20)

Country Link
US (1) US5571807A (enExample)
EP (1) EP0526495A1 (enExample)
JP (1) JPH05506654A (enExample)
CN (1) CN1056101A (enExample)
AU (1) AU645317B2 (enExample)
BG (1) BG97014A (enExample)
BR (1) BR9106372A (enExample)
CA (1) CA2081204A1 (enExample)
CS (1) CS120991A2 (enExample)
FI (1) FI924756A7 (enExample)
HU (1) HU9203326D0 (enExample)
IE (1) IE71033B1 (enExample)
IL (1) IL97859A0 (enExample)
IN (1) IN172160B (enExample)
IT (1) IT1240686B (enExample)
MA (1) MA22143A1 (enExample)
PT (1) PT97508A (enExample)
RO (1) RO111269B1 (enExample)
WO (1) WO1991017153A1 (enExample)
ZA (1) ZA913171B (enExample)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ATE167858T1 (de) * 1994-09-16 1998-07-15 Orion Corp Fermion Verfahren zur herstellung von pharmazeutisch aktiven benzothiazepinderivaten.
FI97725C (fi) * 1995-02-17 1997-02-10 Orion Yhtymae Oy Menetelmä diltiatseemin valmistamiseksi
US5559229A (en) * 1995-06-01 1996-09-24 Acic (Canada) Inc. Method for the manufacture of benzothiazepine
WO1996038429A1 (en) * 1995-06-01 1996-12-05 Acic (Canada) Inc. Method for the manufacture of benzothiazepine derivatives
WO2006079077A2 (en) * 2005-01-20 2006-07-27 Acadia Pharmaceuticals Inc. Use of diltiazem or analogs thereof as modulators of ghrelin receptor

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3562257A (en) * 1967-10-28 1971-02-09 Tanabe Seiyaku Co Benzothiazepine derivatives
IT1206505B (it) * 1983-07-22 1989-04-27 Schiapparelli Farma Nuovi derivati benzotiazepinonici, metodo per la loro preparazione e composizioni farmaceutiche che licontengono.
DE3771143D1 (de) * 1986-08-20 1991-08-08 Mcneilab Inc Benzothiazepin-vasodilatoren mit aralkylsubstitution.
US4902684A (en) * 1988-06-20 1990-02-20 E. R. Squibb & Sons, Inc. Benzazepine and benzothiazepine derivatives
US4902687A (en) * 1989-03-27 1990-02-20 Eli Lilly And Company Excitatory amino acid receptor antagonists
ATE116643T1 (de) * 1989-04-28 1995-01-15 Tanabe Seiyaku Co Verfahren zur herstellung von 1,5- benzothiazepinderivaten.
JPH085869B2 (ja) * 1990-03-08 1996-01-24 田辺製薬株式会社 1,5−ベンゾチアゼピン誘導体の製法

Also Published As

Publication number Publication date
EP0526495A1 (en) 1993-02-10
ZA913171B (en) 1992-02-26
RO111269B1 (ro) 1996-08-30
AU7695491A (en) 1991-11-27
IT1240686B (it) 1993-12-17
AU645317B2 (en) 1994-01-13
CS120991A2 (en) 1991-12-17
FI924756L (fi) 1992-10-20
IT9020160A1 (it) 1991-10-27
JPH05506654A (ja) 1993-09-30
PT97508A (pt) 1992-01-31
HU9203326D0 (en) 1993-01-28
FI924756A0 (fi) 1992-10-20
IL97859A0 (en) 1992-06-21
IT9020160A0 (it) 1990-04-27
MA22143A1 (fr) 1991-12-31
WO1991017153A1 (en) 1991-11-14
US5571807A (en) 1996-11-05
IE911411A1 (en) 1991-11-06
IN172160B (enExample) 1993-04-17
CN1056101A (zh) 1991-11-13
BR9106372A (pt) 1993-04-27
BG97014A (bg) 1993-12-24
CA2081204A1 (en) 1991-10-28
IE71033B1 (en) 1997-01-15

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