FI902522A0 - Menetelmä terapeuttisesti käyttökelpoisten imidatsopyridiini-, imidatsopyrimidiini-, imidatsopyridatsiini- ja imidatsopyratsiinijohdannaisten valmistamiseksi - Google Patents

Menetelmä terapeuttisesti käyttökelpoisten imidatsopyridiini-, imidatsopyrimidiini-, imidatsopyridatsiini- ja imidatsopyratsiinijohdannaisten valmistamiseksi

Info

Publication number
FI902522A0
FI902522A0 FI902522A FI902522A FI902522A0 FI 902522 A0 FI902522 A0 FI 902522A0 FI 902522 A FI902522 A FI 902522A FI 902522 A FI902522 A FI 902522A FI 902522 A0 FI902522 A0 FI 902522A0
Authority
FI
Finland
Prior art keywords
imidazopyridazine
imidazopyrimidine
imidazopyridine
preparation
therapeutically useful
Prior art date
Application number
FI902522A
Other languages
English (en)
Swedish (sv)
Other versions
FI93449B (fi
FI93449C (fi
Inventor
David Anthony Roberts
Simon Thomas Russel
Keith Hopkinson Gibson
Robin Wood
Arnold Harry Ratcliffe
Original Assignee
Ici Plc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=26295388&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=FI902522(A0) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from GB898911855A external-priority patent/GB8911855D0/en
Priority claimed from GB909005843A external-priority patent/GB9005843D0/en
Application filed by Ici Plc filed Critical Ici Plc
Publication of FI902522A0 publication Critical patent/FI902522A0/fi
Publication of FI93449B publication Critical patent/FI93449B/fi
Application granted granted Critical
Publication of FI93449C publication Critical patent/FI93449C/fi

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D473/00—Heterocyclic compounds containing purine ring systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Diabetes (AREA)
  • Emergency Medicine (AREA)
  • Endocrinology (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
FI902522A 1989-05-23 1990-05-22 Menetelmä terapeuttisesti käyttökelpoisten imidatsopyridiini-, imidatsopyrimidiini-, imidatsopyridatsiini- ja imidatsopyratsiinijohdannaisten valmistamiseksi FI93449C (fi)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
GB8911855 1989-05-23
GB898911855A GB8911855D0 (en) 1989-05-23 1989-05-23 Azaindenes
GB9005843 1990-03-15
GB909005843A GB9005843D0 (en) 1990-03-15 1990-03-15 Nitrogen heterocycles

Publications (3)

Publication Number Publication Date
FI902522A0 true FI902522A0 (fi) 1990-05-22
FI93449B FI93449B (fi) 1994-12-30
FI93449C FI93449C (fi) 1995-04-10

Family

ID=26295388

Family Applications (1)

Application Number Title Priority Date Filing Date
FI902522A FI93449C (fi) 1989-05-23 1990-05-22 Menetelmä terapeuttisesti käyttökelpoisten imidatsopyridiini-, imidatsopyrimidiini-, imidatsopyridatsiini- ja imidatsopyratsiinijohdannaisten valmistamiseksi

Country Status (14)

Country Link
EP (1) EP0399731B2 (fi)
JP (1) JPH0749429B2 (fi)
AT (1) ATE98245T1 (fi)
AU (1) AU621483B2 (fi)
CA (1) CA2017066C (fi)
DE (1) DE69005026T3 (fi)
DK (1) DK0399731T4 (fi)
ES (1) ES2060951T5 (fi)
FI (1) FI93449C (fi)
IE (1) IE64514B1 (fi)
IL (1) IL94282A (fi)
NO (1) NO174202C (fi)
NZ (1) NZ233581A (fi)
PT (1) PT94114B (fi)

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US5128327A (en) * 1991-03-25 1992-07-07 Merck & Co., Inc. Angiotensin II antagonists incorporating a nitrogen containing six membered ring heterocycle
US5177074A (en) * 1991-03-26 1993-01-05 Merck & Co., Inc. Angiotensin ii antagonists incorporating a substituted thiophene or furan
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US5798364A (en) * 1992-03-26 1998-08-25 Merck Patent Gesellschaft Mit Beschrankter Haftung Imidazopyridines
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US5198438A (en) * 1991-05-07 1993-03-30 Merck & Co., Inc. Angiotensin ii antagonists incorporating a substituted thiophene or furan
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JP5202301B2 (ja) 2005-04-12 2013-06-05 ヴィコール・ファルマ・アーベー 新規な三環系アンジオテンシンｉｉアゴニスト
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CN109715615A (zh) 2016-06-29 2019-05-03 蒙特利尔大学 联芳甲基杂环

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Also Published As

Publication number Publication date
DE69005026T3 (de) 2002-02-14
EP0399731A1 (en) 1990-11-28
ES2060951T3 (es) 1994-12-01
EP0399731B1 (en) 1993-12-08
DK0399731T3 (da) 1994-02-14
AU621483B2 (en) 1992-03-12
JPH035480A (ja) 1991-01-11
DE69005026T2 (de) 1994-04-21
NO174202C (no) 1994-04-06
PT94114A (pt) 1991-01-08
DE69005026D1 (de) 1994-01-20
NO174202B (no) 1993-12-20
PT94114B (pt) 2001-04-30
IL94282A0 (en) 1991-03-10
FI93449B (fi) 1994-12-30
IE64514B1 (en) 1995-08-09
AU5477990A (en) 1990-11-29
NZ233581A (en) 1992-10-28
NO902262D0 (no) 1990-05-22
CA2017066A1 (en) 1990-11-23
IE901594L (en) 1990-11-23
NO902262L (no) 1990-11-26
JPH0749429B2 (ja) 1995-05-31
ES2060951T5 (es) 2001-10-16
CA2017066C (en) 2000-08-08
IL94282A (en) 1995-12-31
ATE98245T1 (de) 1993-12-15
EP0399731B2 (en) 2001-07-11
FI93449C (fi) 1995-04-10
DK0399731T4 (da) 2001-09-17

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Legal Events

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Owner name: ZENECA LIMITED

BB Publication of examined application
FG Patent granted

Owner name: ASTRAZENECA UK LIMITED