FI872379A0 - Förfarande för framställning av farmakologiskt verkande 1,5-diaryl-3-(w-substituerad-lägrealkyl)-pyrazoler - Google Patents

Förfarande för framställning av farmakologiskt verkande 1,5-diaryl-3-(w-substituerad-lägrealkyl)-pyrazoler

Info

Publication number
FI872379A0
FI872379A0 FI872379A FI872379A FI872379A0 FI 872379 A0 FI872379 A0 FI 872379A0 FI 872379 A FI872379 A FI 872379A FI 872379 A FI872379 A FI 872379A FI 872379 A0 FI872379 A0 FI 872379A0
Authority
FI
Finland
Prior art keywords
pyrazoles
diaryl
substituted
preparation
lower alkyl
Prior art date
Application number
FI872379A
Other languages
English (en)
Finnish (fi)
Other versions
FI94340B (sv
FI872379A (sv
FI94340C (sv
Inventor
Michael Paul Wachter
Michael Paul Ferro
Original Assignee
Ortho Pharma Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ortho Pharma Corp filed Critical Ortho Pharma Corp
Publication of FI872379A0 publication Critical patent/FI872379A0/sv
Publication of FI872379A publication Critical patent/FI872379A/sv
Publication of FI94340B publication Critical patent/FI94340B/sv
Application granted granted Critical
Publication of FI94340C publication Critical patent/FI94340C/sv

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/14Antitussive agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/08Antiallergic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/04Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C59/00Compounds having carboxyl groups bound to acyclic carbon atoms and containing any of the groups OH, O—metal, —CHO, keto, ether, groups, groups, or groups
    • C07C59/40Unsaturated compounds
    • C07C59/76Unsaturated compounds containing keto groups
    • C07C59/84Unsaturated compounds containing keto groups containing six membered aromatic rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C59/00Compounds having carboxyl groups bound to acyclic carbon atoms and containing any of the groups OH, O—metal, —CHO, keto, ether, groups, groups, or groups
    • C07C59/40Unsaturated compounds
    • C07C59/76Unsaturated compounds containing keto groups
    • C07C59/88Unsaturated compounds containing keto groups containing halogen
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Cardiology (AREA)
  • Pulmonology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Hospice & Palliative Care (AREA)
  • Vascular Medicine (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Urology & Nephrology (AREA)
  • Immunology (AREA)
  • Dermatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
FI872379A 1986-05-29 1987-05-28 Förfarande för framställning av farmakologiskt verkande 1,5-diaryl-3-(w-substituerad-lägrealkyl)-pyrazoler FI94340C (sv)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US86799686A 1986-05-29 1986-05-29
US86799686 1986-05-29
US4266187 1987-04-29
US07/042,661 US4826868A (en) 1986-05-29 1987-04-29 1,5-Diaryl-3-substituted pyrazoles pharmaceutical compositions and use

Publications (4)

Publication Number Publication Date
FI872379A0 true FI872379A0 (sv) 1987-05-28
FI872379A FI872379A (sv) 1987-11-30
FI94340B FI94340B (sv) 1995-05-15
FI94340C FI94340C (sv) 1995-08-25

Family

ID=26719497

Family Applications (1)

Application Number Title Priority Date Filing Date
FI872379A FI94340C (sv) 1986-05-29 1987-05-28 Förfarande för framställning av farmakologiskt verkande 1,5-diaryl-3-(w-substituerad-lägrealkyl)-pyrazoler

Country Status (21)

Country Link
US (1) US4826868A (sv)
EP (1) EP0248594B1 (sv)
JP (1) JP2512751B2 (sv)
KR (1) KR960007163B1 (sv)
CN (1) CN1028227C (sv)
AU (1) AU596844B2 (sv)
CA (1) CA1337122C (sv)
DE (2) DE10199049I2 (sv)
DK (1) DK170202B1 (sv)
ES (1) ES2059377T3 (sv)
FI (1) FI94340C (sv)
HK (1) HK14094A (sv)
HU (1) HU221300B1 (sv)
IE (1) IE63856B1 (sv)
IL (1) IL82671A0 (sv)
LU (1) LU90829I2 (sv)
NL (1) NL300057I2 (sv)
NO (2) NO172236C (sv)
NZ (1) NZ220353A (sv)
PH (1) PH25126A (sv)
PT (1) PT84964B (sv)

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US4956379A (en) * 1990-02-13 1990-09-11 Bristol-Myers Squibb Company Pyrazole carboxylic acids and esters and inhibition of blood platelet aggregation therewith
FR2665898B1 (fr) * 1990-08-20 1994-03-11 Sanofi Derives d'amido-3 pyrazole, procede pour leur preparation et compositions pharmaceutiques les contenant.
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Also Published As

Publication number Publication date
NO172236C (no) 1993-06-23
FI94340B (sv) 1995-05-15
FI872379A (sv) 1987-11-30
NO2001016I1 (no) 2001-10-01
HUT68247A (en) 1995-06-28
PH25126A (en) 1991-02-19
DE10199049I2 (de) 2003-01-09
NO872228D0 (no) 1987-05-27
AU7360887A (en) 1987-12-10
JPS6322080A (ja) 1988-01-29
PT84964B (pt) 1990-02-08
DK273587A (da) 1987-11-30
DE3788244T2 (de) 1994-04-14
CN1028227C (zh) 1995-04-19
NO872228L (no) 1987-11-30
PT84964A (en) 1987-06-01
NL300057I2 (nl) 2002-01-02
IE871403L (en) 1987-11-29
EP0248594A3 (en) 1988-11-17
IL82671A0 (en) 1987-11-30
NL300057I1 (nl) 2001-12-01
EP0248594A2 (en) 1987-12-09
LU90829I2 (fr) 2001-11-12
HK14094A (en) 1994-03-04
AU596844B2 (en) 1990-05-17
IE63856B1 (en) 1995-06-14
NO172236B (no) 1993-03-15
EP0248594B1 (en) 1993-11-24
JP2512751B2 (ja) 1996-07-03
DK170202B1 (da) 1995-06-12
DE3788244D1 (de) 1994-01-05
DK273587D0 (da) 1987-05-27
HU221300B1 (en) 2002-09-28
US4826868A (en) 1989-05-02
ES2059377T3 (es) 1994-11-16
FI94340C (sv) 1995-08-25
DE10199049I1 (de) 2002-01-10
KR870011100A (ko) 1987-12-21
KR960007163B1 (ko) 1996-05-29
CN87103953A (zh) 1987-12-09
NZ220353A (en) 1989-05-29
CA1337122C (en) 1995-09-26

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