FI871479A0 - Menetelmä lääkeaineina käyttökelpoisten perhydrotiatsepiini- ja perhydroatsepiinijohdannaisten valmistamiseksi - Google Patents

Menetelmä lääkeaineina käyttökelpoisten perhydrotiatsepiini- ja perhydroatsepiinijohdannaisten valmistamiseksi

Info

Publication number
FI871479A0
FI871479A0 FI871479A FI871479A FI871479A0 FI 871479 A0 FI871479 A0 FI 871479A0 FI 871479 A FI871479 A FI 871479A FI 871479 A FI871479 A FI 871479A FI 871479 A0 FI871479 A0 FI 871479A0
Authority
FI
Finland
Prior art keywords
perhydrotiazepine
perhydroazepine
pharmaceuticals
derivatives
useful
Prior art date
Application number
FI871479A
Other languages
English (en)
Swedish (sv)
Other versions
FI90418B (fi
FI871479A (fi
FI90418C (fi
Inventor
Hiroaki Yanagisawa
Sadao Ishihara
Akiko Ando
Hiroyuki Koike
Yasuteru Iijima
Original Assignee
Sankyo Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sankyo Co filed Critical Sankyo Co
Publication of FI871479A0 publication Critical patent/FI871479A0/fi
Publication of FI871479A publication Critical patent/FI871479A/fi
Publication of FI90418B publication Critical patent/FI90418B/fi
Application granted granted Critical
Publication of FI90418C publication Critical patent/FI90418C/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K5/00Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/02Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link
    • C07K5/022Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the structure -X-C(=O)-(C)n-N-C-C(=O)-Y-; X and Y being heteroatoms; n being 1 or 2
    • C07K5/0222Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the structure -X-C(=O)-(C)n-N-C-C(=O)-Y-; X and Y being heteroatoms; n being 1 or 2 with the first amino acid being heterocyclic, e.g. Pro, Trp
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
FI871479A 1986-04-04 1987-04-03 Menetelmä lääkeaineina käyttökelpoisten perhydrotiatsepiini- ja perhydroatsepiinijohdannaisten valmistamiseksi FI90418C (fi)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
JP7790486 1986-04-04
JP7790486 1986-04-04
JP18357686 1986-08-05
JP18357686 1986-08-05

Publications (4)

Publication Number Publication Date
FI871479A0 true FI871479A0 (fi) 1987-04-03
FI871479A FI871479A (fi) 1987-10-05
FI90418B FI90418B (fi) 1993-10-29
FI90418C FI90418C (fi) 1994-02-10

Family

ID=26418950

Family Applications (1)

Application Number Title Priority Date Filing Date
FI871479A FI90418C (fi) 1986-04-04 1987-04-03 Menetelmä lääkeaineina käyttökelpoisten perhydrotiatsepiini- ja perhydroatsepiinijohdannaisten valmistamiseksi

Country Status (15)

Country Link
US (1) US4778790A (fi)
EP (1) EP0240366B1 (fi)
KR (1) KR930002508B1 (fi)
CN (1) CN1015260B (fi)
AU (1) AU599642B2 (fi)
CA (1) CA1336774C (fi)
DE (1) DE3788888T2 (fi)
DK (1) DK173287A (fi)
ES (1) ES2061490T3 (fi)
FI (1) FI90418C (fi)
HK (1) HK1005735A1 (fi)
HU (1) HU208121B (fi)
IE (1) IE61433B1 (fi)
NZ (1) NZ219884A (fi)
SU (1) SU1598876A3 (fi)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4959359A (en) * 1989-10-06 1990-09-25 Hoffmann-La Roche Inc. Phenyl-thiazepinones as calcium regulating agents
EP0669936B1 (en) * 1992-10-30 2000-11-22 Merrell Pharmaceuticals Inc. Mercaptoacetylamide bicyclic lactam derivatives useful as inhibitors of enkephalinase and ace
US7015212B1 (en) 1999-05-12 2006-03-21 The United States Of America As Represented By The Department Of Health And Human Services Thiazepine inhibitors of HIV-1 integrase

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GR74635B (fi) * 1980-08-18 1984-06-29 Merck & Co Inc
US4629787A (en) * 1980-08-18 1986-12-16 Merck & Co., Inc. Substituted caprolactam derivatives as antihypertensives
US4680392A (en) * 1980-08-18 1987-07-14 Merck & Co., Inc. Substituted caprolactam derivatives as antihypertensives
US4587050A (en) * 1980-08-18 1986-05-06 Merck & Co., Inc. Substituted enantholactam derivatives as antihypertensives
EP0068173B1 (en) * 1981-06-05 1984-09-26 Merck & Co. Inc. Perhydro-1,4-thiazepin-5-one and perhydro-1,4-thiazocin-5-one derivatives, process for preparing and pharmceutical composition containing the same
US4460579A (en) * 1983-02-28 1984-07-17 E. R. Squibb & Sons, Inc. Thiazine and thiazepine containing compounds
US4512988A (en) * 1984-03-01 1985-04-23 E. R. Squibb & Sons, Inc. Acylamino oxo or hydroxy substituted alkylamino thiazines and thiazepines
SU1435151A3 (ru) * 1984-04-10 1988-10-30 Санкио Компани Лимитед (Фирма) Способ получени производных пергидротиазепина или их кислотно-аддитивных фармацевтически приемлемых солей
US4666901A (en) * 1984-05-17 1987-05-19 Merck & Co., Inc. Substituted lactams useful as angiotensin converting enzyme inhibitors
JPH0637473B2 (ja) * 1985-10-11 1994-05-18 三共株式会社 ラクタム化合物

Also Published As

Publication number Publication date
FI90418B (fi) 1993-10-29
HU208121B (en) 1993-08-30
US4778790A (en) 1988-10-18
EP0240366A3 (en) 1989-05-10
AU7111587A (en) 1987-10-08
KR930002508B1 (ko) 1993-04-03
NZ219884A (en) 1989-06-28
CN87103684A (zh) 1987-12-09
DK173287A (da) 1987-10-05
AU599642B2 (en) 1990-07-26
HUT47569A (en) 1989-03-28
EP0240366A2 (en) 1987-10-07
KR870010042A (ko) 1987-11-30
SU1598876A3 (ru) 1990-10-07
CN1015260B (zh) 1992-01-01
ES2061490T3 (es) 1994-12-16
FI871479A (fi) 1987-10-05
HK1005735A1 (en) 1999-01-22
DE3788888T2 (de) 1994-06-23
IE61433B1 (en) 1994-11-02
IE870861L (en) 1987-10-04
EP0240366B1 (en) 1994-01-26
DK173287D0 (da) 1987-04-03
FI90418C (fi) 1994-02-10
DE3788888D1 (de) 1994-03-10
CA1336774C (en) 1995-08-22

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Legal Events

Date Code Title Description
BB Publication of examined application
MM Patent lapsed

Owner name: SANKYO COMPANY LIMITED