FI102169B1 - 3-aminopyrrolit, menetelmä niiden valmistamiseksi ja niiden käyttö lääkeaineina - Google Patents

3-aminopyrrolit, menetelmä niiden valmistamiseksi ja niiden käyttö lääkeaineina

Info

Publication number
FI102169B1
FI102169B1 FI905689A FI905689A FI102169B1 FI 102169 B1 FI102169 B1 FI 102169B1 FI 905689 A FI905689 A FI 905689A FI 905689 A FI905689 A FI 905689A FI 102169 B1 FI102169 B1 FI 102169B1
Authority
FI
Finland
Prior art keywords
aminopyrroles
pharmaceuticals
preparation
Prior art date
Application number
FI905689A
Other languages
English (en)
Swedish (sv)
Other versions
FI905689A0 (fi
FI905689A (fi
FI102169B (fi
Inventor
Juergen Liebscher
Alexander Knoll
Alexej Uschmajew
Andreas Rolfs
Dieter Lohmann
Gottfried Faust
Eveline Morgenstern
Peter Scharfenberg
Original Assignee
Dresden Arzneimittel
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Dresden Arzneimittel filed Critical Dresden Arzneimittel
Publication of FI905689A0 publication Critical patent/FI905689A0/fi
Publication of FI905689A publication Critical patent/FI905689A/fi
Application granted granted Critical
Publication of FI102169B1 publication Critical patent/FI102169B1/fi
Publication of FI102169B publication Critical patent/FI102169B/fi

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/30—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
    • C07D207/34—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/08—Antiepileptics; Anticonvulsants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
FI905689A 1989-11-17 1990-11-16 3-aminopyrrolit, menetelmä niiden valmistamiseksi ja niiden käyttö lää keaineina FI102169B (fi)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DD89334670A DD298912A5 (de) 1989-11-17 1989-11-17 Verfahren zur herstellung von 3-aminopyrrolen

Publications (4)

Publication Number Publication Date
FI905689A0 FI905689A0 (fi) 1990-11-16
FI905689A FI905689A (fi) 1991-05-18
FI102169B1 true FI102169B1 (fi) 1998-10-30
FI102169B FI102169B (fi) 1998-10-30

Family

ID=5613902

Family Applications (1)

Application Number Title Priority Date Filing Date
FI905689A FI102169B (fi) 1989-11-17 1990-11-16 3-aminopyrrolit, menetelmä niiden valmistamiseksi ja niiden käyttö lää keaineina

Country Status (10)

Country Link
US (2) US5502051A (fi)
EP (1) EP0431371B1 (fi)
JP (1) JPH07113015B2 (fi)
DD (1) DD298912A5 (fi)
DE (1) DE59010759D1 (fi)
ES (1) ES2108005T3 (fi)
FI (1) FI102169B (fi)
HU (1) HUT56343A (fi)
RU (2) RU2120796C1 (fi)
YU (1) YU48469B (fi)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE4227479A1 (de) * 1992-08-20 1994-02-24 Dresden Arzneimittel Verfahren zur Herstellung von 1-unsubstituierten 3-Aminopyrrolen
US5792778A (en) * 1995-08-10 1998-08-11 Merck & Co., Inc. 2-substituted aryl pyrroles, compositions containing such compounds and methods of use
US5837719A (en) * 1995-08-10 1998-11-17 Merck & Co., Inc. 2,5-substituted aryl pyrroles, compositions containing such compounds and methods of use
WO1997016441A1 (en) * 1995-10-31 1997-05-09 Merck & Co., Inc. Substituted aryl pyrroles, compositions containing such compounds and methods of use
US5908858A (en) 1996-04-05 1999-06-01 Sankyo Company, Limited 1,2-diphenylpyrrole derivatives, their preparation and their therapeutic uses
DE19629976A1 (de) * 1996-07-25 1998-01-29 Dresden Arzneimittel Verwendung von 4-(p-Halogenphenyl)-3-morpholinopyrrol-2-carbonsäuremethylester zur Prophylaxe und Behandlung der Folgen der akuten und chronischen zerebralen Minderdurchblutung sowie neurodegenerativer Erkrankungen
US5776954A (en) * 1996-10-30 1998-07-07 Merck & Co., Inc. Substituted pyridyl pyrroles, compositions containing such compounds and methods of use
US7122666B2 (en) * 1999-07-21 2006-10-17 Sankyo Company, Limited Heteroaryl-substituted pyrrole derivatives, their preparation and their therapeutic uses
US8247423B2 (en) 2007-07-12 2012-08-21 Tragara Pharmaceuticals, Inc. Methods and compositions for the treatment of cancer, tumors, and tumor-related disorders
US9944597B2 (en) 2013-09-16 2018-04-17 The Board Of Regents Of The University Of Texas System Polysubstituted pyrroles having microtubule-disrupting, cytotoxic and antitumor activities and methods of use thereof

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4198502A (en) * 1973-08-22 1980-04-15 Gruppo Lepetit S.P.A. Aminopyrrole derivatives
US4748183A (en) * 1986-06-13 1988-05-31 Warner-Lambert Company N-1H-tetrazol-5-yl-2-thiophene carboxamides, N-1H-tetrazol-5-yl-2-pyrrole carboxamides, N-1H-tetrazol-5-yl-2-furan carboxamides, and anti-allergic and anti-inflammatory use thereof

Also Published As

Publication number Publication date
EP0431371A1 (de) 1991-06-12
RU2060991C1 (ru) 1996-05-27
JPH07113015B2 (ja) 1995-12-06
YU48469B (sh) 1998-08-14
EP0431371B1 (de) 1997-09-10
FI905689A0 (fi) 1990-11-16
DE59010759D1 (de) 1997-10-16
ES2108005T3 (es) 1997-12-16
JPH03271271A (ja) 1991-12-03
US5502051A (en) 1996-03-26
DD298912A5 (de) 1992-03-19
RU2120796C1 (ru) 1998-10-27
HU907176D0 (en) 1991-05-28
HUT56343A (en) 1991-08-28
YU217390A (sh) 1993-05-28
US5684160A (en) 1997-11-04
FI905689A (fi) 1991-05-18
FI102169B (fi) 1998-10-30

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Legal Events

Date Code Title Description
MM Patent lapsed

Owner name: ARZNEIMITTELWERK DRESDEN GMBH