FI102169B1 - 3-aminopyrroler, förfaranden för deras framställning, och deras användning som läkemedel - Google Patents

3-aminopyrroler, förfaranden för deras framställning, och deras användning som läkemedel

Info

Publication number
FI102169B1
FI102169B1 FI905689A FI905689A FI102169B1 FI 102169 B1 FI102169 B1 FI 102169B1 FI 905689 A FI905689 A FI 905689A FI 905689 A FI905689 A FI 905689A FI 102169 B1 FI102169 B1 FI 102169B1
Authority
FI
Finland
Prior art keywords
aminopyrroles
pharmaceuticals
preparation
Prior art date
Application number
FI905689A
Other languages
English (en)
Finnish (fi)
Other versions
FI905689A0 (fi
FI102169B (sv
FI905689A (fi
Inventor
Juergen Liebscher
Alexander Knoll
Alexej Uschmajew
Andreas Rolfs
Dieter Lohmann
Gottfried Faust
Eveline Morgenstern
Peter Scharfenberg
Original Assignee
Dresden Arzneimittel
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Dresden Arzneimittel filed Critical Dresden Arzneimittel
Publication of FI905689A0 publication Critical patent/FI905689A0/fi
Publication of FI905689A publication Critical patent/FI905689A/fi
Application granted granted Critical
Publication of FI102169B publication Critical patent/FI102169B/sv
Publication of FI102169B1 publication Critical patent/FI102169B1/sv

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/30—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
    • C07D207/34—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/08—Antiepileptics; Anticonvulsants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pain & Pain Management (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyrrole Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
FI905689A 1989-11-17 1990-11-16 3-aminopyrroler, förfaranden för deras framställning, och deras användning som läkemedel FI102169B1 (sv)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DD89334670A DD298912A5 (de) 1989-11-17 1989-11-17 Verfahren zur herstellung von 3-aminopyrrolen

Publications (4)

Publication Number Publication Date
FI905689A0 FI905689A0 (fi) 1990-11-16
FI905689A FI905689A (fi) 1991-05-18
FI102169B FI102169B (sv) 1998-10-30
FI102169B1 true FI102169B1 (sv) 1998-10-30

Family

ID=5613902

Family Applications (1)

Application Number Title Priority Date Filing Date
FI905689A FI102169B1 (sv) 1989-11-17 1990-11-16 3-aminopyrroler, förfaranden för deras framställning, och deras användning som läkemedel

Country Status (10)

Country Link
US (2) US5502051A (sv)
EP (1) EP0431371B1 (sv)
JP (1) JPH07113015B2 (sv)
DD (1) DD298912A5 (sv)
DE (1) DE59010759D1 (sv)
ES (1) ES2108005T3 (sv)
FI (1) FI102169B1 (sv)
HU (1) HUT56343A (sv)
RU (2) RU2060991C1 (sv)
YU (1) YU48469B (sv)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE4227479A1 (de) * 1992-08-20 1994-02-24 Dresden Arzneimittel Verfahren zur Herstellung von 1-unsubstituierten 3-Aminopyrrolen
US5837719A (en) * 1995-08-10 1998-11-17 Merck & Co., Inc. 2,5-substituted aryl pyrroles, compositions containing such compounds and methods of use
US5792778A (en) * 1995-08-10 1998-08-11 Merck & Co., Inc. 2-substituted aryl pyrroles, compositions containing such compounds and methods of use
WO1997016441A1 (en) * 1995-10-31 1997-05-09 Merck & Co., Inc. Substituted aryl pyrroles, compositions containing such compounds and methods of use
US5908858A (en) 1996-04-05 1999-06-01 Sankyo Company, Limited 1,2-diphenylpyrrole derivatives, their preparation and their therapeutic uses
DE19629976A1 (de) * 1996-07-25 1998-01-29 Dresden Arzneimittel Verwendung von 4-(p-Halogenphenyl)-3-morpholinopyrrol-2-carbonsäuremethylester zur Prophylaxe und Behandlung der Folgen der akuten und chronischen zerebralen Minderdurchblutung sowie neurodegenerativer Erkrankungen
US5776954A (en) * 1996-10-30 1998-07-07 Merck & Co., Inc. Substituted pyridyl pyrroles, compositions containing such compounds and methods of use
US7122666B2 (en) * 1999-07-21 2006-10-17 Sankyo Company, Limited Heteroaryl-substituted pyrrole derivatives, their preparation and their therapeutic uses
CA2692977A1 (en) 2007-07-12 2009-01-15 Tragara Pharmaceuticals, Inc. Methods and compositions for the treatment of cancer, tumors, and tumor-related disorders
WO2015039073A1 (en) 2013-09-16 2015-03-19 Kellogg Glen E Polysubstituted pyrroles having microtubule-disrupting, cytotoxic and antitumor activities and methds of use thereof

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4198502A (en) * 1973-08-22 1980-04-15 Gruppo Lepetit S.P.A. Aminopyrrole derivatives
US4748183A (en) * 1986-06-13 1988-05-31 Warner-Lambert Company N-1H-tetrazol-5-yl-2-thiophene carboxamides, N-1H-tetrazol-5-yl-2-pyrrole carboxamides, N-1H-tetrazol-5-yl-2-furan carboxamides, and anti-allergic and anti-inflammatory use thereof

Also Published As

Publication number Publication date
YU217390A (sh) 1993-05-28
ES2108005T3 (es) 1997-12-16
RU2060991C1 (ru) 1996-05-27
US5684160A (en) 1997-11-04
RU2120796C1 (ru) 1998-10-27
DE59010759D1 (de) 1997-10-16
EP0431371A1 (de) 1991-06-12
HU907176D0 (en) 1991-05-28
DD298912A5 (de) 1992-03-19
EP0431371B1 (de) 1997-09-10
YU48469B (sh) 1998-08-14
HUT56343A (en) 1991-08-28
US5502051A (en) 1996-03-26
FI905689A0 (fi) 1990-11-16
JPH07113015B2 (ja) 1995-12-06
FI102169B (sv) 1998-10-30
JPH03271271A (ja) 1991-12-03
FI905689A (fi) 1991-05-18

Similar Documents

Publication Publication Date Title
FI111263B (sv) Nya erytromycinderivater, förfarande för framställning av dessa och deras användning som läkemedel samt mellanproduktaminer för förfarandet
BR8006404A (pt) Derivados de imidazo-diazepina, processo para sua preparacao, medicamento e uso
BR9000116A (pt) Alfa-diazo-beta-cetoester polifuncional,processo para sua preparacao e sua utilizacao
EE9800265A (et) Erütromütsiini derivaadid, nende valmistamismeetod ja kasutamine ravimitena
BR8804191A (pt) Derivados de avermectina,processo para sua preparacao,composicoes praguicidas e aplicacao
DK0562583T3 (da) Hidtil ukendte alkylendiammoniumdiclavulanatderivater, fremgangsmåde til fremstilling deraf samt anvendelse deraf
FI885488A (sv) 2,2-difluorcyklopropyletanderivat, förfarande för deras framställning och deras användning som medel för bekämpande av skadeinsekter
BR8603592A (pt) Derivados de piridazinona,processo para sua preparacao,e composicoes inseticidas
AR243499A1 (es) Un procedimiento para la preparacion de derivados de sulfonanilida.
GB8917687D0 (en) Aminopiperazine derivatives,processes for preparation thereof and pharmaceutical composition comprising the same
FI102169B1 (sv) 3-aminopyrroler, förfaranden för deras framställning, och deras användning som läkemedel
EE200000129A (et) Asendatud 1,2,3,4,5,6-heksahüdro-2,6-metano-3-bensasotsiin-10-oolid, nende valmistamise meetod ja kasutamine ravimitena
FI960316A (sv) Oxatiolaner, förfarande för deras framställning och farmaceutiska kompositioner innehållande desamma
EP0255601A3 (en) Dialkylnaleinimides, process for their preparation and their use as herbicide
FI941912A (sv) 3-kinolylsubstituerade dihydropyridiner, förfarande för framställning av dessa samt använding av dessa i läkemedel
BR9600370A (pt) Benzenossulfoniluréias e-tiouréias substituídas processo para a sua preparação seus usos e medicamento contendo as mesmas
BR8704325A (pt) Compostos,processo para sua preparacao e utilizacao
ZA905147B (en) Substituted 3-aminosydnone imines,process for their preparation and their use
BR8706059A (pt) Pirazolinas,processo para sua preparacao,composicao inseticida e aplicacao
BR8805857A (pt) Poliazocorantes,processo para sua preparacao e utilizacao
ZA879706B (en) New alkanesulfonanilide derivatives,processes for preparation thereof and pharmaceutical composition comprising the same
BR8705442A (pt) Compostos de halogenociclo-propila,processo para sua preparacao,composicao com efeito herbicida e aplicacao
BR8602597A (pt) Produto de adicao,processo para sua preparacao e composicao compreendendo o mesmo
FI102370B (sv) Förfarande för framställnig av N-metyl-3,4-dimetoxifenyletylamin
FI933004A (sv) Foerfarande foer framstaellning av N-alkyl-3,4-dialkyloxianiliner och derivat daerav

Legal Events

Date Code Title Description
MM Patent lapsed

Owner name: ARZNEIMITTELWERK DRESDEN GMBH