FI753045A - - Google Patents

Info

Publication number
FI753045A
FI753045A FI753045A FI753045A FI753045A FI 753045 A FI753045 A FI 753045A FI 753045 A FI753045 A FI 753045A FI 753045 A FI753045 A FI 753045A FI 753045 A FI753045 A FI 753045A
Authority
FI
Finland
Application number
FI753045A
Other languages
Finnish (fi)
Other versions
FI58918B (fi
FI58918C (fi
Inventor
Amedeo Omodei-Sale
Emilio Toia
Giulio Galliani
Leonard J Lerner
Original Assignee
Lepetit Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lepetit Spa filed Critical Lepetit Spa
Publication of FI753045A publication Critical patent/FI753045A/fi
Publication of FI58918B publication Critical patent/FI58918B/fi
Application granted granted Critical
Publication of FI58918C publication Critical patent/FI58918C/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D235/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D209/00Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/44Iso-indoles; Hydrogenated iso-indoles
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Investigating Or Analysing Biological Materials (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Peptides Or Proteins (AREA)
FI753045A 1974-11-23 1975-10-31 Foerfarande foer framstaellning av imidazo(2,1-a)isokinoliner och 5,6-dihydro-imidazo(2,1-a)isokinoliner med antireproduktiv aktivitet FI58918C (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB50855/74A GB1484615A (en) 1974-11-23 1974-11-23 Tricyclic n-containing derivatives
GB5085574 1974-11-23

Publications (3)

Publication Number Publication Date
FI753045A true FI753045A (ja) 1976-05-24
FI58918B FI58918B (fi) 1981-01-30
FI58918C FI58918C (fi) 1981-05-11

Family

ID=10457662

Family Applications (2)

Application Number Title Priority Date Filing Date
FI753046A FI58919C (fi) 1974-11-23 1975-10-31 Foerfarande foer framstaellning av pyrazolo(5,1-a)isokinoliner och 5,6-dihydropyrazolo(5,1-a)isokinoliner med antireproduktiv aktivitet
FI753045A FI58918C (fi) 1974-11-23 1975-10-31 Foerfarande foer framstaellning av imidazo(2,1-a)isokinoliner och 5,6-dihydro-imidazo(2,1-a)isokinoliner med antireproduktiv aktivitet

Family Applications Before (1)

Application Number Title Priority Date Filing Date
FI753046A FI58919C (fi) 1974-11-23 1975-10-31 Foerfarande foer framstaellning av pyrazolo(5,1-a)isokinoliner och 5,6-dihydropyrazolo(5,1-a)isokinoliner med antireproduktiv aktivitet

Country Status (25)

Country Link
US (1) US4075342A (ja)
JP (1) JPS5516513B2 (ja)
AR (2) AR210476A1 (ja)
AT (2) AT346332B (ja)
BE (1) BE835836A (ja)
CA (2) CA1068274A (ja)
CH (2) CH614208A5 (ja)
DD (2) DD122819A5 (ja)
DE (1) DE2551868C2 (ja)
DK (2) DK522275A (ja)
ES (2) ES442863A1 (ja)
FI (2) FI58919C (ja)
FR (1) FR2291747A1 (ja)
GB (1) GB1484615A (ja)
GR (2) GR58293B (ja)
IE (1) IE43567B1 (ja)
IL (1) IL48389A (ja)
IN (2) IN141710B (ja)
LU (2) LU73849A1 (ja)
NL (1) NL165741C (ja)
NO (2) NO143578C (ja)
SE (2) SE421619B (ja)
SU (3) SU569290A3 (ja)
YU (1) YU37328B (ja)
ZA (1) ZA756792B (ja)

Families Citing this family (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4075343A (en) * 1976-09-13 1978-02-21 Pfizer Inc. Anti-allergenic 5-alkoxyimidazo[1,2-A]quinoline-2-carboxylic acids and derivatives thereof
GR70248B (ja) * 1978-10-30 1982-09-01 Lepetit Spa
US4313950A (en) * 1978-10-30 1982-02-02 Gruppo Lepetit S.P.A. Antireproductive tricyclic ortho-fused nitrogen containing compounds
DE2964567D1 (en) * 1978-12-21 1983-02-24 Lepetit Spa New 3h-naphtho(1,2-d)imidazoles, processes for preparing them, compounds for use as antiinflammatory and antimicrobial agents and compositions for that use containing them
US4644002A (en) * 1979-02-09 1987-02-17 Roussel Uclaf Imidazo[2,1-C]quinolines, useful as antiallergic agents
IT1150955B (it) * 1980-06-06 1986-12-17 Lepetit Spa Derivati 3h-naft(1.2-d)-imidazolici il procedimento per la loro preparazione, il loro uso come agenti antiinfiammatori e le composizioni farmaceutiche che li contengono
DE3314843A1 (de) * 1983-04-23 1984-10-25 Beiersdorf Ag, 2000 Hamburg 1-amidino-2,3,3a,8-tetrahydro-1h-pyrazolo (5,1-a)isoindol, verfahren zu dessen herstellung, diese verbindung enthaltende zubereitungen und zwischenprodukte
GB8415540D0 (en) * 1984-06-18 1984-07-25 Fujisawa Pharmaceutical Co Imidazoisoquinoline compounds
EP0607076A1 (fr) * 1993-01-15 1994-07-20 Synthelabo Dérivés de 9h-imidazo 1,2-a benzimidazole-3-acétamide à activité GABA
JP3332929B2 (ja) * 1995-02-15 2002-10-07 ニューロゲン コーポレイション ある種の架橋4−フェニル−2−アミノメチルイミダゾール:新しいドパミン受容体サブタイプ特異的リガンド
US5948912A (en) * 1995-02-15 1999-09-07 Neurogen Corporation Certain bridged 4-phenyl-2-aminomethylimidazoles; new dopamine receptor subtype specific ligands
TW416953B (en) 1996-09-25 2001-01-01 Takeda Chemical Industries Ltd Tricyclic compounds for eliciting a prostaglandin I2 receptor agonistic effect, their production and use
WO2002088092A1 (fr) * 2001-04-19 2002-11-07 Eisai Co., Ltd. Derive de 2-imino-imidazole (2)
WO2002098863A1 (fr) * 2001-06-05 2002-12-12 Fujisawa Pharmaceutical Co., Ltd. Derive d'imidazole fondu
CA2515715C (en) * 2003-02-19 2012-05-08 Eisai Co., Ltd. Methods for producing cyclic benzamidine derivatives
AU2005287170B2 (en) * 2004-09-17 2012-03-29 Exelixis, Inc Pyrazole kinase modulators and methods of use
US11142504B2 (en) 2016-03-07 2021-10-12 Northwestern University Substituted heterocycles as c-MYC targeting agents
WO2017155942A2 (en) * 2016-03-07 2017-09-14 Northwestern University Substituted heterocycles as c-myc targeting agents
US11420957B2 (en) 2019-06-17 2022-08-23 Northwestern University Substituted heterocycles as c-MYC targeting agents
CN110294758B (zh) * 2019-07-06 2021-10-22 湘潭大学 2-取代5,6-二氢吡唑并[5,1-α]异喹啉、衍生物及其合成方法

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1244501A (en) * 1968-03-09 1971-09-02 Aspro Nicholas Ltd Heterocyclic amines
GB1347493A (en) * 1971-02-11 1974-02-27 Aspro Nicholas Ltd Benzazine derivatives

Also Published As

Publication number Publication date
DK152756C (da) 1988-09-26
NL165741C (nl) 1981-05-15
NL7512848A (nl) 1976-05-25
DK522175A (da) 1976-05-24
BE835836A (fr) 1976-03-16
SU582764A3 (ru) 1977-11-30
SU578883A3 (ru) 1977-10-30
NO753854L (ja) 1976-05-25
NO143577B (no) 1980-12-01
DK522275A (da) 1976-05-24
NL165741B (nl) 1980-12-15
JPS5516513B2 (ja) 1980-05-02
DD122819A5 (ja) 1976-11-05
JPS5175098A (ja) 1976-06-29
DK152756B (da) 1988-05-09
AR209459A1 (es) 1977-04-29
SU569290A3 (ru) 1977-08-15
CH614208A5 (ja) 1979-11-15
ZA756792B (en) 1976-10-27
CA1068273A (en) 1979-12-18
FR2291747A1 (fr) 1976-06-18
ATA884575A (de) 1977-11-15
NO143578B (no) 1980-12-01
GR58293B (en) 1977-09-20
YU292775A (en) 1983-04-27
SE421620B (sv) 1982-01-18
US4075342A (en) 1978-02-21
AT346332B (de) 1978-11-10
FI58919C (fi) 1981-05-11
ES442863A1 (es) 1977-08-16
GR58292B (en) 1977-09-20
LU73849A1 (ja) 1976-06-11
CH614444A5 (ja) 1979-11-30
GB1484615A (en) 1977-09-01
SE7513137L (sv) 1976-05-24
IN141710B (ja) 1977-04-09
IN142014B (ja) 1977-05-21
FI58919B (fi) 1981-01-30
YU37328B (en) 1984-08-31
ES442864A1 (es) 1977-08-16
FI753046A (ja) 1976-05-24
NO753853L (ja) 1976-05-25
NO143577C (no) 1981-03-11
LU73850A1 (ja) 1976-06-11
FR2291747B1 (ja) 1978-11-17
SE7513138L (sv) 1976-05-24
CA1068274A (en) 1979-12-18
IL48389A (en) 1979-01-31
IL48389A0 (en) 1975-12-31
AT344176B (de) 1978-07-10
DE2551868A1 (de) 1976-08-12
FI58918B (fi) 1981-01-30
AR210476A1 (es) 1977-08-15
IE43567B1 (en) 1981-04-08
AU8620475A (en) 1977-05-05
IE43567L (en) 1976-05-23
FI58918C (fi) 1981-05-11
ATA884675A (de) 1978-03-15
DE2551868C2 (de) 1982-07-15
DD122818A5 (ja) 1976-11-05
SE421619B (sv) 1982-01-18
NO143578C (no) 1981-03-11

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Legal Events

Date Code Title Description
MM Patent lapsed

Owner name: GRUPPO LEPETIT S.P.A.