FI70574C - Foerfarande foer framstaellning av nya farmaceutiskt anvaendbara derivat av 2-7(4-kinolinyl)-amino/-5-fluorbensoesyra - Google Patents

Foerfarande foer framstaellning av nya farmaceutiskt anvaendbara derivat av 2-7(4-kinolinyl)-amino/-5-fluorbensoesyra Download PDF

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Publication number
FI70574C
FI70574C FI783833A FI783833A FI70574C FI 70574 C FI70574 C FI 70574C FI 783833 A FI783833 A FI 783833A FI 783833 A FI783833 A FI 783833A FI 70574 C FI70574 C FI 70574C
Authority
FI
Finland
Prior art keywords
trifluoromethyl
quinolinylamino
acid
ester
fluoro
Prior art date
Application number
FI783833A
Other languages
English (en)
Finnish (fi)
Swedish (sv)
Other versions
FI783833A (fi
FI70574B (fi
Inventor
Andre Allais
Jean Meier
Roger Deraedt
Original Assignee
Roussel Uclaf
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from FR7737836A external-priority patent/FR2411833A1/fr
Priority claimed from FR7737835A external-priority patent/FR2411832A1/fr
Application filed by Roussel Uclaf filed Critical Roussel Uclaf
Publication of FI783833A publication Critical patent/FI783833A/fi
Application granted granted Critical
Publication of FI70574B publication Critical patent/FI70574B/fi
Publication of FI70574C publication Critical patent/FI70574C/fi

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/38—Nitrogen atoms
    • C07D215/42—Nitrogen atoms attached in position 4
    • C07D215/44—Nitrogen atoms attached in position 4 with aryl radicals attached to said nitrogen atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A61P29/02—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID] without antiinflammatory effect

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Pain & Pain Management (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Rheumatology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Quinoline Compounds (AREA)
FI783833A 1977-12-15 1978-12-13 Foerfarande foer framstaellning av nya farmaceutiskt anvaendbara derivat av 2-7(4-kinolinyl)-amino/-5-fluorbensoesyra FI70574C (fi)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
FR7737836 1977-12-15
FR7737836A FR2411833A1 (fr) 1977-12-15 1977-12-15 Nouveaux derives de l'acide 2(/4-quinoleinyl/amino) 5-fluoro benzoique, leur procede de preparation et leur application comme medicament
FR7737835 1977-12-15
FR7737835A FR2411832A1 (fr) 1977-12-15 1977-12-15 Nouveaux derives de l'acide 2/(4-quinoleinyl) amino/5-fluorobenzoique, leur procede de preparation et leur application comme medicament.

Publications (3)

Publication Number Publication Date
FI783833A FI783833A (fi) 1979-06-16
FI70574B FI70574B (fi) 1986-06-06
FI70574C true FI70574C (fi) 1986-09-24

Family

ID=26220343

Family Applications (1)

Application Number Title Priority Date Filing Date
FI783833A FI70574C (fi) 1977-12-15 1978-12-13 Foerfarande foer framstaellning av nya farmaceutiskt anvaendbara derivat av 2-7(4-kinolinyl)-amino/-5-fluorbensoesyra

Country Status (21)

Country Link
US (1) US4233305A (fr)
JP (1) JPS5488277A (fr)
AR (1) AR224116A1 (fr)
AT (1) AT365578B (fr)
AU (1) AU520983B2 (fr)
CA (1) CA1115276A (fr)
CH (1) CH636350A5 (fr)
DE (1) DE2854341A1 (fr)
DK (1) DK149845C (fr)
ES (1) ES475686A1 (fr)
FI (1) FI70574C (fr)
GB (1) GB2010243B (fr)
HU (1) HU177031B (fr)
IE (1) IE47618B1 (fr)
IL (1) IL56156A (fr)
IT (1) IT1107671B (fr)
LU (1) LU80660A1 (fr)
NL (1) NL7812206A (fr)
PT (1) PT68916A (fr)
SE (1) SE448091B (fr)
SU (1) SU837322A3 (fr)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS6322584A (ja) * 1986-07-15 1988-01-30 Senjiyu Seiyaku Kk １−ハイドロキシ−５−オキソ−５Ｈ−ピリド〔３，２−ａ〕フエノキサジン−３−カルボン酸エステル類
IL89029A (en) * 1988-01-29 1993-01-31 Lilly Co Eli Fungicidal quinoline and cinnoline derivatives, compositions containing them, and fungicidal methods of using them

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3232944A (en) * 1966-02-01 Monoglycerides 0f (carbgxy pl-ienyl amtno) chlgroqukngltnes
CH408915A (fr) * 1962-02-16 1966-03-15 Roussel Uclaf Procédé de préparation d'un nouveau composé utilisable, notamment, pour le traitement des manifestations inflammatoires et/ou douloureuses
CA731646A (en) * 1962-05-08 1966-04-05 Roussel-Uclaf 4-(2'(.beta.-MORPHOLYLETHOXYCARBONYL) PHENYLAMINE) 7-CHLORO QUINOLEINE ET SES SELS, AINSI QUE LEUR PROCEDE DE PREPARATION
FR6935M (fr) * 1967-12-29 1969-05-05
FR7870M (fr) * 1968-11-08 1970-04-27
ZA726593B (en) * 1971-10-19 1973-06-27 Abbott Lab Novel derivatives of 2,3-dihydroxypropyl-n-(7 or 8-chloro-4-quinolinyl)anthranilate
CH585221A5 (fr) * 1972-07-28 1977-02-28 Synthelabo
US3971789A (en) * 1972-10-21 1976-07-27 John Wyeth & Brother Limited O-(4-Quinolylamino)benzamides
FR2233059B1 (fr) * 1973-06-13 1976-09-03 Roussel Uclaf
GB1474296A (en) * 1975-01-23 1977-05-18 Wyeth John & Brother Ltd 4-aminoquinoline derivatives

Also Published As

Publication number Publication date
IT7852296A0 (it) 1978-12-14
LU80660A1 (fr) 1979-07-20
HU177031B (hu) 1981-06-28
GB2010243A (en) 1979-06-27
SE448091B (sv) 1987-01-19
IE47618B1 (en) 1984-05-02
CH636350A5 (fr) 1983-05-31
AU4252878A (en) 1979-06-21
ATA897378A (de) 1981-06-15
FI783833A (fi) 1979-06-16
IE782476L (en) 1979-06-15
IL56156A0 (en) 1979-03-12
DK149845B (da) 1986-10-13
DE2854341C2 (fr) 1990-05-23
DK149845C (da) 1987-03-02
ES475686A1 (es) 1979-04-16
DE2854341A1 (de) 1979-06-28
SE7811839L (sv) 1979-06-16
US4233305A (en) 1980-11-11
IL56156A (en) 1984-11-30
AR224116A1 (es) 1981-10-30
JPS631305B2 (fr) 1988-01-12
NL7812206A (nl) 1979-06-19
AU520983B2 (en) 1982-03-11
IT1107671B (it) 1985-11-25
AT365578B (de) 1982-01-25
JPS5488277A (en) 1979-07-13
GB2010243B (en) 1982-05-19
PT68916A (fr) 1979-01-01
CA1115276A (fr) 1981-12-29
DK561278A (da) 1979-06-16
FI70574B (fi) 1986-06-06
SU837322A3 (ru) 1981-06-07

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Owner name: ROUSSEL UCLAF SOCIETE ANONYME