FI70220C - Foerfarande foer framstaellning av en ny som antibakteriellt medel anvaendbara alfa-substituerad ureidobensylpenicillansyra - Google Patents

Foerfarande foer framstaellning av en ny som antibakteriellt medel anvaendbara alfa-substituerad ureidobensylpenicillansyra Download PDF

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Publication number
FI70220C
FI70220C FI812395A FI812395A FI70220C FI 70220 C FI70220 C FI 70220C FI 812395 A FI812395 A FI 812395A FI 812395 A FI812395 A FI 812395A FI 70220 C FI70220 C FI 70220C
Authority
FI
Finland
Prior art keywords
acid
formula
group
compound
conh
Prior art date
Application number
FI812395A
Other languages
English (en)
Finnish (fi)
Swedish (sv)
Other versions
FI70220B (fi
FI812395L (fi
Inventor
Nobuhiro Oi
Bunya Aoki
Teizo Shinozaki
Kanji Moro
Toshio Kuroki
Isao Matsunaga
Takao Nato
Toshiyuki Nebashi
Yusuke Harada
Hisao Endo
Takao Kimura
Kana Kojima
Masahiko Matsumoto
Hirohi Okazaki
Haruki Ogawa
Minoru Shindo
Original Assignee
Chugai Pharmaceutical Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Chugai Pharmaceutical Co Ltd filed Critical Chugai Pharmaceutical Co Ltd
Publication of FI812395L publication Critical patent/FI812395L/fi
Application granted granted Critical
Publication of FI70220B publication Critical patent/FI70220B/fi
Publication of FI70220C publication Critical patent/FI70220C/fi

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D499/00Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D499/21Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with a nitrogen atom directly attached in position 6 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
    • C07D499/44Compounds with an amino radical acylated by carboxylic acids, attached in position 6
    • C07D499/48Compounds with an amino radical acylated by carboxylic acids, attached in position 6 with a carbon chain, substituted by hetero atoms or by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, attached to the carboxamido radical
    • C07D499/58Compounds with an amino radical acylated by carboxylic acids, attached in position 6 with a carbon chain, substituted by hetero atoms or by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, attached to the carboxamido radical substituted in alpha-position to the carboxamido radical
    • C07D499/64Compounds with an amino radical acylated by carboxylic acids, attached in position 6 with a carbon chain, substituted by hetero atoms or by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, attached to the carboxamido radical substituted in alpha-position to the carboxamido radical by nitrogen atoms
    • C07D499/68Compounds with an amino radical acylated by carboxylic acids, attached in position 6 with a carbon chain, substituted by hetero atoms or by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, attached to the carboxamido radical substituted in alpha-position to the carboxamido radical by nitrogen atoms with aromatic rings as additional substituents on the carbon chain
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D499/00Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Cephalosporin Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Measuring Or Testing Involving Enzymes Or Micro-Organisms (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
FI812395A 1980-08-05 1981-07-31 Foerfarande foer framstaellning av en ny som antibakteriellt medel anvaendbara alfa-substituerad ureidobensylpenicillansyra FI70220C (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP10677580A JPS5732289A (en) 1980-08-05 1980-08-05 Alpha-substituted ureidobenzylpenicillin
JP10677580 1980-08-05

Publications (3)

Publication Number Publication Date
FI812395L FI812395L (fi) 1982-02-06
FI70220B FI70220B (fi) 1986-02-28
FI70220C true FI70220C (fi) 1986-09-15

Family

ID=14442271

Family Applications (1)

Application Number Title Priority Date Filing Date
FI812395A FI70220C (fi) 1980-08-05 1981-07-31 Foerfarande foer framstaellning av en ny som antibakteriellt medel anvaendbara alfa-substituerad ureidobensylpenicillansyra

Country Status (14)

Country Link
US (1) US4355038A (ru)
EP (1) EP0045523B1 (ru)
JP (1) JPS5732289A (ru)
KR (2) KR850000049B1 (ru)
AT (1) ATE10635T1 (ru)
AU (1) AU542522B2 (ru)
CA (1) CA1203530A (ru)
DE (1) DE3167610D1 (ru)
DK (1) DK159272C (ru)
FI (1) FI70220C (ru)
IL (1) IL63456A (ru)
MX (1) MX6943E (ru)
NO (1) NO158300C (ru)
ZA (1) ZA815222B (ru)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5810585A (ja) * 1981-07-10 1983-01-21 Chugai Pharmaceut Co Ltd α−置換ウレイドベンジルペニシラン酸
GB2168975A (en) * 1984-12-20 1986-07-02 Procter & Gamble Amides and compositions thereof having anti-inflammatory and analgesic activity
JPH06159622A (ja) * 1992-11-19 1994-06-07 Miura Kenkyusho:Kk 燃焼ガス自己循環式気化燃焼バーナ

Family Cites Families (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1250611A (ru) 1968-02-03 1971-10-20
IE32700B1 (en) 1968-02-03 1973-10-31 Beecham Group Ltd Penicillins
DE1770620A1 (de) 1968-06-12 1971-11-11 Bayer Ag Neue Penicilline
US3933795A (en) * 1970-05-25 1976-01-20 Hans-Bodo Konig Ureidoacetamido-penicillins
US3980792A (en) * 1970-05-25 1976-09-14 Bayer Aktiengesellschaft Ureidoacetamido-penicillins
US3959258A (en) * 1970-05-25 1976-05-25 Bayer Aktiengesellschaft Ureidoacetamido-penicillins
US3978223A (en) * 1970-05-25 1976-08-31 Bayer Aktiengesellschaft Ureidoacetamido-penicillins for treating bacterial infections
US4016282A (en) * 1970-05-25 1977-04-05 Bayer Aktiengesellschaft Ureidoacetamido-penicillins
CH562249A5 (ru) 1970-05-25 1975-05-30 Bayer Ag
US3936442A (en) * 1970-05-25 1976-02-03 Bayer Aktiengesellschaft Unreidoacetamido-penicilins
US3974140A (en) * 1970-05-25 1976-08-10 Bayer Aktiengesellschaft Ureidoacetamido-penicillins
US3939149A (en) * 1970-05-25 1976-02-17 Bayer Aktiengesellschaft Ureidoacetamido-penicillins
GB1433131A (en) 1972-03-13 1976-04-22 Astra Laekemedel Ab Penicillins
DE2258973A1 (de) 1972-12-01 1974-06-06 Bayer Ag Penicilline, verfahren zu ihrer herstellung sowie ihre verwendung als arzneimittel
GB1562802A (en) 1976-06-26 1980-03-19 Beecham Group Ltd Pharmaceutical compositions containing containing clavulanic acid
JPS5524135A (en) * 1978-08-11 1980-02-21 Chugai Pharmaceut Co Ltd Penicillin derivative and its preparation
CA1133896A (en) * 1978-05-26 1982-10-19 Nobuhiro Oi Penicillanic acid derivative and process for preparing the same
JPS54163590A (en) * 1978-06-13 1979-12-26 Chugai Pharmaceutical Co Ltd Penicilunic acid derivative and salt thereof
JPS54154782A (en) * 1978-05-26 1979-12-06 Chugai Pharmaceut Co Ltd Penicillin derivative and its salt
JPS5583789A (en) 1978-12-18 1980-06-24 Bristol Myers Co Preparation of penicillin
US4240960A (en) * 1979-03-19 1980-12-23 Bristol-Myers Company Trimethylsilyl substituted penicillins

Also Published As

Publication number Publication date
CA1203530A (en) 1986-04-22
NO158300B (no) 1988-05-09
DK159272B (da) 1990-09-24
ZA815222B (en) 1982-08-25
ATE10635T1 (de) 1984-12-15
MX6943E (es) 1986-12-17
KR850000049B1 (ko) 1985-02-14
AU7354981A (en) 1982-02-11
KR830006306A (ko) 1983-09-20
NO158300C (no) 1988-08-17
EP0045523A1 (en) 1982-02-10
US4355038A (en) 1982-10-19
JPS5732289A (en) 1982-02-20
DK159272C (da) 1991-02-18
EP0045523B1 (en) 1984-12-05
AU542522B2 (en) 1985-02-21
IL63456A0 (en) 1981-10-30
FI70220B (fi) 1986-02-28
KR850000048B1 (ko) 1985-02-14
NO812630L (no) 1982-02-08
DK343481A (da) 1982-02-06
IL63456A (en) 1984-12-31
JPH0118916B2 (ru) 1989-04-07
FI812395L (fi) 1982-02-06
DE3167610D1 (en) 1985-01-17

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Owner name: CHUGAI SEIYAKU KABUSHIKI KAISHA