FI66380C - Foerfarande foer framstaellning av nya antireproduktiva 1,2,4-triazolo(5,1-a)isoindoler -isokinoliner och -bensazepiner - Google Patents
Foerfarande foer framstaellning av nya antireproduktiva 1,2,4-triazolo(5,1-a)isoindoler -isokinoliner och -bensazepiner Download PDFInfo
- Publication number
- FI66380C FI66380C FI793215A FI793215A FI66380C FI 66380 C FI66380 C FI 66380C FI 793215 A FI793215 A FI 793215A FI 793215 A FI793215 A FI 793215A FI 66380 C FI66380 C FI 66380C
- Authority
- FI
- Finland
- Prior art keywords
- compounds
- triazolo
- compound
- formula
- antireproductive
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D223/00—Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom
- C07D223/14—Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
- C07D223/16—Benzazepines; Hydrogenated benzazepines
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D217/00—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems
- C07D217/22—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the nitrogen-containing ring
- C07D217/24—Oxygen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Tropical Medicine & Parasitology (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Applications Claiming Priority (4)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GB7842415 | 1978-10-30 | ||
GB7842415 | 1978-10-30 | ||
US06/087,371 US4275066A (en) | 1978-10-30 | 1979-10-23 | Antireproductive tricyclic ortho-fused nitrogen containing compounds |
US8737179 | 1979-10-23 |
Publications (3)
Publication Number | Publication Date |
---|---|
FI793215A FI793215A (fi) | 1980-05-01 |
FI66380B FI66380B (fi) | 1984-06-29 |
FI66380C true FI66380C (fi) | 1984-10-10 |
Family
ID=26269380
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
FI793215A FI66380C (fi) | 1978-10-30 | 1979-10-16 | Foerfarande foer framstaellning av nya antireproduktiva 1,2,4-triazolo(5,1-a)isoindoler -isokinoliner och -bensazepiner |
Country Status (18)
Country | Link |
---|---|
US (1) | US4275066A (de) |
JP (1) | JPS5562086A (de) |
AT (2) | AT374803B (de) |
AU (1) | AU532045B2 (de) |
BE (1) | BE879729A (de) |
CA (1) | CA1123827A (de) |
CH (1) | CH650261A5 (de) |
DE (1) | DE2943286A1 (de) |
DK (1) | DK154298C (de) |
FI (1) | FI66380C (de) |
FR (1) | FR2440370A1 (de) |
GB (1) | GB2039888B (de) |
GR (1) | GR70248B (de) |
HK (1) | HK24383A (de) |
IE (1) | IE49625B1 (de) |
LU (1) | LU81833A1 (de) |
NL (1) | NL7907783A (de) |
ZA (1) | ZA795743B (de) |
Families Citing this family (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CA1211437A (en) * | 1981-08-12 | 1986-09-16 | Rene Borer | Benzazepines |
US5302589A (en) * | 1992-08-07 | 1994-04-12 | Glaxo, Inc. | Heterocyclic inhibitors of 5-α-testosterone reductase |
CN100432074C (zh) * | 2006-06-29 | 2008-11-12 | 浙江大学 | 2-芳基咪唑并[2,1-a]异喹啉的合成方法 |
JP5412809B2 (ja) * | 2008-11-21 | 2014-02-12 | コニカミノルタ株式会社 | イミダゾール化合物の製造方法 |
RU2657832C1 (ru) * | 2017-06-07 | 2018-06-15 | федеральное государственное автономное образовательное учреждение высшего образования "Южный федеральный университет" | Антидиабетическое средство |
Family Cites Families (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3758480A (en) * | 1968-07-10 | 1973-09-11 | Mallinckrodt Chemical Works | S-triazolo(5,1-a)isoquinolines and derivatives thereof |
US3775417A (en) * | 1971-08-05 | 1973-11-27 | Mallinckrodt Chemical Works | Selective hydrogenation of tri-and tetrazoloisoquinolines |
GB1477302A (en) * | 1973-05-25 | 1977-06-22 | Lepetit Spa | Triazolo-isoindole and triazolo-isoquinoline derivatives and their manufacture and uses |
RO66059A (ro) * | 1973-05-25 | 1981-05-30 | Gruppo Lepetit Spa,It | Procedeu de obtinere a unor derivati de triazolochinoline |
US4075341A (en) * | 1974-05-24 | 1978-02-21 | Gruppo Lepetit S.P.A. | 2-Substituted phenyl-5-triazols [5,1-a] isoquinoline compounds |
GB1484615A (en) * | 1974-11-23 | 1977-09-01 | Lepetit Spa | Tricyclic n-containing derivatives |
IT1054655B (it) * | 1975-08-27 | 1981-11-30 | Lepetit Spa | Derivati condensati del l isochinolina |
DE2707272C2 (de) * | 1977-02-19 | 1982-12-02 | Gruppo Lepetit S.p.A., 20158 Milano | 2-(p-Chlorphenyl)-s-triazolo [5,1-a] isochinolin |
US4093728A (en) * | 1977-08-18 | 1978-06-06 | E. R. Squibb & Sons, Inc. | Triazoloisoindoles |
-
1979
- 1979-10-13 GR GR60257A patent/GR70248B/el unknown
- 1979-10-16 FI FI793215A patent/FI66380C/fi not_active IP Right Cessation
- 1979-10-18 AU AU51908/79A patent/AU532045B2/en not_active Ceased
- 1979-10-23 NL NL7907783A patent/NL7907783A/nl not_active Application Discontinuation
- 1979-10-23 US US06/087,371 patent/US4275066A/en not_active Expired - Lifetime
- 1979-10-26 DK DK452779A patent/DK154298C/da not_active IP Right Cessation
- 1979-10-26 IE IE2067/79A patent/IE49625B1/en unknown
- 1979-10-26 DE DE19792943286 patent/DE2943286A1/de active Granted
- 1979-10-26 ZA ZA00795743A patent/ZA795743B/xx unknown
- 1979-10-29 JP JP13971079A patent/JPS5562086A/ja active Granted
- 1979-10-29 LU LU81833A patent/LU81833A1/fr unknown
- 1979-10-29 GB GB7937388A patent/GB2039888B/en not_active Expired
- 1979-10-29 AT AT0697179A patent/AT374803B/de not_active IP Right Cessation
- 1979-10-29 CH CH9672/79A patent/CH650261A5/it not_active IP Right Cessation
- 1979-10-30 FR FR7926902A patent/FR2440370A1/fr active Granted
- 1979-10-30 CA CA338,698A patent/CA1123827A/en not_active Expired
- 1979-10-30 BE BE0/197894A patent/BE879729A/fr not_active IP Right Cessation
-
1983
- 1983-06-20 AT AT0226083A patent/AT384427B/de not_active IP Right Cessation
- 1983-07-28 HK HK243/83A patent/HK24383A/xx unknown
Also Published As
Publication number | Publication date |
---|---|
FI66380B (fi) | 1984-06-29 |
DE2943286C2 (de) | 1990-05-23 |
ATA697179A (de) | 1983-10-15 |
FI793215A (fi) | 1980-05-01 |
GR70248B (de) | 1982-09-01 |
LU81833A1 (fr) | 1980-05-07 |
AT374803B (de) | 1984-06-12 |
GB2039888B (en) | 1982-11-03 |
ZA795743B (en) | 1980-10-29 |
CA1123827A (en) | 1982-05-18 |
CH650261A5 (it) | 1985-07-15 |
AU532045B2 (en) | 1983-09-15 |
DK154298C (da) | 1989-03-28 |
ATA226083A (de) | 1987-04-15 |
BE879729A (fr) | 1980-04-30 |
US4275066A (en) | 1981-06-23 |
IE49625B1 (en) | 1985-11-13 |
GB2039888A (en) | 1980-08-20 |
JPS6354716B2 (de) | 1988-10-28 |
FR2440370A1 (fr) | 1980-05-30 |
DK154298B (da) | 1988-10-31 |
DE2943286A1 (de) | 1980-05-14 |
IE792067L (en) | 1980-04-30 |
AU5190879A (en) | 1980-05-08 |
AT384427B (de) | 1987-11-10 |
FR2440370B1 (de) | 1982-10-29 |
DK452779A (da) | 1980-05-01 |
HK24383A (en) | 1983-08-05 |
NL7907783A (nl) | 1980-05-02 |
JPS5562086A (en) | 1980-05-10 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
MM | Patent lapsed |
Owner name: GRUPPO LEPETIT S.P.A. |