FI65250C - Foerfarande foer framstaellning av terapeutiskt anvaendbara 3-cetyl-1,2,3,3a,4,5,6,7-oktahydro-3,6,7a-triaza-syklohepta (j)fluorenderivat - Google Patents

Foerfarande foer framstaellning av terapeutiskt anvaendbara 3-cetyl-1,2,3,3a,4,5,6,7-oktahydro-3,6,7a-triaza-syklohepta (j)fluorenderivat Download PDF

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Publication number
FI65250C
FI65250C FI792366A FI792366A FI65250C FI 65250 C FI65250 C FI 65250C FI 792366 A FI792366 A FI 792366A FI 792366 A FI792366 A FI 792366A FI 65250 C FI65250 C FI 65250C
Authority
FI
Finland
Prior art keywords
alkyl
octahydro
compound
compounds
therapeutic
Prior art date
Application number
FI792366A
Other languages
English (en)
Finnish (fi)
Other versions
FI65250B (fi
FI792366A7 (fi
Inventor
Regis Dupont
Patrick Lardenois
Claude Morel
Jonathan Frost
Gabor Istvan Koletar
Original Assignee
Synthelabo
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from FR7822352A external-priority patent/FR2432025A1/fr
Priority claimed from FR7822353A external-priority patent/FR2432026A1/fr
Application filed by Synthelabo filed Critical Synthelabo
Publication of FI792366A7 publication Critical patent/FI792366A7/fi
Publication of FI65250B publication Critical patent/FI65250B/fi
Application granted granted Critical
Publication of FI65250C publication Critical patent/FI65250C/fi

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
    • C07D471/14—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Steroid Compounds (AREA)
  • Medicinal Preparation (AREA)
FI792366A 1978-07-28 1979-07-27 Foerfarande foer framstaellning av terapeutiskt anvaendbara 3-cetyl-1,2,3,3a,4,5,6,7-oktahydro-3,6,7a-triaza-syklohepta (j)fluorenderivat FI65250C (fi)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
FR7822353 1978-07-28
FR7822352 1978-07-28
FR7822352A FR2432025A1 (fr) 1978-07-28 1978-07-28 Derives d'imidazo et de pyrimido-pyrido-indoles, leur preparation et leur application en therapeutique
FR7822353A FR2432026A1 (fr) 1978-07-28 1978-07-28 Derives de fluorenes et de fluoranthenes et leur application en therapeutique

Publications (3)

Publication Number Publication Date
FI792366A7 FI792366A7 (fi) 1980-01-29
FI65250B FI65250B (fi) 1983-12-30
FI65250C true FI65250C (fi) 1984-04-10

Family

ID=26220699

Family Applications (1)

Application Number Title Priority Date Filing Date
FI792366A FI65250C (fi) 1978-07-28 1979-07-27 Foerfarande foer framstaellning av terapeutiskt anvaendbara 3-cetyl-1,2,3,3a,4,5,6,7-oktahydro-3,6,7a-triaza-syklohepta (j)fluorenderivat

Country Status (13)

Country Link
US (1) US4277476A (https=)
EP (1) EP0008249B1 (https=)
AT (1) ATE165T1 (https=)
AU (1) AU524307B2 (https=)
CA (1) CA1107729A (https=)
DE (1) DE2960689D1 (https=)
DK (1) DK316279A (https=)
ES (1) ES482889A1 (https=)
FI (1) FI65250C (https=)
GR (1) GR75070B (https=)
NO (1) NO792476L (https=)
NZ (1) NZ191141A (https=)
PT (1) PT69988A (https=)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2455044A1 (fr) * 1979-04-26 1980-11-21 Synthelabo Pyrido-indoles et leur application en therapeutique
US4367230A (en) * 1980-01-04 1983-01-04 Tanabe Seiyaku Co., Ltd. Novel triazafluoranthene compound and processes for preparing the same
US4428880A (en) 1981-05-04 1984-01-31 S.A. Omnichem Azepino[4,5-d]indole derivatives and preparation thereof
GB2184685B (en) * 1985-12-19 1989-10-11 Braas & Co Gmbh Plastically deformable sheet material
JP4202250B2 (ja) 2001-07-25 2008-12-24 バイオマリン ファーマシューティカル インコーポレイテッド 血液脳関門輸送を調節するための組成物および方法
US7767689B2 (en) 2004-03-15 2010-08-03 Ptc Therapeutics, Inc. Carboline derivatives useful in the treatment of cancer
MXPA06010543A (es) 2004-03-15 2007-03-26 Ptc Therapeutics Inc Derivados de carbolina utiles en la inhibicion de la angiogenesis.
US8076352B2 (en) 2004-03-15 2011-12-13 Ptc Therapeutics, Inc. Administration of carboline derivatives useful in the treatment of cancer and other diseases
US8076353B2 (en) 2004-03-15 2011-12-13 Ptc Therapeutics, Inc. Inhibition of VEGF translation
EP2671507A3 (en) 2005-04-28 2014-02-19 Proteus Digital Health, Inc. Pharma-informatics system
MX2009002893A (es) 2006-09-18 2009-07-10 Raptor Pharmaceutical Inc Tratamiento de trastornos hepaticos mediante la administracion de conjugados de la proteina asociada al receptor (rap).
CA2752373C (en) 2009-02-20 2017-10-10 To-Bbb Holding B.V. Glutathione-based drug delivery system
IL255113B (en) 2009-05-06 2022-09-01 Laboratory Skin Care Inc Dermal delivery compositions comprising active agent-calcium phosphate particle complexes and methods of using the same
US20120077778A1 (en) 2010-09-29 2012-03-29 Andrea Bourdelais Ladder-Frame Polyether Conjugates

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2556574A (en) * 1949-06-24 1951-06-12 Allen & Hanburys Ltd Indolopteridines and process for preparing same
US3108108A (en) * 1959-09-25 1963-10-22 Bayer Ag Aza analogues of polynuclear o-quinones
US3122544A (en) * 1962-11-13 1964-02-25 American Home Prod 4-amino-2-aryl-6h-indeno(2, 3-g)-pteridin-6-ones
US3470181A (en) * 1967-10-23 1969-09-30 American Home Prod Fused 2-pyrimidinepropionic acid compounds,related compounds,and the process for their preparation
US3631046A (en) * 1969-05-28 1971-12-28 Sandoz Ag Tetracyclic quinazolin-ones
BE759337A (fr) * 1969-11-24 1971-05-24 Lilly Co Eli Benzimidazol (2,1-b)-quinazolin (6h) ones qui sont des immuno-depresseurs, et nouvelles benzimidazo (2,1-b) quinazolin-12-(6h) ones
US3963720A (en) * 1972-10-27 1976-06-15 Sandoz, Inc. Tetracyclic imidazo [2,1-b] quinazolinone derivatives
CH601299A5 (en) * 1973-11-07 1978-07-14 Vni Khim Farmatsevtichesky I I Pyrazino(1,2,3-ab)beta carbolines and homologues

Also Published As

Publication number Publication date
FI65250B (fi) 1983-12-30
ES482889A1 (es) 1980-04-16
ATE165T1 (de) 1981-09-15
EP0008249B1 (fr) 1981-08-26
CA1107729A (en) 1981-08-25
PT69988A (fr) 1979-08-01
US4277476A (en) 1981-07-07
DK316279A (da) 1980-01-29
AU524307B2 (en) 1982-09-09
AU4927879A (en) 1980-01-31
NO792476L (no) 1980-01-29
FI792366A7 (fi) 1980-01-29
EP0008249A3 (en) 1980-05-14
DE2960689D1 (en) 1981-11-19
EP0008249A2 (fr) 1980-02-20
GR75070B (https=) 1984-07-13
NZ191141A (en) 1983-02-15

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Owner name: SYNTHELABO