FI64576C - Foerfarande foer framstaellning av en terapeutiskt anvaendbar somatostatinanalog - Google Patents
Foerfarande foer framstaellning av en terapeutiskt anvaendbar somatostatinanalog Download PDFInfo
- Publication number
- FI64576C FI64576C FI781184A FI781184A FI64576C FI 64576 C FI64576 C FI 64576C FI 781184 A FI781184 A FI 781184A FI 781184 A FI781184 A FI 781184A FI 64576 C FI64576 C FI 64576C
- Authority
- FI
- Finland
- Prior art keywords
- resin
- acid
- somatostatin
- minutes
- val
- Prior art date
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- 239000011975 tartaric acid Substances 0.000 description 1
- 235000002906 tartaric acid Nutrition 0.000 description 1
- 125000000999 tert-butyl group Chemical group [H]C([H])([H])C(*)(C([H])([H])[H])C([H])([H])[H] 0.000 description 1
- 125000005931 tert-butyloxycarbonyl group Chemical group [H]C([H])([H])C(OC(*)=O)(C([H])([H])[H])C([H])([H])[H] 0.000 description 1
- 150000003512 tertiary amines Chemical class 0.000 description 1
- RGYLYUZOGHTBRF-BIHRQFPBSA-N tetragastrin Chemical compound C([C@H](NC(=O)[C@H](CC(O)=O)NC(=O)[C@@H](NC(=O)[C@@H](N)CC=1C2=CC=CC=C2NC=1)CCSC)C(N)=O)C1=CC=CC=C1 RGYLYUZOGHTBRF-BIHRQFPBSA-N 0.000 description 1
- 150000003573 thiols Chemical group 0.000 description 1
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Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- C07K14/575—Hormones
- C07K14/655—Somatostatins
- C07K14/6555—Somatostatins at least 1 amino acid in D-form
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y10—TECHNICAL SUBJECTS COVERED BY FORMER USPC
- Y10S—TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y10S930/00—Peptide or protein sequence
- Y10S930/01—Peptide or protein sequence
- Y10S930/16—Somatostatin; related peptides
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y10—TECHNICAL SUBJECTS COVERED BY FORMER USPC
- Y10S—TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y10S930/00—Peptide or protein sequence
- Y10S930/01—Peptide or protein sequence
- Y10S930/28—Bound to a nonpeptide drug, nonpeptide label, nonpeptide carrier, or a nonpeptide resin
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Biophysics (AREA)
- Medicinal Chemistry (AREA)
- Zoology (AREA)
- Biochemistry (AREA)
- Toxicology (AREA)
- General Health & Medical Sciences (AREA)
- Genetics & Genomics (AREA)
- Gastroenterology & Hepatology (AREA)
- Molecular Biology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Endocrinology (AREA)
- Peptides Or Proteins (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Steroid Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US05/789,472 US4100117A (en) | 1977-04-21 | 1977-04-21 | Somatostatin analogs and intermediates thereto |
| US78947277 | 1977-04-21 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| FI781184A7 FI781184A7 (fi) | 1978-10-22 |
| FI64576B FI64576B (fi) | 1983-08-31 |
| FI64576C true FI64576C (fi) | 1983-12-12 |
Family
ID=25147748
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| FI781184A FI64576C (fi) | 1977-04-21 | 1978-04-18 | Foerfarande foer framstaellning av en terapeutiskt anvaendbar somatostatinanalog |
Country Status (31)
| Country | Link |
|---|---|
| US (1) | US4100117A (ro) |
| JP (1) | JPS53132588A (ro) |
| AR (1) | AR221699A1 (ro) |
| AT (1) | AT361142B (ro) |
| AU (1) | AU519275B2 (ro) |
| BE (1) | BE866117A (ro) |
| BG (1) | BG28703A3 (ro) |
| CA (2) | CA1102315A (ro) |
| CH (1) | CH634039A5 (ro) |
| CS (1) | CS202096B2 (ro) |
| DD (1) | DD135900A5 (ro) |
| DE (1) | DE2816854A1 (ro) |
| DK (1) | DK174278A (ro) |
| ES (2) | ES469005A1 (ro) |
| FI (1) | FI64576C (ro) |
| FR (1) | FR2387941A1 (ro) |
| GB (1) | GB1596328A (ro) |
| GR (1) | GR68945B (ro) |
| HU (1) | HU177435B (ro) |
| IE (1) | IE46868B1 (ro) |
| IL (1) | IL54533A (ro) |
| IT (1) | IT1094462B (ro) |
| NL (1) | NL7804218A (ro) |
| NZ (1) | NZ187009A (ro) |
| PL (2) | PL114533B1 (ro) |
| PT (1) | PT67913B (ro) |
| RO (2) | RO81079A (ro) |
| SE (1) | SE7804397L (ro) |
| SU (2) | SU730295A3 (ro) |
| YU (1) | YU91578A (ro) |
| ZA (1) | ZA782247B (ro) |
Families Citing this family (31)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4202802A (en) * | 1978-10-02 | 1980-05-13 | Eli Lilly And Company | Peptides related to somatostatin |
| US4199501A (en) * | 1978-11-20 | 1980-04-22 | Eli Lilly And Company | Peptides related to somatostatin |
| US4199500A (en) * | 1978-11-20 | 1980-04-22 | Eli Lilly And Company | Peptides related to somatostatin |
| US4428942A (en) | 1982-05-17 | 1984-01-31 | The Salk Institute For Biological Studies | Analogs of somatostatin |
| GB8423431D0 (en) * | 1984-09-17 | 1984-10-24 | Sandoz Ltd | Organic compounds |
| SE8702550D0 (sv) * | 1987-06-18 | 1987-06-18 | Anders Grubb | Cysteinproteashemmare |
| NZ240214A (en) | 1990-10-16 | 1993-02-25 | Takeda Chemical Industries Ltd | Polymer compositions comprising a polylactic acid and a copolymer of glycolic acid and a hydroxycarboxylic acid; use as carrier for prolonged release pharmaceutical compositions of water soluble drugs |
| EP0582459B1 (en) | 1992-08-07 | 1998-01-07 | Takeda Chemical Industries, Ltd. | Production of microcapsules of water-soluble drugs |
| US5594091A (en) * | 1994-02-21 | 1997-01-14 | Takeda Chemical Industries, Ltd. | Matrix for sustained-release preparation |
| US6117455A (en) * | 1994-09-30 | 2000-09-12 | Takeda Chemical Industries, Ltd. | Sustained-release microcapsule of amorphous water-soluble pharmaceutical active agent |
| CA2192782C (en) | 1995-12-15 | 2008-10-14 | Nobuyuki Takechi | Production of microspheres |
| CA2208336A1 (en) * | 1996-06-20 | 1997-12-20 | Hisamitsu Pharmaceuticals Co., Inc. | A device structure for iontophoresis |
| US7169889B1 (en) | 1999-06-19 | 2007-01-30 | Biocon Limited | Insulin prodrugs hydrolyzable in vivo to yield peglylated insulin |
| US6309633B1 (en) | 1999-06-19 | 2001-10-30 | Nobex Corporation | Amphiphilic drug-oligomer conjugates with hydroyzable lipophile components and methods for making and using the same |
| ATE416784T1 (de) | 2000-12-01 | 2008-12-15 | Takeda Pharmaceutical | Verfahren zur herstellung einer zubereitung mit einer bioaktiven substanz |
| US6867183B2 (en) * | 2001-02-15 | 2005-03-15 | Nobex Corporation | Pharmaceutical compositions of insulin drug-oligomer conjugates and methods of treating diseases therewith |
| US7060675B2 (en) * | 2001-02-15 | 2006-06-13 | Nobex Corporation | Methods of treating diabetes mellitus |
| US7713932B2 (en) | 2001-06-04 | 2010-05-11 | Biocon Limited | Calcitonin drug-oligomer conjugates, and uses thereof |
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| Publication number | Priority date | Publication date | Assignee | Title |
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| DE2608336A1 (de) * | 1975-03-11 | 1976-09-30 | Sandoz Ag | Neue organische verbindungen, ihre herstellung und verwendung |
| US4372884A (en) * | 1975-08-06 | 1983-02-08 | The Salk Institute For Biological Studies | Pharmaceutically active peptides |
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| MM | Patent lapsed |
Owner name: ELI LILLY AND COMPANY |