FI62304C - Foerfarande foer framstaellning av ataraktiska trans-1,3,4,4a 5,9b-heksahydro-5-fenyl-2h-pyrido(4,3-b)indol-2-alkansyror -alkansyraestrar -alkanonitriler och -alkanoner - Google Patents

Foerfarande foer framstaellning av ataraktiska trans-1,3,4,4a 5,9b-heksahydro-5-fenyl-2h-pyrido(4,3-b)indol-2-alkansyror -alkansyraestrar -alkanonitriler och -alkanoner Download PDF

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Publication number
FI62304C
FI62304C FI771088A FI771088A FI62304C FI 62304 C FI62304 C FI 62304C FI 771088 A FI771088 A FI 771088A FI 771088 A FI771088 A FI 771088A FI 62304 C FI62304 C FI 62304C
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FI
Finland
Prior art keywords
formula
compound
phenyl
pyrido
trans
Prior art date
Application number
FI771088A
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English (en)
Finnish (fi)
Other versions
FI62304B (fi
FI771088A7 (cg-RX-API-DMAC10.html
Inventor
Joel Gilbert Berger
Original Assignee
Endo Lab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Endo Lab filed Critical Endo Lab
Publication of FI771088A7 publication Critical patent/FI771088A7/fi
Publication of FI62304B publication Critical patent/FI62304B/fi
Application granted granted Critical
Publication of FI62304C publication Critical patent/FI62304C/fi

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Anesthesiology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biomedical Technology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
FI771088A 1976-04-08 1977-04-06 Foerfarande foer framstaellning av ataraktiska trans-1,3,4,4a 5,9b-heksahydro-5-fenyl-2h-pyrido(4,3-b)indol-2-alkansyror -alkansyraestrar -alkanonitriler och -alkanoner FI62304C (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US67511276A 1976-04-08 1976-04-08
US67511276 1976-04-08

Publications (3)

Publication Number Publication Date
FI771088A7 FI771088A7 (cg-RX-API-DMAC10.html) 1977-10-09
FI62304B FI62304B (fi) 1982-08-31
FI62304C true FI62304C (fi) 1982-12-10

Family

ID=24709111

Family Applications (1)

Application Number Title Priority Date Filing Date
FI771088A FI62304C (fi) 1976-04-08 1977-04-06 Foerfarande foer framstaellning av ataraktiska trans-1,3,4,4a 5,9b-heksahydro-5-fenyl-2h-pyrido(4,3-b)indol-2-alkansyror -alkansyraestrar -alkanonitriler och -alkanoner

Country Status (28)

Country Link
US (1) US4141980A (cg-RX-API-DMAC10.html)
JP (1) JPS52125197A (cg-RX-API-DMAC10.html)
AR (1) AR218246A1 (cg-RX-API-DMAC10.html)
AT (1) AT360533B (cg-RX-API-DMAC10.html)
AU (1) AU516432B2 (cg-RX-API-DMAC10.html)
BE (1) BE853422A (cg-RX-API-DMAC10.html)
CA (1) CA1071210A (cg-RX-API-DMAC10.html)
CH (1) CH633795A5 (cg-RX-API-DMAC10.html)
DD (1) DD132015A5 (cg-RX-API-DMAC10.html)
DE (1) DE2715355A1 (cg-RX-API-DMAC10.html)
DK (1) DK154877A (cg-RX-API-DMAC10.html)
ES (1) ES457665A1 (cg-RX-API-DMAC10.html)
FI (1) FI62304C (cg-RX-API-DMAC10.html)
FR (1) FR2347365A1 (cg-RX-API-DMAC10.html)
GB (1) GB1572057A (cg-RX-API-DMAC10.html)
GR (1) GR63666B (cg-RX-API-DMAC10.html)
HU (1) HU176956B (cg-RX-API-DMAC10.html)
IE (1) IE45189B1 (cg-RX-API-DMAC10.html)
IL (1) IL51840A (cg-RX-API-DMAC10.html)
LU (1) LU77091A1 (cg-RX-API-DMAC10.html)
NL (1) NL7703898A (cg-RX-API-DMAC10.html)
NO (1) NO771242L (cg-RX-API-DMAC10.html)
NZ (1) NZ183824A (cg-RX-API-DMAC10.html)
PH (1) PH13152A (cg-RX-API-DMAC10.html)
PT (1) PT66407B (cg-RX-API-DMAC10.html)
SE (1) SE7702301L (cg-RX-API-DMAC10.html)
SU (1) SU719503A3 (cg-RX-API-DMAC10.html)
ZA (1) ZA772166B (cg-RX-API-DMAC10.html)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SE7702300L (sv) * 1976-04-15 1977-10-16 Endo Lab Reduktionsforlopp
US4224329A (en) * 1979-01-23 1980-09-23 Pfizer Inc. 2-Substituted-trans-5-aryl-2,3,4,4a,5,9b-hexahydro-1H-pyrido[4,3-b]indoles
US4252812A (en) * 1977-05-23 1981-02-24 Pfizer Inc. 2-Substituted-trans-5-aryl-2,3,4,4a,5,9b-hexahydro-1H-pyrido[4,3-b]indoles
US4267331A (en) * 1979-01-23 1981-05-12 Pfizer Inc. Process for the production of 2-substituted pyrido[4,3-b]-indoles
US4432978A (en) * 1979-07-30 1984-02-21 Pfizer Inc. Hexahydro-trans-pyridoindole
US4352807A (en) * 1979-07-30 1982-10-05 Pfizer Inc. Hexahydro-trans-pyridoindole neuroleptic agents
US4337250A (en) * 1979-07-30 1982-06-29 Pfizer Inc. Hexahydro-trans- and tetrahydropyridoindole neuroleptic agents
US4431649A (en) * 1979-07-30 1984-02-14 Pfizer Inc. Hexahydro-trans- and tetrahydropyridoindole neuroleptic agents
US4252811A (en) * 1979-07-30 1981-02-24 Pfizer Inc. Hexahydro-trans-pyridoindole neuroleptic agents
US4431646A (en) * 1979-07-30 1984-02-14 Pfizer Inc. Hexahydro-trans- and tetrahydropyridoindole neuroleptic agents
US4427679A (en) 1981-01-16 1984-01-24 Pfizer Inc. Hexahydro-trans- and tetrahydropyridoindole neuroleptic agents
US5319087A (en) * 1987-04-16 1994-06-07 Eli Lilly And Company Piperidine opioid antagonists
US4992450A (en) * 1987-04-16 1991-02-12 Eli Lilly And Company Piperidine opioid antagonists
US4891379A (en) * 1987-04-16 1990-01-02 Kabushiki Kaisha Kobe Seikosho Piperidine opioid antagonists
US5270328A (en) * 1991-03-29 1993-12-14 Eli Lilly And Company Peripherally selective piperidine opioid antagonists
US5159081A (en) * 1991-03-29 1992-10-27 Eli Lilly And Company Intermediates of peripherally selective n-carbonyl-3,4,4-trisubstituted piperidine opioid antagonists
US5250542A (en) * 1991-03-29 1993-10-05 Eli Lilly And Company Peripherally selective piperidine carboxylate opioid antagonists

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH303833A (de) * 1951-04-30 1954-12-15 Bayer Ag Verfahren zur Herstellung von Derivaten des Tetrahydro-y-carbolins.
JPS50126699A (cg-RX-API-DMAC10.html) * 1974-03-20 1975-10-04

Also Published As

Publication number Publication date
DK154877A (da) 1977-10-09
JPS52125197A (en) 1977-10-20
AU2401277A (en) 1978-10-12
AU516432B2 (en) 1981-06-04
NZ183824A (en) 1980-10-24
ES457665A1 (es) 1978-07-16
IE45189L (en) 1977-10-08
ZA772166B (en) 1978-05-30
IE45189B1 (en) 1982-07-14
DD132015A5 (de) 1978-08-16
FR2347365B1 (cg-RX-API-DMAC10.html) 1979-03-02
FR2347365A1 (fr) 1977-11-04
GB1572057A (en) 1980-07-23
AT360533B (de) 1981-01-12
NO771242L (no) 1977-10-11
BE853422A (fr) 1977-10-10
IL51840A (en) 1980-10-26
FI62304B (fi) 1982-08-31
ATA242377A (de) 1980-06-15
GR63666B (en) 1979-11-28
FI771088A7 (cg-RX-API-DMAC10.html) 1977-10-09
IL51840A0 (en) 1977-06-30
SE7702301L (sv) 1977-10-09
SU719503A3 (ru) 1980-02-29
PT66407B (en) 1978-09-13
US4141980A (en) 1979-02-27
AR218246A1 (es) 1980-05-30
PH13152A (en) 1979-12-18
HU176956B (hu) 1981-06-28
CH633795A5 (de) 1982-12-31
NL7703898A (nl) 1977-10-11
LU77091A1 (cg-RX-API-DMAC10.html) 1977-12-01
PT66407A (en) 1977-05-01
CA1071210A (en) 1980-02-05
DE2715355A1 (de) 1977-10-20

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Owner name: ENDO LABORATORIES, INC.