AR218246A1 - Procedimiento para la produccion de trans-1,3,4,4a,5,9b-hexahidro-5-fenil-2-h-pirido(4,3-b)-indoles 2-sustituidos - Google Patents

Procedimiento para la produccion de trans-1,3,4,4a,5,9b-hexahidro-5-fenil-2-h-pirido(4,3-b)-indoles 2-sustituidos

Info

Publication number
AR218246A1
AR218246A1 AR267148A AR26714877A AR218246A1 AR 218246 A1 AR218246 A1 AR 218246A1 AR 267148 A AR267148 A AR 267148A AR 26714877 A AR26714877 A AR 26714877A AR 218246 A1 AR218246 A1 AR 218246A1
Authority
AR
Argentina
Prior art keywords
hexahidro
pirido
fenil
indoles
trans
Prior art date
Application number
AR267148A
Other languages
English (en)
Original Assignee
Endo Lab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Endo Lab filed Critical Endo Lab
Application granted granted Critical
Publication of AR218246A1 publication Critical patent/AR218246A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Anesthesiology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biomedical Technology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
AR267148A 1976-04-08 1977-04-06 Procedimiento para la produccion de trans-1,3,4,4a,5,9b-hexahidro-5-fenil-2-h-pirido(4,3-b)-indoles 2-sustituidos AR218246A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US67511276A 1976-04-08 1976-04-08

Publications (1)

Publication Number Publication Date
AR218246A1 true AR218246A1 (es) 1980-05-30

Family

ID=24709111

Family Applications (1)

Application Number Title Priority Date Filing Date
AR267148A AR218246A1 (es) 1976-04-08 1977-04-06 Procedimiento para la produccion de trans-1,3,4,4a,5,9b-hexahidro-5-fenil-2-h-pirido(4,3-b)-indoles 2-sustituidos

Country Status (28)

Country Link
US (1) US4141980A (es)
JP (1) JPS52125197A (es)
AR (1) AR218246A1 (es)
AT (1) AT360533B (es)
AU (1) AU516432B2 (es)
BE (1) BE853422A (es)
CA (1) CA1071210A (es)
CH (1) CH633795A5 (es)
DD (1) DD132015A5 (es)
DE (1) DE2715355A1 (es)
DK (1) DK154877A (es)
ES (1) ES457665A1 (es)
FI (1) FI62304C (es)
FR (1) FR2347365A1 (es)
GB (1) GB1572057A (es)
GR (1) GR63666B (es)
HU (1) HU176956B (es)
IE (1) IE45189B1 (es)
IL (1) IL51840A (es)
LU (1) LU77091A1 (es)
NL (1) NL7703898A (es)
NO (1) NO771242L (es)
NZ (1) NZ183824A (es)
PH (1) PH13152A (es)
PT (1) PT66407B (es)
SE (1) SE7702301L (es)
SU (1) SU719503A3 (es)
ZA (1) ZA772166B (es)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SE7702300L (sv) * 1976-04-15 1977-10-16 Endo Lab Reduktionsforlopp
US4224329A (en) * 1979-01-23 1980-09-23 Pfizer Inc. 2-Substituted-trans-5-aryl-2,3,4,4a,5,9b-hexahydro-1H-pyrido[4,3-b]indoles
US4252812A (en) * 1977-05-23 1981-02-24 Pfizer Inc. 2-Substituted-trans-5-aryl-2,3,4,4a,5,9b-hexahydro-1H-pyrido[4,3-b]indoles
US4267331A (en) * 1979-01-23 1981-05-12 Pfizer Inc. Process for the production of 2-substituted pyrido[4,3-b]-indoles
US4337250A (en) * 1979-07-30 1982-06-29 Pfizer Inc. Hexahydro-trans- and tetrahydropyridoindole neuroleptic agents
US4432978A (en) * 1979-07-30 1984-02-21 Pfizer Inc. Hexahydro-trans-pyridoindole
US4431649A (en) * 1979-07-30 1984-02-14 Pfizer Inc. Hexahydro-trans- and tetrahydropyridoindole neuroleptic agents
US4352807A (en) * 1979-07-30 1982-10-05 Pfizer Inc. Hexahydro-trans-pyridoindole neuroleptic agents
US4252811A (en) * 1979-07-30 1981-02-24 Pfizer Inc. Hexahydro-trans-pyridoindole neuroleptic agents
US4431646A (en) * 1979-07-30 1984-02-14 Pfizer Inc. Hexahydro-trans- and tetrahydropyridoindole neuroleptic agents
US4427679A (en) 1981-01-16 1984-01-24 Pfizer Inc. Hexahydro-trans- and tetrahydropyridoindole neuroleptic agents
US5319087A (en) * 1987-04-16 1994-06-07 Eli Lilly And Company Piperidine opioid antagonists
US4891379A (en) * 1987-04-16 1990-01-02 Kabushiki Kaisha Kobe Seikosho Piperidine opioid antagonists
US4992450A (en) * 1987-04-16 1991-02-12 Eli Lilly And Company Piperidine opioid antagonists
US5159081A (en) * 1991-03-29 1992-10-27 Eli Lilly And Company Intermediates of peripherally selective n-carbonyl-3,4,4-trisubstituted piperidine opioid antagonists
US5270328A (en) * 1991-03-29 1993-12-14 Eli Lilly And Company Peripherally selective piperidine opioid antagonists
US5250542A (en) * 1991-03-29 1993-10-05 Eli Lilly And Company Peripherally selective piperidine carboxylate opioid antagonists

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH303833A (de) * 1951-04-30 1954-12-15 Bayer Ag Verfahren zur Herstellung von Derivaten des Tetrahydro-y-carbolins.
JPS50126699A (es) * 1974-03-20 1975-10-04

Also Published As

Publication number Publication date
ES457665A1 (es) 1978-07-16
SE7702301L (sv) 1977-10-09
AT360533B (de) 1981-01-12
SU719503A3 (ru) 1980-02-29
IL51840A0 (en) 1977-06-30
CH633795A5 (de) 1982-12-31
ATA242377A (de) 1980-06-15
NZ183824A (en) 1980-10-24
PT66407A (en) 1977-05-01
DE2715355A1 (de) 1977-10-20
IL51840A (en) 1980-10-26
CA1071210A (en) 1980-02-05
PT66407B (en) 1978-09-13
NO771242L (no) 1977-10-11
BE853422A (fr) 1977-10-10
GB1572057A (en) 1980-07-23
ZA772166B (en) 1978-05-30
PH13152A (en) 1979-12-18
HU176956B (hu) 1981-06-28
AU2401277A (en) 1978-10-12
IE45189B1 (en) 1982-07-14
DD132015A5 (de) 1978-08-16
NL7703898A (nl) 1977-10-11
FI771088A (es) 1977-10-09
FI62304B (fi) 1982-08-31
FI62304C (fi) 1982-12-10
FR2347365A1 (fr) 1977-11-04
US4141980A (en) 1979-02-27
IE45189L (en) 1977-10-08
AU516432B2 (en) 1981-06-04
LU77091A1 (es) 1977-12-01
DK154877A (da) 1977-10-09
GR63666B (en) 1979-11-28
JPS52125197A (en) 1977-10-20
FR2347365B1 (es) 1979-03-02

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