FI61480C - Foerfarande foer framstaellning av antiemetiskt verksamma n-(1-substituerade-3-pyrrolidinyl)-1-naftalen- och -4-kinolinkarboxamider - Google Patents

Foerfarande foer framstaellning av antiemetiskt verksamma n-(1-substituerade-3-pyrrolidinyl)-1-naftalen- och -4-kinolinkarboxamider Download PDF

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Publication number
FI61480C
FI61480C FI753606A FI753606A FI61480C FI 61480 C FI61480 C FI 61480C FI 753606 A FI753606 A FI 753606A FI 753606 A FI753606 A FI 753606A FI 61480 C FI61480 C FI 61480C
Authority
FI
Finland
Prior art keywords
pyrrolidinyl
naphthalene
preparation
antiemetic
substituted
Prior art date
Application number
FI753606A
Other languages
English (en)
Finnish (fi)
Other versions
FI753606A (fr
FI61480B (fi
Inventor
Jr Albert Duncan Cale
Original Assignee
Robins Co Inc A H
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Robins Co Inc A H filed Critical Robins Co Inc A H
Publication of FI753606A publication Critical patent/FI753606A/fi
Application granted granted Critical
Publication of FI61480B publication Critical patent/FI61480B/fi
Publication of FI61480C publication Critical patent/FI61480C/fi

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D207/10—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D207/14—Nitrogen atoms not forming part of a nitro radical
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics

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  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Otolaryngology (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Hospice & Palliative Care (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pyrrole Compounds (AREA)
FI753606A 1974-12-26 1975-12-19 Foerfarande foer framstaellning av antiemetiskt verksamma n-(1-substituerade-3-pyrrolidinyl)-1-naftalen- och -4-kinolinkarboxamider FI61480C (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US53651474 1974-12-26
US05/536,514 US4002757A (en) 1974-12-26 1974-12-26 N-(1-substituted-3-pyrrolidinyl)-4-quinolinecarboxamides

Publications (3)

Publication Number Publication Date
FI753606A FI753606A (fr) 1976-06-27
FI61480B FI61480B (fi) 1982-04-30
FI61480C true FI61480C (fi) 1982-08-10

Family

ID=24138812

Family Applications (1)

Application Number Title Priority Date Filing Date
FI753606A FI61480C (fi) 1974-12-26 1975-12-19 Foerfarande foer framstaellning av antiemetiskt verksamma n-(1-substituerade-3-pyrrolidinyl)-1-naftalen- och -4-kinolinkarboxamider

Country Status (18)

Country Link
US (3) US4002757A (fr)
JP (2) JPS5191254A (fr)
AU (1) AU499075B2 (fr)
BE (1) BE836975A (fr)
CA (1) CA1071636A (fr)
CH (1) CH611603A5 (fr)
DE (1) DE2558348A1 (fr)
DK (1) DK138536B (fr)
ES (1) ES443845A1 (fr)
FI (1) FI61480C (fr)
FR (1) FR2295744A1 (fr)
GB (1) GB1537848A (fr)
IE (1) IE43819B1 (fr)
NL (1) NL7515084A (fr)
NO (1) NO144670C (fr)
PH (1) PH13883A (fr)
SE (1) SE408417B (fr)
ZA (1) ZA757972B (fr)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4279822A (en) * 1972-04-03 1981-07-21 A. H. Robins Company, Inc. N-(1-Substituted-3-pyrrolidinyl)benzamides
US4002757A (en) * 1974-12-26 1977-01-11 A. H. Robins Company, Incorporated N-(1-substituted-3-pyrrolidinyl)-4-quinolinecarboxamides
US4143150A (en) * 1977-08-19 1979-03-06 A. H. Robins Company, Inc. Derivatives of oxanilic acid
EP0134225B1 (fr) * 1983-01-21 1988-08-17 ALKALOIDA VEGYéSZETI GYáR Nouveaux derives de diamines d'alcoyle
US5210329A (en) * 1992-02-18 1993-05-11 General Electric Company Process for preparing bisphenol-A
ATE479655T1 (de) 2001-09-14 2010-09-15 High Point Pharmaceuticals Llc Neue aminoazetidin-, aminopyrrolidin- und aminopiperidinderivative
US6673829B2 (en) 2001-09-14 2004-01-06 Novo Nordisk A/S Aminoazetidine,-pyrrolidine and -piperidine derivatives
NZ544046A (en) * 2003-06-17 2009-08-28 Pfizer N-pyrrolidin-3-yl-amide derivatives as serotonin and noradrenaline re-uptake inhibitors
US7348434B2 (en) * 2003-08-08 2008-03-25 Antony Bigot 4-substituted quinoline derivatives, method and intermediates for their preparation and pharmaceutical compositions containing them
US20090239929A1 (en) * 2004-12-14 2009-09-24 Paul Vincent Fish N-Pyrrolidin-3-YL-Amide Derivatives As Serotonin and Noradrenalin Re-Uptake Inhibitors
CA2590229A1 (fr) * 2004-12-14 2006-06-22 Pfizer Limited Nouveaux composes
CA2591415A1 (fr) * 2004-12-16 2006-06-22 Pfizer Limited Nouveaux composes
EP2481735A1 (fr) * 2007-05-09 2012-08-01 Pfizer Inc. Dérivés hétérocycliques substitués et leur utilisation pharmaceutique et compositions

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE67123C (de) * L. THOMAS in Montegnee-les-Siege, Belgien Handdrehbohrmaschine für Gruben und Steinbrüche
US1825623A (en) * 1931-09-29 Oonhohachzn
US3133061A (en) * 1962-11-13 1964-05-12 Sterling Drug Inc Piperidine carboxamides and derivatives thereof
US3342826A (en) * 1964-01-13 1967-09-19 Ile De France Heterocyclic aminoalkyl benzamides
GB1364231A (en) * 1968-12-23 1974-08-21 Robins Co Inc A H N-/1-substituted-3-pyrrolidinyl/benzamides and thiobenzamides
US3577440A (en) * 1968-12-23 1971-05-04 Robins Co Inc A H 1-substituted-3-amido-pyrrolidines
US3829434A (en) * 1972-11-10 1974-08-13 Pfizer Piperidinesulfonylurea derivatives
US4002757A (en) * 1974-12-26 1977-01-11 A. H. Robins Company, Incorporated N-(1-substituted-3-pyrrolidinyl)-4-quinolinecarboxamides

Also Published As

Publication number Publication date
CA1071636A (fr) 1980-02-12
JPS60248684A (ja) 1985-12-09
DK589075A (fr) 1976-06-27
DE2558348A1 (de) 1976-07-08
US4073796A (en) 1978-02-14
JPS5191254A (en) 1976-08-10
BE836975A (fr) 1976-04-16
ZA757972B (en) 1976-12-29
NL7515084A (nl) 1976-06-29
JPS611426B2 (fr) 1986-01-17
US4002757A (en) 1977-01-11
US4087428A (en) 1978-05-02
FR2295744A1 (fr) 1976-07-23
DK138536B (da) 1978-09-25
DK138536C (fr) 1979-03-05
FI753606A (fr) 1976-06-27
ES443845A1 (es) 1977-04-16
SE7514374L (sv) 1976-06-28
AU8755075A (en) 1977-06-23
CH611603A5 (fr) 1979-06-15
NO144670C (no) 1981-10-14
GB1537848A (en) 1979-01-04
FR2295744B1 (fr) 1978-07-28
IE43819L (en) 1976-06-26
FI61480B (fi) 1982-04-30
PH13883A (en) 1980-10-27
NO144670B (no) 1981-07-06
AU499075B2 (en) 1979-04-05
JPS619314B2 (fr) 1986-03-22
IE43819B1 (en) 1981-06-03
SE408417B (sv) 1979-06-11
NO754376L (fr) 1976-06-29

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Legal Events

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MM Patent lapsed

Owner name: A.H. ROBINS COMPANY, INCORPORATED