SE408417B - Forfarande for framstellning av n-(1-substituerade-3-pyrrolidinyl)-1-naftalen- och 4-kinolin-karboxamider med anti-emetiska terapeutiska egenskaper - Google Patents
Forfarande for framstellning av n-(1-substituerade-3-pyrrolidinyl)-1-naftalen- och 4-kinolin-karboxamider med anti-emetiska terapeutiska egenskaperInfo
- Publication number
- SE408417B SE408417B SE7514374A SE7514374A SE408417B SE 408417 B SE408417 B SE 408417B SE 7514374 A SE7514374 A SE 7514374A SE 7514374 A SE7514374 A SE 7514374A SE 408417 B SE408417 B SE 408417B
- Authority
- SE
- Sweden
- Prior art keywords
- kinoline
- carboxamides
- pyrrolidinyl
- naphthalene
- substituted
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D207/10—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D207/14—Nitrogen atoms not forming part of a nitro radical
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Veterinary Medicine (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Otolaryngology (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Hospice & Palliative Care (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pyrrole Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US05/536,514 US4002757A (en) | 1974-12-26 | 1974-12-26 | N-(1-substituted-3-pyrrolidinyl)-4-quinolinecarboxamides |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| SE7514374L SE7514374L (sv) | 1976-06-28 |
| SE408417B true SE408417B (sv) | 1979-06-11 |
Family
ID=24138812
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| SE7514374A SE408417B (sv) | 1974-12-26 | 1975-12-18 | Forfarande for framstellning av n-(1-substituerade-3-pyrrolidinyl)-1-naftalen- och 4-kinolin-karboxamider med anti-emetiska terapeutiska egenskaper |
Country Status (18)
| Country | Link |
|---|---|
| US (3) | US4002757A (xx) |
| JP (2) | JPS5191254A (xx) |
| AU (1) | AU499075B2 (xx) |
| BE (1) | BE836975A (xx) |
| CA (1) | CA1071636A (xx) |
| CH (1) | CH611603A5 (xx) |
| DE (1) | DE2558348A1 (xx) |
| DK (1) | DK138536B (xx) |
| ES (1) | ES443845A1 (xx) |
| FI (1) | FI61480C (xx) |
| FR (1) | FR2295744A1 (xx) |
| GB (1) | GB1537848A (xx) |
| IE (1) | IE43819B1 (xx) |
| NL (1) | NL7515084A (xx) |
| NO (1) | NO144670C (xx) |
| PH (1) | PH13883A (xx) |
| SE (1) | SE408417B (xx) |
| ZA (1) | ZA757972B (xx) |
Families Citing this family (13)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4279822A (en) * | 1972-04-03 | 1981-07-21 | A. H. Robins Company, Inc. | N-(1-Substituted-3-pyrrolidinyl)benzamides |
| US4002757A (en) * | 1974-12-26 | 1977-01-11 | A. H. Robins Company, Incorporated | N-(1-substituted-3-pyrrolidinyl)-4-quinolinecarboxamides |
| US4143150A (en) * | 1977-08-19 | 1979-03-06 | A. H. Robins Company, Inc. | Derivatives of oxanilic acid |
| JPH0615527B2 (ja) * | 1983-01-21 | 1994-03-02 | アルカロイダ ベギエスゼテイ ギヤル | アルキルジアミン誘導体、その製造法および抗不整脈剤 |
| US5210329A (en) * | 1992-02-18 | 1993-05-11 | General Electric Company | Process for preparing bisphenol-A |
| US6673829B2 (en) | 2001-09-14 | 2004-01-06 | Novo Nordisk A/S | Aminoazetidine,-pyrrolidine and -piperidine derivatives |
| DE60237528D1 (de) | 2001-09-14 | 2010-10-14 | High Point Pharmaceuticals Llc | Neue aminoazetidin-, aminopyrrolidin- und aminopiperidinderivative |
| AP2005003467A0 (en) * | 2003-06-17 | 2006-12-31 | Pfizer | N-pyrrolidin-3-YL-amide derivatives as serotonin and noradrenaline reuptake inhibitors. |
| US7348434B2 (en) * | 2003-08-08 | 2008-03-25 | Antony Bigot | 4-substituted quinoline derivatives, method and intermediates for their preparation and pharmaceutical compositions containing them |
| EP1828119A1 (en) * | 2004-12-14 | 2007-09-05 | Pfizer Limited | N-pyrrolidin-3-yl-amide derivatives as serotonin and noradrenalin re-uptake inhibitors |
| JP2008523137A (ja) * | 2004-12-14 | 2008-07-03 | ファイザー・リミテッド | セロトニンおよびノルアドレナリン再取込み阻害剤としてのｎ−ピロリジン−３−イル−アミド誘導体 |
| CA2591415A1 (en) * | 2004-12-16 | 2006-06-22 | Pfizer Limited | N-pyrrolidin-3-yl-amide derivatives as serotonin and noradrenalin re-uptake inhibitors |
| KR20090130347A (ko) * | 2007-05-09 | 2009-12-22 | 화이자 인코포레이티드 | 치환된 헤테로사이클릭 유도체 및 조성물 및 항균제로서의 이의 약학적 용도 |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE67123C (de) * | L. THOMAS in Montegnee-les-Siege, Belgien | Handdrehbohrmaschine für Gruben und Steinbrüche | ||
| US1825623A (en) * | 1931-09-29 | Oonhohachzn | ||
| US3133061A (en) * | 1962-11-13 | 1964-05-12 | Sterling Drug Inc | Piperidine carboxamides and derivatives thereof |
| US3342826A (en) * | 1964-01-13 | 1967-09-19 | Ile De France | Heterocyclic aminoalkyl benzamides |
| US3577440A (en) * | 1968-12-23 | 1971-05-04 | Robins Co Inc A H | 1-substituted-3-amido-pyrrolidines |
| GB1364231A (en) * | 1968-12-23 | 1974-08-21 | Robins Co Inc A H | N-/1-substituted-3-pyrrolidinyl/benzamides and thiobenzamides |
| US3829434A (en) * | 1972-11-10 | 1974-08-13 | Pfizer | Piperidinesulfonylurea derivatives |
| US4002757A (en) * | 1974-12-26 | 1977-01-11 | A. H. Robins Company, Incorporated | N-(1-substituted-3-pyrrolidinyl)-4-quinolinecarboxamides |
-
1974
- 1974-12-26 US US05/536,514 patent/US4002757A/en not_active Expired - Lifetime
-
1975
- 1975-12-15 AU AU87550/75A patent/AU499075B2/en not_active Expired
- 1975-12-18 SE SE7514374A patent/SE408417B/xx not_active IP Right Cessation
- 1975-12-19 FI FI753606A patent/FI61480C/fi not_active IP Right Cessation
- 1975-12-22 CH CH1660375A patent/CH611603A5/xx not_active IP Right Cessation
- 1975-12-22 BE BE163038A patent/BE836975A/xx not_active IP Right Cessation
- 1975-12-23 NO NO754376A patent/NO144670C/no unknown
- 1975-12-23 IE IE2822/75A patent/IE43819B1/en unknown
- 1975-12-23 ZA ZA00757972A patent/ZA757972B/xx unknown
- 1975-12-23 FR FR7539569A patent/FR2295744A1/fr active Granted
- 1975-12-23 GB GB52612/75A patent/GB1537848A/en not_active Expired
- 1975-12-23 CA CA242,432A patent/CA1071636A/en not_active Expired
- 1975-12-23 DE DE19752558348 patent/DE2558348A1/de not_active Ceased
- 1975-12-23 DK DK589075AA patent/DK138536B/da not_active IP Right Cessation
- 1975-12-24 PH PH17926A patent/PH13883A/en unknown
- 1975-12-24 NL NL7515084A patent/NL7515084A/xx active Search and Examination
- 1975-12-24 ES ES443845A patent/ES443845A1/es not_active Expired
- 1975-12-26 JP JP50159797A patent/JPS5191254A/ja active Granted
-
1976
- 1976-05-05 US US05/683,604 patent/US4087428A/en not_active Expired - Lifetime
- 1976-05-05 US US05/683,605 patent/US4073796A/en not_active Expired - Lifetime
-
1985
- 1985-04-25 JP JP60089861A patent/JPS60248684A/ja active Granted
Also Published As
| Publication number | Publication date |
|---|---|
| US4087428A (en) | 1978-05-02 |
| CH611603A5 (xx) | 1979-06-15 |
| FI61480C (fi) | 1982-08-10 |
| FR2295744A1 (fr) | 1976-07-23 |
| FI753606A (xx) | 1976-06-27 |
| US4073796A (en) | 1978-02-14 |
| FR2295744B1 (xx) | 1978-07-28 |
| DK138536B (da) | 1978-09-25 |
| NO754376L (xx) | 1976-06-29 |
| JPS60248684A (ja) | 1985-12-09 |
| BE836975A (fr) | 1976-04-16 |
| US4002757A (en) | 1977-01-11 |
| CA1071636A (en) | 1980-02-12 |
| PH13883A (en) | 1980-10-27 |
| ES443845A1 (es) | 1977-04-16 |
| AU499075B2 (en) | 1979-04-05 |
| ZA757972B (en) | 1976-12-29 |
| SE7514374L (sv) | 1976-06-28 |
| JPS5191254A (en) | 1976-08-10 |
| NO144670C (no) | 1981-10-14 |
| NL7515084A (nl) | 1976-06-29 |
| IE43819L (en) | 1976-06-26 |
| GB1537848A (en) | 1979-01-04 |
| DE2558348A1 (de) | 1976-07-08 |
| IE43819B1 (en) | 1981-06-03 |
| DK138536C (xx) | 1979-03-05 |
| NO144670B (no) | 1981-07-06 |
| AU8755075A (en) | 1977-06-23 |
| JPS611426B2 (xx) | 1986-01-17 |
| JPS619314B2 (xx) | 1986-03-22 |
| DK589075A (xx) | 1976-06-27 |
| FI61480B (fi) | 1982-04-30 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| NUG | Patent has lapsed |
Ref document number: 7514374-3 Effective date: 19920704 Format of ref document f/p: F |