FI57410C - Foerfarande foer framstaellning av nya neuroleptiskt aktiva 6-fluor-substituerade tiaxantenfoereningar och dessas salter - Google Patents

Foerfarande foer framstaellning av nya neuroleptiskt aktiva 6-fluor-substituerade tiaxantenfoereningar och dessas salter Download PDF

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Publication number
FI57410C
FI57410C FI3618/73A FI361873A FI57410C FI 57410 C FI57410 C FI 57410C FI 3618/73 A FI3618/73 A FI 3618/73A FI 361873 A FI361873 A FI 361873A FI 57410 C FI57410 C FI 57410C
Authority
FI
Finland
Prior art keywords
formula
compound
color
fluoro
thiaxanthene
Prior art date
Application number
FI3618/73A
Other languages
English (en)
Finnish (fi)
Other versions
FI57410B (fi
Inventor
Joern Lasse Martin Buus
Niels Lassen
Allan Johan Bigler
Original Assignee
Kefalas As
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Kefalas As filed Critical Kefalas As
Application granted granted Critical
Publication of FI57410B publication Critical patent/FI57410B/fi
Publication of FI57410C publication Critical patent/FI57410C/fi

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/04—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
    • C07D295/08—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms
    • C07D295/084—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms with the ring nitrogen atoms and the oxygen or sulfur atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings
    • C07D295/088—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms with the ring nitrogen atoms and the oxygen or sulfur atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings to an acyclic saturated chain
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C323/00—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D337/00—Heterocyclic compounds containing rings of more than six members having one sulfur atom as the only ring hetero atom
    • C07D337/02—Seven-membered rings
    • C07D337/06—Seven-membered rings condensed with carbocyclic rings or ring systems
    • C07D337/10—Seven-membered rings condensed with carbocyclic rings or ring systems condensed with two six-membered rings
    • C07D337/14—[b,f]-condensed

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
FI3618/73A 1972-12-08 1973-11-23 Foerfarande foer framstaellning av nya neuroleptiskt aktiva 6-fluor-substituerade tiaxantenfoereningar och dessas salter FI57410C (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB5691072A GB1453828A (en) 1972-12-08 1972-12-08 Fluoro-substituted thiaxanthene derivatives
GB5691072 1972-12-08

Publications (2)

Publication Number Publication Date
FI57410B FI57410B (fi) 1980-04-30
FI57410C true FI57410C (fi) 1980-08-11

Family

ID=10477876

Family Applications (1)

Application Number Title Priority Date Filing Date
FI3618/73A FI57410C (fi) 1972-12-08 1973-11-23 Foerfarande foer framstaellning av nya neuroleptiskt aktiva 6-fluor-substituerade tiaxantenfoereningar och dessas salter

Country Status (19)

Country Link
JP (1) JPS594436B2 (fr)
AR (2) AR202805A1 (fr)
AT (1) AT332395B (fr)
BE (1) BE808347A (fr)
CH (2) CH590272A5 (fr)
CS (1) CS176259B2 (fr)
DE (1) DE2359359C3 (fr)
DK (1) DK145576C (fr)
ES (2) ES421098A1 (fr)
FI (1) FI57410C (fr)
FR (1) FR2209573B1 (fr)
GB (1) GB1453828A (fr)
HU (1) HU167778B (fr)
IE (1) IE38554B1 (fr)
NL (1) NL7316035A (fr)
NO (1) NO138806C (fr)
PL (1) PL95266B1 (fr)
SE (1) SE400287B (fr)
ZA (1) ZA738990B (fr)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NZ189108A (en) * 1977-12-29 1982-02-23 Kefalas As 2-methylthio-6-fluoro-9-(1-methyl-4-piperidylidene)-thioxanthene and pharmaceutical compositions intermediate 2-methylthio-6-fluoro-9-(1-methyl-4-piperidyl)-thioxanthen-9-ol
US5173489A (en) * 1986-04-10 1992-12-22 The Dupont Merck Pharmaceutical Co. α,α-disubstituted aromatics and heteroaromatics as cognition enhancers
GB8628903D0 (en) * 1986-12-03 1987-01-07 Lunbeck A S H Neuroleptic compounds
US6395752B1 (en) * 1999-03-04 2002-05-28 Pharmaquest Limited Method of treating depression using 1-threo-methylphenidate
US6127385A (en) * 1999-03-04 2000-10-03 Pharmaquest Limited Method of treating depression using l-threo-methylphenidate
WO2008080398A1 (fr) * 2007-01-05 2008-07-10 Bkg Pharma Aps Agents anti-infectieux tels que des dérivés de phénothiazine et de thioxanthène pour traiter les maladies infectieuses

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE585338A (fr) * 1958-12-04
FR1463787A (fr) * 1963-10-14 1966-07-22 Pfizer & Co C Composés de phosphonium aminoalcoyl-trisubstitués, dérivés de tels composés, et procédés pour leur préparation

Also Published As

Publication number Publication date
AT332395B (de) 1976-09-27
ZA738990B (en) 1974-11-27
AR202672A1 (es) 1975-06-30
ES421098A1 (es) 1976-08-01
FR2209573B1 (fr) 1977-12-09
DE2359359A1 (de) 1974-06-27
NO138806C (no) 1978-11-15
ES444294A1 (es) 1977-10-01
PL95266B1 (pl) 1977-10-31
DE2359359C3 (de) 1978-11-02
AR202805A1 (es) 1975-07-24
SE400287B (sv) 1978-03-20
FI57410B (fi) 1980-04-30
AU6296673A (en) 1975-05-29
IE38554B1 (en) 1978-04-12
HU167778B (fr) 1975-12-25
JPS4994691A (fr) 1974-09-09
FR2209573A1 (fr) 1974-07-05
DK145576C (da) 1983-06-13
BE808347A (fr) 1974-03-29
IE38554L (en) 1974-06-08
ATA1000373A (de) 1976-01-15
CH590272A5 (fr) 1977-07-29
GB1453828A (en) 1976-10-27
CS176259B2 (fr) 1977-06-30
NO138806B (no) 1978-08-07
DK145576B (da) 1982-12-13
DE2359359B2 (de) 1978-02-16
JPS594436B2 (ja) 1984-01-30
CH592085A5 (fr) 1977-10-14
NL7316035A (fr) 1974-06-11

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