FI57400C - Foerfarande foer framstaellning av 2,4-diamino-5-bensylpyrimidiner - Google Patents

Foerfarande foer framstaellning av 2,4-diamino-5-bensylpyrimidiner Download PDF

Info

Publication number
FI57400C
FI57400C FI1064/72A FI106472A FI57400C FI 57400 C FI57400 C FI 57400C FI 1064/72 A FI1064/72 A FI 1064/72A FI 106472 A FI106472 A FI 106472A FI 57400 C FI57400 C FI 57400C
Authority
FI
Finland
Prior art keywords
diamino
formula
pyrimidine
group
ethanol
Prior art date
Application number
FI1064/72A
Other languages
English (en)
Finnish (fi)
Other versions
FI57400B (fi
Inventor
Barbara Roth
Original Assignee
Wellcome Found
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Wellcome Found filed Critical Wellcome Found
Application granted granted Critical
Publication of FI57400B publication Critical patent/FI57400B/fi
Publication of FI57400C publication Critical patent/FI57400C/fi

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/48—Two nitrogen atoms
    • C07D239/49—Two nitrogen atoms with an aralkyl radical, or substituted aralkyl radical, attached in position 5, e.g. trimethoprim
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/48—Two nitrogen atoms
    • H—ELECTRICITY
    • H01—ELECTRIC ELEMENTS
    • H01L—SEMICONDUCTOR DEVICES NOT COVERED BY CLASS H10
    • H01L2224/00—Indexing scheme for arrangements for connecting or disconnecting semiconductor or solid-state bodies and methods related thereto as covered by H01L24/00
    • H01L2224/01—Means for bonding being attached to, or being formed on, the surface to be connected, e.g. chip-to-package, die-attach, "first-level" interconnects; Manufacturing methods related thereto
    • H01L2224/26—Layer connectors, e.g. plate connectors, solder or adhesive layers; Manufacturing methods related thereto
    • H01L2224/2612—Auxiliary members for layer connectors, e.g. spacers

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Macromolecular Compounds Obtained By Forming Nitrogen-Containing Linkages In General (AREA)
FI1064/72A 1971-04-16 1972-04-14 Foerfarande foer framstaellning av 2,4-diamino-5-bensylpyrimidiner FI57400C (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB964071 1971-04-16
GB964071A GB1401612A (en) 1971-04-16 1971-04-16 2,4-diamino-5-benzylpyrimidines and preparations thereof

Publications (2)

Publication Number Publication Date
FI57400B FI57400B (fi) 1980-04-30
FI57400C true FI57400C (fi) 1980-08-11

Family

ID=9875907

Family Applications (1)

Application Number Title Priority Date Filing Date
FI1064/72A FI57400C (fi) 1971-04-16 1972-04-14 Foerfarande foer framstaellning av 2,4-diamino-5-bensylpyrimidiner

Country Status (25)

Country Link
US (1) US3822264A (xx)
JP (1) JPS5324433B1 (xx)
AR (1) AR193078A1 (xx)
AT (1) AT316560B (xx)
AU (1) AU468410B2 (xx)
BE (1) BE782154R (xx)
CA (1) CA978954A (xx)
CH (1) CH565159A5 (xx)
CS (2) CS178105B2 (xx)
DD (1) DD97653A6 (xx)
DE (2) DE2265413C2 (xx)
DK (1) DK132221C (xx)
ES (1) ES401796A2 (xx)
FI (1) FI57400C (xx)
FR (1) FR2133753B2 (xx)
GB (1) GB1401612A (xx)
HU (1) HU165865B (xx)
IE (1) IE36289B1 (xx)
IL (1) IL39221A (xx)
NL (1) NL163214C (xx)
NO (1) NO136046C (xx)
PL (1) PL75399B3 (xx)
SE (2) SE405118B (xx)
ZA (1) ZA722533B (xx)
ZM (1) ZM7072A1 (xx)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4515948A (en) * 1973-09-12 1985-05-07 Hoffmann-La Roche Inc. 2,4-Diamino-5-(4-amino and 4-dimethylamino-3,5-dimethoxy benzyl)pyrimidines
US4039543A (en) * 1974-12-24 1977-08-02 Hoffmann-La Roche Inc. Benzylpyrimidines
DE2720771C3 (de) * 1977-05-09 1979-11-29 Ludwig Heumann & Co Gmbh, 8500 Nuernberg 2,4-Diamino-5-(33-dimethoxy-4thioalkyl-benzyD-pyrimidine, Verfahren zu ihrer Herstellung und diese Verbindungen enthaltende Arzneimittel
DE3250132C2 (de) * 1981-11-09 1997-01-16 Mallinckrodt Veterinary Inc Verfahren zur Herstellung von 2,4-Diamino-5-benzyl-pyrimidinen und neue Zwischenprodukte des Verfahrens
CH664960A5 (de) * 1981-11-09 1988-04-15 Wellcome Found Verfahren zur herstellung von substituierten 2,4-diamino-5-benzylpyrimidinen.

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1720031A1 (de) * 1966-02-19 1972-08-03 Wellcome Found Biologisch wirksame 5-Benzylpyrimidin-Derivate und Verfahren zu ihrer Herstellung

Also Published As

Publication number Publication date
DE2218221B2 (de) 1978-05-24
BE782154R (fr) 1972-10-16
PL75399B3 (en) 1974-12-31
AU468410B2 (en) 1973-10-18
AR193078A1 (es) 1973-03-30
DE2218221C3 (de) 1979-02-01
ZM7072A1 (en) 1974-03-21
DE2265413B1 (de) 1980-04-10
FR2133753A2 (xx) 1972-12-01
CA978954A (en) 1975-12-02
NL7205046A (xx) 1972-10-18
ES401796A2 (es) 1975-03-01
DK132221B (da) 1975-11-10
CH565159A5 (xx) 1975-08-15
SE417097B (sv) 1981-02-23
IL39221A (en) 1975-11-25
CS178140B2 (xx) 1977-08-31
DD97653A6 (xx) 1973-05-14
ZA722533B (en) 1973-11-28
FR2133753B2 (xx) 1975-10-10
IE36289L (en) 1972-10-16
SE405118B (sv) 1978-11-20
DK132221C (da) 1976-04-20
US3822264A (en) 1974-07-02
JPS5324433B1 (xx) 1978-07-20
HU165865B (xx) 1974-11-28
NL163214C (nl) 1980-08-15
NO136046C (no) 1977-07-13
GB1401612A (en) 1975-07-16
SE7503993L (xx) 1975-04-08
AT316560B (de) 1974-07-25
DE2265413C2 (de) 1980-12-04
CS178105B2 (xx) 1977-08-31
FI57400B (fi) 1980-04-30
NL163214B (nl) 1980-03-17
DE2218221A1 (de) 1972-11-02
AU4117772A (en) 1973-10-18
NO136046B (xx) 1977-04-04
IE36289B1 (en) 1976-09-29
IL39221A0 (en) 1972-06-28

Similar Documents

Publication Publication Date Title
US4323570A (en) Substituted aminopyrimidines
FI73682B (fi) Foerfarande foer framstaellning av antiviralt 9-(1,3-dihydroxi-2-propoximetyl)guanin samt mellanprodukt.
SI9010633A (en) Process for preparing pteridine-4(3h)-ones and medicaments containing them
US2602794A (en) Process for preparation of x-amino-s
Roth et al. 2, 4-Diamino-5-benzylpyrimidines as antibacterial agents. 4. 6-Substituted trimethoprim derivatives from phenolic Mannich intermediates. Application to the synthesis of trimethoprim and 3, 5-dialkylbenzyl analogs
FI57400B (fi) Foerfarande foer framstaellning av 2,4-diamino-5-bensylpyrimidiner
US3071587A (en) Cyanoethyl-pteridines
CN110981816B (zh) 一种4-氨基-2.6-二甲氧基嘧啶的合成方法
Rose 663. New syntheses based on 5-aminopyrimidines
US4027025A (en) 8-Azapurine derivatives
DK156722B (da) Analogifremgangsmaade til fremstilling af 2-piperazinopyrimidinderivater
US3432493A (en) Substituted sulfanilamides
HU180321B (en) Process for producing 6- and 9-substituted 2-amino-purine derivatives
ROTH et al. 5-Arylthiopyrimidines. II. 2-and 4-Alkylamino and 4-Amino Derivatives1
US4024145A (en) Benzylpyrimidine derivatives
US4066645A (en) Derivatives of pyrazolo [1,5-a]pyrido[3,4-e]pyrimidine
NZ194228A (en) 2-(1,4-diazacycloalk-1-yl)-4-(morpholino or thiomorpholino)-8-substituted pyrimido(4,5-b)pyrimidines
NO783775L (no) 2,4-diamino-5-benzylpyrimidiner og fremgangsmaate ved fremstilling av disse
US3849407A (en) 5-benzyl pyrimidines intermediates
FI56375C (fi) Saosom mellanprodukt anvaendbar beta-hydroxy-beta-3,4,5-trialkoxyfenetylmetylsulfon eller sulfoxid foer framstaellning av antibakteriska 2,4-diamino-5-bensylpyrimidiner
US3772289A (en) Alkyl substituted benzyl pyrimidines
Russell et al. The Reaction of Aromatic Nitriles with Guanidine1
US5698580A (en) Antiviral agent containing benzodithiin derivative as active ingredient
US4179509A (en) (Substituted 2-carboxyanilino)nicotinic acids as inhibitors of allergic reactions
FI65991C (fi) Foerfarande foer framstaellning av terapeutiskt vaerdefull 5((3,4,5-trimetoxifenyl)metyl)-2,4-pyrimidindiamin