FI105917B - Menetelmä terapeuttisesti aktiivisen 5-kloori-2,3-dihydro-2,2-dimetyylibentsofuraani-7-karboksyylihappo-oktahydro-3-hydroksi-2,6-metano-2H-kinolitsin-8-yyliesterin valmistamiseksi - Google Patents
Menetelmä terapeuttisesti aktiivisen 5-kloori-2,3-dihydro-2,2-dimetyylibentsofuraani-7-karboksyylihappo-oktahydro-3-hydroksi-2,6-metano-2H-kinolitsin-8-yyliesterin valmistamiseksi Download PDFInfo
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- FI105917B FI105917B FI943872A FI943872A FI105917B FI 105917 B FI105917 B FI 105917B FI 943872 A FI943872 A FI 943872A FI 943872 A FI943872 A FI 943872A FI 105917 B FI105917 B FI 105917B
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- farm farm
- methano
- dihydro
- chloro
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Classifications
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- C—CHEMISTRY; METALLURGY
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- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
- C07D471/18—Bridged systems
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- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/26—Psychostimulants, e.g. nicotine, cocaine
Landscapes
- Health & Medical Sciences (AREA)
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- Organic Chemistry (AREA)
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- Neurosurgery (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Psychiatry (AREA)
- Pain & Pain Management (AREA)
- Hospice & Palliative Care (AREA)
- Otolaryngology (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP92400474 | 1992-02-24 | ||
| EP92400474 | 1992-02-24 | ||
| PCT/US1993/000880 WO1993017019A1 (en) | 1992-02-24 | 1993-02-03 | 2,6-methano-2h-quinolizin derivative as 5-ht3-receptor antagonist |
| US9300880 | 1993-02-03 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| FI943872L FI943872L (fi) | 1994-08-23 |
| FI943872A0 FI943872A0 (fi) | 1994-08-23 |
| FI105917B true FI105917B (fi) | 2000-10-31 |
Family
ID=8211614
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| FI943872A FI105917B (fi) | 1992-02-24 | 1994-08-23 | Menetelmä terapeuttisesti aktiivisen 5-kloori-2,3-dihydro-2,2-dimetyylibentsofuraani-7-karboksyylihappo-oktahydro-3-hydroksi-2,6-metano-2H-kinolitsin-8-yyliesterin valmistamiseksi |
Country Status (14)
| Country | Link |
|---|---|
| EP (1) | EP0628043A1 (enExample) |
| JP (1) | JPH07504192A (enExample) |
| KR (1) | KR100287933B1 (enExample) |
| AU (1) | AU675060B2 (enExample) |
| CA (1) | CA2130563C (enExample) |
| FI (1) | FI105917B (enExample) |
| HU (1) | HU216831B (enExample) |
| IL (1) | IL104821A (enExample) |
| MX (1) | MX9300948A (enExample) |
| NO (1) | NO943101L (enExample) |
| NZ (1) | NZ249346A (enExample) |
| TW (1) | TW226374B (enExample) |
| WO (1) | WO1993017019A1 (enExample) |
| ZA (1) | ZA931146B (enExample) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2002537255A (ja) | 1999-02-18 | 2002-11-05 | ノバルティス アクチエンゲゼルシャフト | リウマチ性炎症性プロセスに対する５−ｈｔ３レセプターアンタゴニストの全身的使用 |
| US8524731B2 (en) | 2005-03-07 | 2013-09-03 | The University Of Chicago | Use of opioid antagonists to attenuate endothelial cell proliferation and migration |
| US8518962B2 (en) | 2005-03-07 | 2013-08-27 | The University Of Chicago | Use of opioid antagonists |
| US9662325B2 (en) | 2005-03-07 | 2017-05-30 | The University Of Chicago | Use of opioid antagonists to attenuate endothelial cell proliferation and migration |
| MX2007010833A (es) | 2005-03-07 | 2009-02-17 | Univ Chicago | Uso de antagonistas opioides para atenuar proliferacion y migracion de células endoteliales. |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0329932B1 (en) * | 1988-02-23 | 1995-10-18 | Merrell Pharmaceuticals Inc. | Use of quinolizine and quinolizinone derivatives in the manufacture of medicaments |
| EP0517984A1 (en) * | 1991-06-11 | 1992-12-16 | Merrell Dow Pharmaceuticals Inc. | Derivatives of amide analogs of certain methano bridged quinolizines |
-
1993
- 1993-02-03 KR KR1019940702945A patent/KR100287933B1/ko not_active Expired - Lifetime
- 1993-02-03 JP JP5514868A patent/JPH07504192A/ja active Pending
- 1993-02-03 WO PCT/US1993/000880 patent/WO1993017019A1/en not_active Ceased
- 1993-02-03 EP EP93904797A patent/EP0628043A1/en not_active Withdrawn
- 1993-02-03 AU AU36034/93A patent/AU675060B2/en not_active Expired
- 1993-02-03 HU HU9402436A patent/HU216831B/hu unknown
- 1993-02-03 NZ NZ249346A patent/NZ249346A/en not_active IP Right Cessation
- 1993-02-03 CA CA002130563A patent/CA2130563C/en not_active Expired - Lifetime
- 1993-02-18 ZA ZA931146A patent/ZA931146B/xx unknown
- 1993-02-19 TW TW082101189A patent/TW226374B/zh not_active IP Right Cessation
- 1993-02-22 IL IL10482193A patent/IL104821A/xx not_active IP Right Cessation
- 1993-02-22 MX MX9300948A patent/MX9300948A/es unknown
-
1994
- 1994-08-23 NO NO943101A patent/NO943101L/no unknown
- 1994-08-23 FI FI943872A patent/FI105917B/fi not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| MX9300948A (es) | 1993-08-01 |
| CA2130563C (en) | 1997-11-11 |
| HU216831B (hu) | 1999-09-28 |
| ZA931146B (en) | 1993-09-14 |
| NO943101D0 (no) | 1994-08-23 |
| NO943101L (no) | 1994-08-23 |
| HUT68249A (en) | 1995-06-28 |
| AU675060B2 (en) | 1997-01-23 |
| FI943872L (fi) | 1994-08-23 |
| KR100287933B1 (ko) | 2001-05-02 |
| EP0628043A1 (en) | 1994-12-14 |
| JPH07504192A (ja) | 1995-05-11 |
| NZ249346A (en) | 1995-10-26 |
| AU3603493A (en) | 1993-09-13 |
| CA2130563A1 (en) | 1993-09-02 |
| IL104821A0 (en) | 1993-06-10 |
| TW226374B (enExample) | 1994-07-11 |
| WO1993017019A1 (en) | 1993-09-02 |
| KR950700297A (ko) | 1995-01-16 |
| HU9402436D0 (en) | 1994-10-28 |
| IL104821A (en) | 1997-01-10 |
| FI943872A0 (fi) | 1994-08-23 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| PC | Transfer of assignment of patent |
Owner name: AVENTIS INC. Free format text: AVENTIS INC. |
|
| PC | Transfer of assignment of patent |
Owner name: AVENTISUB II INC. Free format text: AVENTISUB II INC. |
|
| MA | Patent expired |