ES8604603A1 - Un procedimiento para preparar derivados de 4,5,6,7-tetrahidrotiazolo (4,5-c) piridina - Google Patents

Un procedimiento para preparar derivados de 4,5,6,7-tetrahidrotiazolo (4,5-c) piridina

Info

Publication number
ES8604603A1
ES8604603A1 ES538305A ES538305A ES8604603A1 ES 8604603 A1 ES8604603 A1 ES 8604603A1 ES 538305 A ES538305 A ES 538305A ES 538305 A ES538305 A ES 538305A ES 8604603 A1 ES8604603 A1 ES 8604603A1
Authority
ES
Spain
Prior art keywords
ulcer
tetrahydrothiazole
pyridine derivatives
gastric secretion
secretion inhibiting
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES538305A
Other languages
English (en)
Other versions
ES538305A0 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Italia SRL
Original Assignee
Farmitalia Carlo Erba SRL
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Farmitalia Carlo Erba SRL filed Critical Farmitalia Carlo Erba SRL
Publication of ES8604603A1 publication Critical patent/ES8604603A1/es
Publication of ES538305A0 publication Critical patent/ES538305A0/es
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

PROCEDIMIENTO PARA PREPARAR DERIVADOS DE 4,5,6,7-TERTRAHIDROTIAZOLO4,5-CPIRIDINA. CONSISTENTE EN HACER REACCIONAR UN COMPUESTO DE FORMULA (II) CON UNO DE FORMULA (II) EN DIMETILFORMAMIDA O ACETONITRILO A UNA TEMPERATURA DE 0 A 120J PARA OBTENER COMPUESTOS DE FORMULA (I) O SUS SALES DE ADICION DE ACIDO FARMACEUTICAMENTE ACEPTABLES. SIENDO: A) R1 Y R2 INDEPENDIENTEMENTE H O UN GRUPO ORGANICO; O B) R2 ES H Y R1 ES R6-NH-CFNR7 DONDE R6 Y R7 REPRESENTAN INDEPENDIENTEMENTE H O UN GRUPO ORGANICO; O C) R1 Y R2 UNIDOS FORMAN UN ANILLO HETEROCICLICO; N ES 0 A 3; X ES O, S O NH; Y R3 UN GRUPO FENILETILO, ALQUILO LINEAL O RAMIFICADO, SATURADO O INSATURADO QUE CONTIENE DE 1 A 6 C, Y OTROS. SE UTILIZAN COMO AGENTES ANTI-ULCEROSOS.-
ES538305A 1983-12-16 1984-12-05 Un procedimiento para preparar derivados de 4,5,6,7-tetrahidrotiazolo (4,5-c) piridina Expired ES8604603A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB838333514A GB8333514D0 (en) 1983-12-16 1983-12-16 Tetrahydrothiazolo(5 4-c)pyridine derivatives

Publications (2)

Publication Number Publication Date
ES8604603A1 true ES8604603A1 (es) 1986-02-01
ES538305A0 ES538305A0 (es) 1986-02-01

Family

ID=10553370

Family Applications (1)

Application Number Title Priority Date Filing Date
ES538305A Expired ES8604603A1 (es) 1983-12-16 1984-12-05 Un procedimiento para preparar derivados de 4,5,6,7-tetrahidrotiazolo (4,5-c) piridina

Country Status (27)

Country Link
US (1) US4624956A (es)
JP (1) JPS60146893A (es)
KR (1) KR910009213B1 (es)
AT (1) AT391701B (es)
AU (1) AU568894B2 (es)
BE (1) BE901278A (es)
CA (1) CA1244827A (es)
CH (1) CH660739A5 (es)
CS (1) CS244145B2 (es)
DE (1) DE3445192A1 (es)
DK (1) DK598284A (es)
ES (1) ES8604603A1 (es)
FI (1) FI77248C (es)
FR (1) FR2556725B1 (es)
GB (2) GB8333514D0 (es)
GR (1) GR81232B (es)
HU (1) HU193724B (es)
IL (1) IL73810A (es)
IT (1) IT1221007B (es)
NL (1) NL8403801A (es)
NO (1) NO165595C (es)
NZ (1) NZ210519A (es)
PH (1) PH21312A (es)
PT (1) PT79681B (es)
SE (1) SE455096B (es)
SU (1) SU1364240A3 (es)
ZA (1) ZA849770B (es)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB2173187B (en) * 1985-03-23 1988-05-18 Erba Farmitalia Condensed 2-substituted thiazole derivatives
JPH03148283A (ja) * 1989-11-02 1991-06-25 Terumo Corp チアゾール誘導体またはその塩ならびにこれらを含有する抗潰瘍剤
JPH0618334A (ja) * 1992-06-29 1994-01-25 Mikuni Seisakusho:Kk 被加熱物の温度測定装置
CU22676A1 (es) 1996-06-21 2001-11-16 Univ Las Villas Composición microcida para el control de contaminantes en procesos de producción de vitroplantas
US5718151A (en) * 1996-10-01 1998-02-17 Breed Automotive Technology, Inc. Steering wheel mounting
AR041952A1 (es) * 2002-11-14 2005-06-01 Novartis Ag N-sulfonilaminotiazol
CL2004000553A1 (es) * 2003-03-20 2005-02-04 Actelion Pharmaceuticals Ltd Uso de compuestos derivados de guanidina como antagonistas del receptor de neuropeptido ff; compuestos derivados de guanidina; procedimientos de preparacion; y composicion farmaceutica que los comprende.
US20220009945A1 (en) * 2018-11-02 2022-01-13 Aicuris Gmbh & Co. Kg Novel urea 6,7-dihydro-4h-thiazole[5,4-c]pyridines active against the hepatitis b virus (hbv)

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1620508A1 (de) * 1965-07-23 1969-09-18 Thomae Gmbh Dr K Verfahren zur Herstellung neuer 4,5,6,7-Tetrahydrothiazolo-[5,4-c]-pyridine
DE2205065A1 (de) * 1972-02-03 1973-08-16 Thomae Gmbh Dr K Neue 4,5,6,7-tetrahydro-thiazolo eckige klammer auf 4,5-c eckige klammer zu pyridine
AR208500A1 (es) * 1972-06-14 1977-02-15 Merck & Co Inc Procedimiento para la preparacion de derivados de oxazolo(4,5-b)-piridinas
CA1131226A (en) * 1978-09-28 1982-09-07 Tomohiko Munakata Heterocyclic compounds
DE3134933A1 (de) * 1981-09-03 1983-03-31 Hoechst Ag, 6230 Frankfurt "harnstoffderivate, verfahren zu ihrer herstellung und diese enthaltende medikamente sowie deren verwendung"
CA1260474A (en) * 1984-12-03 1989-09-26 Raymond A. Stokbroekx Benzoxazol- and benzothiazolamine derivatives

Also Published As

Publication number Publication date
DE3445192A1 (de) 1985-06-27
SU1364240A3 (ru) 1987-12-30
NO845038L (no) 1985-06-17
DE3445192C2 (es) 1993-02-18
DK598284D0 (da) 1984-12-13
HUT37625A (en) 1986-01-23
AT391701B (de) 1990-11-26
FR2556725B1 (fr) 1987-11-27
NO165595B (no) 1990-11-26
BE901278A (fr) 1985-03-29
NO165595C (no) 1991-03-06
DK598284A (da) 1985-06-17
FI844900A0 (fi) 1984-12-12
JPH032158B2 (es) 1991-01-14
ATA392484A (de) 1990-05-15
IL73810A (en) 1988-02-29
HU193724B (en) 1987-11-30
IT1221007B (it) 1990-06-21
CA1244827A (en) 1988-11-15
FR2556725A1 (fr) 1985-06-21
JPS60146893A (ja) 1985-08-02
GB2153816B (en) 1987-10-21
FI77248B (fi) 1988-10-31
AU3651784A (en) 1985-06-20
NL8403801A (nl) 1985-07-16
FI77248C (fi) 1989-02-10
KR850004756A (ko) 1985-07-27
CS244145B2 (en) 1986-07-17
PT79681A (en) 1985-01-01
IT8424039A0 (it) 1984-12-13
IL73810A0 (en) 1985-03-31
FI844900L (fi) 1985-06-17
US4624956A (en) 1986-11-25
CS961384A2 (en) 1985-08-15
KR910009213B1 (ko) 1991-11-05
GB8333514D0 (en) 1984-01-25
CH660739A5 (de) 1987-06-15
SE455096B (sv) 1988-06-20
GR81232B (en) 1985-04-16
ZA849770B (en) 1985-08-28
NZ210519A (en) 1988-04-29
ES538305A0 (es) 1986-02-01
AU568894B2 (en) 1988-01-14
PH21312A (en) 1987-09-28
PT79681B (en) 1986-12-10
SE8406338D0 (sv) 1984-12-12
GB8431161D0 (en) 1985-01-23
SE8406338L (sv) 1985-06-17
GB2153816A (en) 1985-08-29

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Legal Events

Date Code Title Description
FD1A Patent lapsed

Effective date: 19970612