ES521224A0 - Un procedimiento para la preparacion de nuevos derivados de carbapenem. - Google Patents

Un procedimiento para la preparacion de nuevos derivados de carbapenem.

Info

Publication number
ES521224A0
ES521224A0 ES521224A ES521224A ES521224A0 ES 521224 A0 ES521224 A0 ES 521224A0 ES 521224 A ES521224 A ES 521224A ES 521224 A ES521224 A ES 521224A ES 521224 A0 ES521224 A0 ES 521224A0
Authority
ES
Spain
Prior art keywords
procedure
preparation
carbapenem derivatives
new carbapenem
new
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
ES521224A
Other languages
English (en)
Other versions
ES8405399A1 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Bristol Myers Co
Original Assignee
Bristol Myers Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bristol Myers Co filed Critical Bristol Myers Co
Publication of ES8405399A1 publication Critical patent/ES8405399A1/es
Publication of ES521224A0 publication Critical patent/ES521224A0/es
Granted legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D477/00Heterocyclic compounds containing 1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. carbapenicillins, thienamycins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulphur-containing hetero ring
    • C07D477/10Heterocyclic compounds containing 1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. carbapenicillins, thienamycins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulphur-containing hetero ring with hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 4, and with a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
    • C07D477/12Heterocyclic compounds containing 1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. carbapenicillins, thienamycins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulphur-containing hetero ring with hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 4, and with a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2 with hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, attached in position 6
    • C07D477/16Heterocyclic compounds containing 1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. carbapenicillins, thienamycins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulphur-containing hetero ring with hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 4, and with a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2 with hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, attached in position 6 with hetero atoms or carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 3
    • C07D477/20Sulfur atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
ES521224A 1982-04-08 1983-04-05 Un procedimiento para la preparacion de nuevos derivados de carbapenem. Granted ES521224A0 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US36662782A 1982-04-08 1982-04-08

Publications (2)

Publication Number Publication Date
ES8405399A1 ES8405399A1 (es) 1984-06-01
ES521224A0 true ES521224A0 (es) 1984-06-01

Family

ID=23443823

Family Applications (1)

Application Number Title Priority Date Filing Date
ES521224A Granted ES521224A0 (es) 1982-04-08 1983-04-05 Un procedimiento para la preparacion de nuevos derivados de carbapenem.

Country Status (25)

Country Link
JP (1) JPS58188887A (es)
KR (1) KR880001055B1 (es)
AT (1) AT383126B (es)
AU (1) AU567092B2 (es)
BE (1) BE896407A (es)
CA (1) CA1198440A (es)
CH (1) CH661927A5 (es)
DE (1) DE3312517A1 (es)
DK (1) DK155983A (es)
ES (1) ES521224A0 (es)
FI (1) FI74009C (es)
FR (1) FR2524888B1 (es)
GB (1) GB2118183B (es)
GR (1) GR78822B (es)
HU (1) HU190716B (es)
IE (1) IE55225B1 (es)
IL (1) IL68295A0 (es)
IT (1) IT1168854B (es)
LU (1) LU84739A1 (es)
MY (1) MY8700945A (es)
NL (1) NL8301193A (es)
OA (1) OA07395A (es)
PT (1) PT76518B (es)
SE (1) SE460197B (es)
ZA (1) ZA832411B (es)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4683301A (en) * 1982-04-08 1987-07-28 Bristol-Myers Company Carbapenem antibiotics
US4552696A (en) * 1982-04-09 1985-11-12 Bristol-Myers Company Carbapenem antibiotics
US4536335A (en) * 1982-06-18 1985-08-20 Bristol-Myers Company Carbapenem antibiotics
AT396473B (de) * 1984-10-02 1993-09-27 Bristol Myers Squibb Co Verfahren zur herstellung von neuen carbapenemderivaten
US4665169A (en) * 1985-09-11 1987-05-12 Bristol-Myers Company Carbapenem antibiotics

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU531084B2 (en) * 1977-10-19 1983-08-11 Merck & Co., Inc. Azetidine derivatives
EP0017992A1 (en) * 1979-04-19 1980-10-29 Merck & Co. Inc. 2-Substituted-6-substituted-1-carbadethiapen-2-em-3-carboxylic acids, processes for preparing them, antibiotic pharmaceutical compositions containing same and process for preparing intermediates
EP0038869A1 (en) * 1980-04-30 1981-11-04 Merck & Co. Inc. Process for the preparation of 1-carbapenems, and intermediates for their preparation
HU185493B (en) * 1981-12-30 1985-02-28 Richter Gedeon Vegyeszet Process for producing new azabicyclo-bracket-3.2.0-bracket closedheptene derivatives
US4552696A (en) * 1982-04-09 1985-11-12 Bristol-Myers Company Carbapenem antibiotics
US4536335A (en) * 1982-06-18 1985-08-20 Bristol-Myers Company Carbapenem antibiotics

Also Published As

Publication number Publication date
ZA832411B (en) 1983-12-28
PT76518B (en) 1986-02-06
AU1319883A (en) 1983-10-13
SE8301928L (sv) 1983-12-02
MY8700945A (en) 1987-12-31
IL68295A0 (en) 1983-07-31
CA1198440A (en) 1985-12-24
IT8348061A0 (it) 1983-04-07
IE830800L (en) 1983-10-08
AT383126B (de) 1987-05-25
GB2118183A (en) 1983-10-26
IE55225B1 (en) 1990-07-04
KR880001055B1 (ko) 1988-06-18
DK155983D0 (da) 1983-04-07
SE460197B (sv) 1989-09-18
GB2118183B (en) 1985-11-27
FI74009B (fi) 1987-08-31
DE3312517C2 (es) 1991-10-31
PT76518A (en) 1983-05-01
CH661927A5 (de) 1987-08-31
FI74009C (fi) 1987-12-10
JPS58188887A (ja) 1983-11-04
BE896407A (fr) 1983-10-07
GR78822B (es) 1984-10-02
OA07395A (fr) 1984-06-30
FR2524888B1 (fr) 1985-12-13
HU190716B (en) 1986-10-28
JPH0524156B2 (es) 1993-04-06
SE8301928D0 (sv) 1983-04-07
FI831135A0 (fi) 1983-04-05
ES8405399A1 (es) 1984-06-01
FI831135L (fi) 1983-10-09
DE3312517A1 (de) 1983-10-20
FR2524888A1 (fr) 1983-10-14
NL8301193A (nl) 1983-11-01
ATA125583A (de) 1986-10-15
DK155983A (da) 1983-10-09
LU84739A1 (fr) 1983-12-05
GB8309505D0 (en) 1983-05-11
AU567092B2 (en) 1987-11-12
KR840004429A (ko) 1984-10-15
IT1168854B (it) 1987-05-20

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Legal Events

Date Code Title Description
FD1A Patent lapsed

Effective date: 19970519