ES482598A1 - Un procedimiento para la preparacion de n-(diaminofosfinil) aril-carboxamidas. - Google Patents

Un procedimiento para la preparacion de n-(diaminofosfinil) aril-carboxamidas.

Info

Publication number
ES482598A1
ES482598A1 ES482598A ES482598A ES482598A1 ES 482598 A1 ES482598 A1 ES 482598A1 ES 482598 A ES482598 A ES 482598A ES 482598 A ES482598 A ES 482598A ES 482598 A1 ES482598 A1 ES 482598A1
Authority
ES
Spain
Prior art keywords
diaminophosphinyl
arylcarboxamides
inhibitors
useful
series
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES482598A
Other languages
English (en)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
ATK Launch Systems LLC
Original Assignee
Morton Norwich Products Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Morton Norwich Products Inc filed Critical Morton Norwich Products Inc
Publication of ES482598A1 publication Critical patent/ES482598A1/es
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/06—Phosphorus compounds without P—C bonds
    • C07F9/22—Amides of acids of phosphorus
    • C07F9/26—Amides of acids of phosphorus containing P-halide groups
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/06—Phosphorus compounds without P—C bonds
    • C07F9/22—Amides of acids of phosphorus
    • C07F9/224—Phosphorus triamides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/553—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having one nitrogen atom as the only ring hetero atom
    • C07F9/576—Six-membered rings
    • C07F9/58—Pyridine rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)

Abstract

Una serie de N-(diaminofosfinil) arilcarboxamidas, útiles como inhibidores de la enzima ureasa. Esta invención se refiere a compuestos químicos. Mas particularmente, se refiere a una serie de N-(diaminofosfinil) arilcarboxamidas, de fórmula **(Fórmula)** donde R es 3-piridilo, 2-furilo, 2-naftilo, cinamenilo, bencilo, fenilo o fenilo sustituido por grupos 3- ó 4-nitro, 4-halo, 4-amino, 4-alcoxi (inferior), 4-alquilo (inferior), 2- metilo, 2,3-dimetilo, 2,4-dimetilo, 2,4,6-trimetilo, 3- trifluorometilo, 4-ciano, 4-fenilo o 3-fenoxi.
ES482598A 1978-07-19 1979-07-18 Un procedimiento para la preparacion de n-(diaminofosfinil) aril-carboxamidas. Expired ES482598A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US05/925,968 US4182881A (en) 1978-07-19 1978-07-19 N-[Diaminophosphinyl]arylcarboxamides

Publications (1)

Publication Number Publication Date
ES482598A1 true ES482598A1 (es) 1980-07-01

Family

ID=25452508

Family Applications (1)

Application Number Title Priority Date Filing Date
ES482598A Expired ES482598A1 (es) 1978-07-19 1979-07-18 Un procedimiento para la preparacion de n-(diaminofosfinil) aril-carboxamidas.

Country Status (15)

Country Link
US (1) US4182881A (es)
JP (1) JPS5515461A (es)
AU (1) AU521741B2 (es)
BE (1) BE877737A (es)
CA (1) CA1125289A (es)
CH (1) CH642084A5 (es)
DE (1) DE2928831C2 (es)
ES (1) ES482598A1 (es)
FR (1) FR2431505A1 (es)
GB (1) GB2025974B (es)
IE (1) IE48326B1 (es)
IT (1) IT1120421B (es)
MX (1) MX5375E (es)
NL (1) NL190781C (es)
SE (1) SE441831B (es)

Families Citing this family (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5899490A (ja) * 1981-10-19 1983-06-13 Eisai Co Ltd リン酸アミド誘導体およびその製造方法ならびにそれを含有する医薬
EP0119494A1 (en) * 1983-03-16 1984-09-26 Allied Corporation Urease inhibited urea based fertilizer compositions containing phosphorus compounds
US4539037A (en) * 1983-03-16 1985-09-03 Allied Corporation Urease inhibited urea based fertilizer compositions containing N-aryl-N-aliphatic phosphorotriamide compounds
US4517002A (en) * 1983-03-16 1985-05-14 Allied Corporation Phosphorodiamide urease inhibitors and urease inhibited urea based fertilizer compositions
US4530714A (en) * 1983-03-16 1985-07-23 Allied Corporation N-aliphatic and N,N-aliphatic phosphoric triamide urease inhibitors and urease inhibited urea based fertilizer compositions
US4540428A (en) * 1983-03-16 1985-09-10 Allied Corporation Phosphorotriamidate urease inhibitors and urease inhibited urea based fertilizer compositions
US4518413A (en) * 1983-06-06 1985-05-21 Allied Corporation Poly-phosphorodiamide urease inhibitors and urease inhibited urea based fertilizer compositions
US4517003A (en) * 1983-06-08 1985-05-14 Allied Corporation N-acyl phosphoric triamide urease inhibitors and urease inhibited urea based fertilizer compositions
US4517007A (en) * 1983-06-09 1985-05-14 Allied Corporation Phosphoroamide urease inhibitors and urease inhibited urea based fertilizer compositions
US4528020A (en) * 1983-06-16 1985-07-09 Allied Corporation Urease inhibited urea based fertilizer compositions
US4824783A (en) * 1983-12-20 1989-04-25 Enichem S.P.A. Oxidized sulfur derivatives of diaminophosphinyl compounds as urease inhibitors
US4629491A (en) * 1983-12-20 1986-12-16 Allied Corporation Oxidized sulfur derivatives of diaminophosphinyl compounds as urease inhibitors and urease inhibited urea based fertilizer compositions
US4624695A (en) * 1983-12-20 1986-11-25 Allied Corporation O-diaminophosphinyl derivatives of oximes as urease inhibitors
US4800194A (en) * 1985-08-01 1989-01-24 Norwich Eaton Pharmaceuticals, Inc. Acylphosphorotriamides useful as lipid-altering agents
US4668667A (en) * 1985-08-01 1987-05-26 Norwich Eaton Pharmaceuticals, Inc. Acylphosphorotriamides useful as lipid-altering agents
EP0852498A1 (en) * 1995-09-26 1998-07-15 Takeda Chemical Industries, Ltd. Phosphorylamides, their preparation and use
AU6422798A (en) * 1997-03-25 1998-10-20 Takeda Chemical Industries Ltd. Stabilized urease inhibitor
DE10118322A1 (de) * 2001-04-12 2002-10-17 Piesteritz Stickstoff Heterozyklisch-substituierte (Thio)Phosphorsäuretriamide, Verfahren zu ihrer Herstellung und deren Verwendung als Mittel zur Regulierung bzw.Hemmung der enzymatischen Harnstoff-Hydrolyse
WO2013182469A2 (en) 2012-06-08 2013-12-12 Basf Se Odour-control superabsorbent
DE102013012500A1 (de) 2013-07-26 2015-01-29 Skw Stickstoffwerke Piesteritz Gmbh Verwendung von Phosphorsäureamiden als Mittel zur Verbesserung der Trockenstresstoleranz

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3317637A (en) * 1961-06-30 1967-05-02 Dow Chemical Co N-haloacylphosphoric amides
US3321516A (en) * 1963-12-06 1967-05-23 Pennsalt Chemicals Corp Dialkylthiocarbamylphosphonic diamides
GB1448241A (en) * 1973-01-23 1976-09-02 Ici Ltd Thiophosphorus acid amides and their use as inhibitors of premature vulcanisation of rubber

Also Published As

Publication number Publication date
IT1120421B (it) 1986-03-26
IE790790L (en) 1980-01-19
GB2025974B (en) 1982-10-27
FR2431505B1 (es) 1984-07-13
DE2928831C2 (de) 1986-10-09
SE441831B (sv) 1985-11-11
FR2431505A1 (fr) 1980-02-15
BE877737A (fr) 1980-01-16
AU4676379A (en) 1980-01-24
CA1125289A (en) 1982-06-08
NL190781C (nl) 1994-08-16
JPS6254117B2 (es) 1987-11-13
NL190781B (nl) 1994-03-16
GB2025974A (en) 1980-01-30
SE7905922L (sv) 1980-01-20
IE48326B1 (en) 1984-12-12
CH642084A5 (de) 1984-03-30
DE2928831A1 (de) 1980-01-31
IT7949148A0 (it) 1979-05-23
JPS5515461A (en) 1980-02-02
US4182881A (en) 1980-01-08
NL7905138A (nl) 1980-01-22
MX5375E (es) 1983-06-30
AU521741B2 (en) 1982-04-29

Similar Documents

Publication Publication Date Title
ES482598A1 (es) Un procedimiento para la preparacion de n-(diaminofosfinil) aril-carboxamidas.
DE2966707D1 (en) Enzymatic processes
ZA772716B (en) Process for the determination of substrates or enzyme activities
BE828052A (fr) Supports mineraux greffes pour fixation d'enzymes
AU4686479A (en) Encapsulatio of nutrients
JPS5664786A (en) Novel microorganism for prducing proteolytic enzyme
JPS5589230A (en) Angiotensin conversion enzyme inhibitor
JPS5221390A (en) Enzymatic reacting method utilizing microorganzsm
GB2044294B (en) Enzymatic bating process
ES460204A1 (es) Un procedimiento para la preparacion de acidos ureido(susti-tuidos) acetohidroxamicos.
BG35746A3 (en) Method for preparing 1- cyclohexenylmethylpyrolidines
IT7819138A0 (it) Procedimento per la coltura di microrganismi.
YU192879A (en) Process for performing enzymatic determinations
AU523544B2 (en) Enzymatic softening of furs
AU3624078A (en) T-factor, coa-spc substantially free of proteolytic enzymes
GB2016497A (en) Microbiological production of amylase inhibitor
SU484250A1 (ru) Способ получени иммобилизованных ферментов
SU686454A1 (ru) Магнитореологическая суспензия
ES477715A1 (es) Un procedimiento para la preparacion de 5-fenil-2-oxazol carboximidamidas.
IT7850955A0 (it) Procedimento per la coltura aerobica di microorganismi
GB1556398A (en) Immobilization of enzymes
SU586662A1 (ru) Способ получения биомассы
JPS54105286A (en) Production of immovilized bacterial enzyme
JPS5322496A (en) Enzyme reaction inhibitor
SU900579A1 (ru) Способ получения диимида пиромеллитовой кислоты