IT7949148A0 - N-(diamminofosfinil)arilcarbossammi di aventi attivita' inibitrice dell'enzima ureasi - Google Patents

N-(diamminofosfinil)arilcarbossammi di aventi attivita' inibitrice dell'enzima ureasi

Info

Publication number
IT7949148A0
IT7949148A0 IT7949148A IT4914879A IT7949148A0 IT 7949148 A0 IT7949148 A0 IT 7949148A0 IT 7949148 A IT7949148 A IT 7949148A IT 4914879 A IT4914879 A IT 4914879A IT 7949148 A0 IT7949148 A0 IT 7949148A0
Authority
IT
Italy
Prior art keywords
diaminophosphinil
arylcarboxames
inhibiting activity
enzyme inhibiting
urease enzyme
Prior art date
Application number
IT7949148A
Other languages
English (en)
Other versions
IT1120421B (it
Original Assignee
Morton Norwich Products Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Morton Norwich Products Inc filed Critical Morton Norwich Products Inc
Publication of IT7949148A0 publication Critical patent/IT7949148A0/it
Application granted granted Critical
Publication of IT1120421B publication Critical patent/IT1120421B/it

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic System
    • C07F9/02Phosphorus compounds
    • C07F9/06Phosphorus compounds without P—C bonds
    • C07F9/22Amides of acids of phosphorus
    • C07F9/26Amides of acids of phosphorus containing P-halide groups
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic System
    • C07F9/02Phosphorus compounds
    • C07F9/06Phosphorus compounds without P—C bonds
    • C07F9/22Amides of acids of phosphorus
    • C07F9/224Phosphorus triamides
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic System
    • C07F9/02Phosphorus compounds
    • C07F9/547Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/553Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having one nitrogen atom as the only ring hetero atom
    • C07F9/576Six-membered rings
    • C07F9/58Pyridine rings
IT49148/79A 1978-07-19 1979-05-23 N-(diamminofosfinil)arilcarbossammi di aventi attivita' inbitrice del l'enzima ureasi IT1120421B (it)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US05/925,968 US4182881A (en) 1978-07-19 1978-07-19 N-[Diaminophosphinyl]arylcarboxamides

Publications (2)

Publication Number Publication Date
IT7949148A0 true IT7949148A0 (it) 1979-05-23
IT1120421B IT1120421B (it) 1986-03-26

Family

ID=25452508

Family Applications (1)

Application Number Title Priority Date Filing Date
IT49148/79A IT1120421B (it) 1978-07-19 1979-05-23 N-(diamminofosfinil)arilcarbossammi di aventi attivita' inbitrice del l'enzima ureasi

Country Status (15)

Country Link
US (1) US4182881A (it)
JP (1) JPS5515461A (it)
AU (1) AU521741B2 (it)
BE (1) BE877737A (it)
CA (1) CA1125289A (it)
CH (1) CH642084A5 (it)
DE (1) DE2928831C2 (it)
ES (1) ES482598A1 (it)
FR (1) FR2431505A1 (it)
GB (1) GB2025974B (it)
IE (1) IE48326B1 (it)
IT (1) IT1120421B (it)
MX (1) MX5375E (it)
NL (1) NL190781C (it)
SE (1) SE441831B (it)

Families Citing this family (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5899490A (ja) * 1981-10-19 1983-06-13 Eisai Co Ltd リン酸アミド誘導体およびその製造方法ならびにそれを含有する医薬
US4539037A (en) * 1983-03-16 1985-09-03 Allied Corporation Urease inhibited urea based fertilizer compositions containing N-aryl-N-aliphatic phosphorotriamide compounds
US4530714A (en) * 1983-03-16 1985-07-23 Allied Corporation N-aliphatic and N,N-aliphatic phosphoric triamide urease inhibitors and urease inhibited urea based fertilizer compositions
US4517002A (en) * 1983-03-16 1985-05-14 Allied Corporation Phosphorodiamide urease inhibitors and urease inhibited urea based fertilizer compositions
US4540428A (en) * 1983-03-16 1985-09-10 Allied Corporation Phosphorotriamidate urease inhibitors and urease inhibited urea based fertilizer compositions
EP0119494A1 (en) * 1983-03-16 1984-09-26 Allied Corporation Urease inhibited urea based fertilizer compositions containing phosphorus compounds
US4518413A (en) * 1983-06-06 1985-05-21 Allied Corporation Poly-phosphorodiamide urease inhibitors and urease inhibited urea based fertilizer compositions
US4517003A (en) * 1983-06-08 1985-05-14 Allied Corporation N-acyl phosphoric triamide urease inhibitors and urease inhibited urea based fertilizer compositions
US4517007A (en) * 1983-06-09 1985-05-14 Allied Corporation Phosphoroamide urease inhibitors and urease inhibited urea based fertilizer compositions
US4528020A (en) * 1983-06-16 1985-07-09 Allied Corporation Urease inhibited urea based fertilizer compositions
US4624695A (en) * 1983-12-20 1986-11-25 Allied Corporation O-diaminophosphinyl derivatives of oximes as urease inhibitors
US4629491A (en) * 1983-12-20 1986-12-16 Allied Corporation Oxidized sulfur derivatives of diaminophosphinyl compounds as urease inhibitors and urease inhibited urea based fertilizer compositions
US4824783A (en) * 1983-12-20 1989-04-25 Enichem S.P.A. Oxidized sulfur derivatives of diaminophosphinyl compounds as urease inhibitors
US4668667A (en) * 1985-08-01 1987-05-26 Norwich Eaton Pharmaceuticals, Inc. Acylphosphorotriamides useful as lipid-altering agents
US4800194A (en) * 1985-08-01 1989-01-24 Norwich Eaton Pharmaceuticals, Inc. Acylphosphorotriamides useful as lipid-altering agents
US5840917A (en) * 1995-09-26 1998-11-24 Takeda Chemical Industries, Ltd. Phosphorylamides, their preparation and use
AU6422798A (en) * 1997-03-25 1998-10-20 Takeda Chemical Industries Ltd. Stabilized urease inhibitor
DE10118322A1 (de) * 2001-04-12 2002-10-17 Piesteritz Stickstoff Heterozyklisch-substituierte (Thio)Phosphorsäuretriamide, Verfahren zu ihrer Herstellung und deren Verwendung als Mittel zur Regulierung bzw.Hemmung der enzymatischen Harnstoff-Hydrolyse
WO2013182469A2 (en) 2012-06-08 2013-12-12 Basf Se Odour-control superabsorbent
DE102013012500A1 (de) 2013-07-26 2015-01-29 Skw Stickstoffwerke Piesteritz Gmbh Verwendung von Phosphorsäureamiden als Mittel zur Verbesserung der Trockenstresstoleranz

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3317637A (en) * 1961-06-30 1967-05-02 Dow Chemical Co N-haloacylphosphoric amides
US3321516A (en) * 1963-12-06 1967-05-23 Pennsalt Chemicals Corp Dialkylthiocarbamylphosphonic diamides
GB1448241A (en) * 1973-01-23 1976-09-02 Ici Ltd Thiophosphorus acid amides and their use as inhibitors of premature vulcanisation of rubber

Also Published As

Publication number Publication date
NL190781C (nl) 1994-08-16
FR2431505A1 (fr) 1980-02-15
JPS6254117B2 (it) 1987-11-13
NL190781B (nl) 1994-03-16
AU4676379A (en) 1980-01-24
FR2431505B1 (it) 1984-07-13
IE48326B1 (en) 1984-12-12
IE790790L (en) 1980-01-19
SE441831B (sv) 1985-11-11
NL7905138A (nl) 1980-01-22
ES482598A1 (es) 1980-07-01
DE2928831A1 (de) 1980-01-31
BE877737A (fr) 1980-01-16
GB2025974B (en) 1982-10-27
US4182881A (en) 1980-01-08
AU521741B2 (en) 1982-04-29
CA1125289A (en) 1982-06-08
GB2025974A (en) 1980-01-30
CH642084A5 (de) 1984-03-30
MX5375E (es) 1983-06-30
JPS5515461A (en) 1980-02-02
SE7905922L (sv) 1980-01-20
DE2928831C2 (de) 1986-10-09
IT1120421B (it) 1986-03-26

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Effective date: 19970530