ES455805A1 - Un procedimiento para preparar derivados de olecendomina. - Google Patents
Un procedimiento para preparar derivados de olecendomina.Info
- Publication number
- ES455805A1 ES455805A1 ES455805A ES455805A ES455805A1 ES 455805 A1 ES455805 A1 ES 455805A1 ES 455805 A ES455805 A ES 455805A ES 455805 A ES455805 A ES 455805A ES 455805 A1 ES455805 A1 ES 455805A1
- Authority
- ES
- Spain
- Prior art keywords
- replaced
- positions
- hydroxyl groups
- aforementioned
- olecendomin
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
- 150000001875 compounds Chemical class 0.000 abstract 2
- 125000002887 hydroxy group Chemical group [H]O* 0.000 abstract 2
- 235000019367 oleandomycin Nutrition 0.000 abstract 2
- RZPAKFUAFGMUPI-UHFFFAOYSA-N Oleandomycin Natural products O1C(C)C(O)C(OC)CC1OC1C(C)C(=O)OC(C)C(C)C(O)C(C)C(=O)C2(OC2)CC(C)C(OC2C(C(CC(C)O2)N(C)C)O)C1C RZPAKFUAFGMUPI-UHFFFAOYSA-N 0.000 abstract 1
- 239000004104 Oleandomycin Substances 0.000 abstract 1
- 125000002777 acetyl group Chemical group [H]C([H])([H])C(*)=O 0.000 abstract 1
- 125000000217 alkyl group Chemical group 0.000 abstract 1
- 239000003242 anti bacterial agent Substances 0.000 abstract 1
- 235000010633 broth Nutrition 0.000 abstract 1
- 125000001589 carboacyl group Chemical group 0.000 abstract 1
- 125000004432 carbon atom Chemical group C* 0.000 abstract 1
- 150000002148 esters Chemical class 0.000 abstract 1
- 230000004151 fermentation Effects 0.000 abstract 1
- 238000000855 fermentation Methods 0.000 abstract 1
- 125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 1
- 238000004519 manufacturing process Methods 0.000 abstract 1
- 238000012986 modification Methods 0.000 abstract 1
- 230000004048 modification Effects 0.000 abstract 1
- RZPAKFUAFGMUPI-KGIGTXTPSA-N oleandomycin Chemical compound O1[C@@H](C)[C@H](O)[C@@H](OC)C[C@@H]1O[C@@H]1[C@@H](C)C(=O)O[C@H](C)[C@H](C)[C@H](O)[C@@H](C)C(=O)[C@]2(OC2)C[C@H](C)[C@H](O[C@H]2[C@@H]([C@H](C[C@@H](C)O2)N(C)C)O)[C@H]1C RZPAKFUAFGMUPI-KGIGTXTPSA-N 0.000 abstract 1
- 229960002351 oleandomycin Drugs 0.000 abstract 1
- 125000001181 organosilyl group Chemical group [SiH3]* 0.000 abstract 1
- 125000004044 trifluoroacetyl group Chemical group FC(C(=O)*)(F)F 0.000 abstract 1
- 125000000026 trimethylsilyl group Chemical group [H]C([H])([H])[Si]([*])(C([H])([H])[H])C([H])([H])[H] 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
- C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
- C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
Landscapes
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Communicable Diseases (AREA)
- Medicinal Chemistry (AREA)
- Genetics & Genomics (AREA)
- Molecular Biology (AREA)
- Biochemistry (AREA)
- Engineering & Computer Science (AREA)
- Oncology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Biotechnology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Saccharide Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US66346776A | 1976-03-03 | 1976-03-03 | |
| US70346476A | 1976-07-08 | 1976-07-08 | |
| US05/709,703 US4069379A (en) | 1976-07-08 | 1976-07-29 | Semi-synthetic oleandomycins |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ES455805A1 true ES455805A1 (es) | 1978-04-01 |
Family
ID=27418084
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES455805A Expired ES455805A1 (es) | 1976-03-03 | 1977-02-10 | Un procedimiento para preparar derivados de olecendomina. |
Country Status (21)
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4166901A (en) * | 1978-01-03 | 1979-09-04 | Pfizer Inc. | 4"-Deoxy-4"-arylglyoxamido- and aroylthioformamido derivatives of oleandomycin and its esters |
| US4180654A (en) * | 1978-01-03 | 1979-12-25 | Pfizer Inc. | 4"-Deoxy-4"-acylamido derivatives of oleandomycin, erythromycin and erythromycin carbonate |
-
1976
- 1976-11-23 IE IE2578/76A patent/IE44509B1/en unknown
- 1976-12-02 DE DE2654627A patent/DE2654627C3/de not_active Expired
- 1976-12-02 DE DE2660089A patent/DE2660089C2/de not_active Expired
-
1977
- 1977-01-25 SE SE7700786A patent/SE436283B/xx unknown
- 1977-01-31 IL IL51361A patent/IL51361A/xx unknown
- 1977-02-01 AT AT62777A patent/AT347586B/de not_active IP Right Cessation
- 1977-02-02 NZ NZ183235A patent/NZ183235A/xx unknown
- 1977-02-02 PH PH19411A patent/PH13171A/en unknown
- 1977-02-04 PT PT66157A patent/PT66157B/pt unknown
- 1977-02-09 FR FR7703604A patent/FR2342989A1/fr active Granted
- 1977-02-09 CA CA271,457A patent/CA1069503A/en not_active Expired
- 1977-02-10 NL NLAANVRAGE7701401,A patent/NL170151C/xx not_active IP Right Cessation
- 1977-02-10 DK DK57177A patent/DK146778C/da not_active IP Right Cessation
- 1977-02-10 FI FI770440A patent/FI770440A7/fi not_active Application Discontinuation
- 1977-02-10 JP JP1403577A patent/JPS52106880A/ja active Granted
- 1977-02-10 ES ES455805A patent/ES455805A1/es not_active Expired
- 1977-02-11 AR AR266519A patent/AR212524A1/es active
- 1977-02-11 LU LU76764A patent/LU76764A1/xx unknown
- 1977-02-11 GB GB5755/77A patent/GB1567390A/en not_active Expired
- 1977-02-23 RO RO7789496A patent/RO72560A/ro unknown
- 1977-02-23 RO RO7797127A patent/RO76882A/ro unknown
- 1977-02-25 BG BG035526A patent/BG27913A3/xx unknown
- 1977-02-25 BG BG036454A patent/BG27914A4/xx unknown
- 1977-02-28 DD DD7700197598A patent/DD129789A5/xx unknown
-
1980
- 1980-07-01 SE SE8004873A patent/SE436284B/sv unknown
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