ES451480A1 - Un procedimiento para la preparacion de nuevos derivados de piridazinona. - Google Patents
Un procedimiento para la preparacion de nuevos derivados de piridazinona.Info
- Publication number
- ES451480A1 ES451480A1 ES451480A ES451480A ES451480A1 ES 451480 A1 ES451480 A1 ES 451480A1 ES 451480 A ES451480 A ES 451480A ES 451480 A ES451480 A ES 451480A ES 451480 A1 ES451480 A1 ES 451480A1
- Authority
- ES
- Spain
- Prior art keywords
- group
- formula
- halogen atom
- carbon atoms
- halogen
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
- AAILEWXSEQLMNI-UHFFFAOYSA-N 1h-pyridazin-6-one Chemical class OC1=CC=CN=N1 AAILEWXSEQLMNI-UHFFFAOYSA-N 0.000 title abstract 2
- -1 6-(substituted phenyl)-pyridazinones Chemical class 0.000 title abstract 2
- 230000000855 fungicidal effect Effects 0.000 title abstract 2
- 239000000203 mixture Substances 0.000 title abstract 2
- 125000005843 halogen group Chemical group 0.000 abstract 8
- 125000004432 carbon atom Chemical group C* 0.000 abstract 5
- 125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 5
- 125000000217 alkyl group Chemical group 0.000 abstract 4
- 125000002887 hydroxy group Chemical group [H]O* 0.000 abstract 4
- 125000003545 alkoxy group Chemical group 0.000 abstract 3
- 150000001875 compounds Chemical class 0.000 abstract 3
- KMQLIDDEQAJAGJ-UHFFFAOYSA-N 4-oxo-4-phenylbutyric acid Chemical class OC(=O)CCC(=O)C1=CC=CC=C1 KMQLIDDEQAJAGJ-UHFFFAOYSA-N 0.000 abstract 2
- OAKJQQAXSVQMHS-UHFFFAOYSA-N Hydrazine Chemical compound NN OAKJQQAXSVQMHS-UHFFFAOYSA-N 0.000 abstract 2
- 125000003302 alkenyloxy group Chemical group 0.000 abstract 2
- 125000005133 alkynyloxy group Chemical group 0.000 abstract 2
- 125000003277 amino group Chemical group 0.000 abstract 2
- 229910052736 halogen Inorganic materials 0.000 abstract 2
- 150000002367 halogens Chemical class 0.000 abstract 2
- 238000000034 method Methods 0.000 abstract 2
- 150000003839 salts Chemical class 0.000 abstract 2
- FALRKNHUBBKYCC-UHFFFAOYSA-N 2-(chloromethyl)pyridine-3-carbonitrile Chemical compound ClCC1=NC=CC=C1C#N FALRKNHUBBKYCC-UHFFFAOYSA-N 0.000 abstract 1
- UFHFLCQGNIYNRP-UHFFFAOYSA-N Hydrogen Chemical compound [H][H] UFHFLCQGNIYNRP-UHFFFAOYSA-N 0.000 abstract 1
- 239000002841 Lewis acid Substances 0.000 abstract 1
- 239000002253 acid Substances 0.000 abstract 1
- 239000013543 active substance Substances 0.000 abstract 1
- 125000005907 alkyl ester group Chemical group 0.000 abstract 1
- 230000002140 halogenating effect Effects 0.000 abstract 1
- 229910052739 hydrogen Inorganic materials 0.000 abstract 1
- 239000001257 hydrogen Substances 0.000 abstract 1
- 150000007517 lewis acids Chemical class 0.000 abstract 1
- 238000004519 manufacturing process Methods 0.000 abstract 1
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 abstract 1
- 125000006239 protecting group Chemical group 0.000 abstract 1
- 125000001424 substituent group Chemical group 0.000 abstract 1
- 229940014800 succinic anhydride Drugs 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D237/00—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings
- C07D237/02—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings
- C07D237/04—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings having less than three double bonds between ring members or between ring members and non-ring members
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C59/00—Compounds having carboxyl groups bound to acyclic carbon atoms and containing any of the groups OH, O—metal, —CHO, keto, ether, groups, groups, or groups
- C07C59/40—Unsaturated compounds
- C07C59/76—Unsaturated compounds containing keto groups
- C07C59/88—Unsaturated compounds containing keto groups containing halogen
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C59/00—Compounds having carboxyl groups bound to acyclic carbon atoms and containing any of the groups OH, O—metal, —CHO, keto, ether, groups, groups, or groups
- C07C59/40—Unsaturated compounds
- C07C59/76—Unsaturated compounds containing keto groups
- C07C59/90—Unsaturated compounds containing keto groups containing singly bound oxygen-containing groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D237/00—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings
- C07D237/02—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings
- C07D237/06—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members
- C07D237/10—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D237/14—Oxygen atoms
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP11033175A JPS5234928A (en) | 1975-09-11 | 1975-09-11 | Fungicides for agriculture and gardening use |
| JP51036453A JPS584681B2 (ja) | 1976-04-01 | 1976-04-01 | 農園芸用殺菌剤 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ES451480A1 true ES451480A1 (es) | 1977-12-01 |
Family
ID=26375516
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES451480A Expired ES451480A1 (es) | 1975-09-11 | 1976-09-11 | Un procedimiento para la preparacion de nuevos derivados de piridazinona. |
| ES463200A Expired ES463200A1 (es) | 1975-09-11 | 1977-10-13 | Un procedimiento para la preparacion de nuevos derivados de piridazinona. |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES463200A Expired ES463200A1 (es) | 1975-09-11 | 1977-10-13 | Un procedimiento para la preparacion de nuevos derivados de piridazinona. |
Country Status (12)
| Country | Link |
|---|---|
| US (1) | US4052395A (cg-RX-API-DMAC10.html) |
| BR (1) | BR7605990A (cg-RX-API-DMAC10.html) |
| CA (1) | CA1082105A (cg-RX-API-DMAC10.html) |
| CH (1) | CH621683A5 (cg-RX-API-DMAC10.html) |
| DE (1) | DE2640806A1 (cg-RX-API-DMAC10.html) |
| ES (2) | ES451480A1 (cg-RX-API-DMAC10.html) |
| FR (2) | FR2323327A1 (cg-RX-API-DMAC10.html) |
| GB (1) | GB1533010A (cg-RX-API-DMAC10.html) |
| IT (1) | IT1071604B (cg-RX-API-DMAC10.html) |
| MY (1) | MY8100058A (cg-RX-API-DMAC10.html) |
| NL (1) | NL7610155A (cg-RX-API-DMAC10.html) |
| PH (1) | PH14059A (cg-RX-API-DMAC10.html) |
Families Citing this family (44)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4189578A (en) * | 1977-10-19 | 1980-02-19 | Smithkline Corporation | 3-(o-Hydroxyphenyl)-5-formylhydrazino-Δ2 -pyrazolines |
| US4279908A (en) * | 1979-04-19 | 1981-07-21 | Sankyo Company Limited | Pyridazine derivatives and their use as agricultural fungicides |
| JPS5826802A (ja) * | 1981-08-10 | 1983-02-17 | Sankyo Co Ltd | 農園芸用殺菌剤 |
| JPS58162577A (ja) * | 1982-03-19 | 1983-09-27 | Sankyo Co Ltd | ６−フエニルピリダジノン化合物の製造法 |
| US4411753A (en) | 1982-04-08 | 1983-10-25 | Eli Lilly And Company | Synthesis of 6-t-alkyl-3-pyridazinones |
| JPS6061570A (ja) * | 1983-09-16 | 1985-04-09 | Sankyo Co Ltd | ピリダジノン誘導体及び農業用殺菌剤 |
| US4731385A (en) * | 1985-10-26 | 1988-03-15 | Nihon Tokushu Noyaku Seizo K.K. | Insecticidal and fungicidal composition for agricultural and horticultural use |
| ES2131506T3 (es) * | 1990-09-21 | 1999-08-01 | Rohm & Haas | Dihidropiridacinonas y piridacinonas como fungicidas. |
| CN1038249C (zh) * | 1991-08-28 | 1998-05-06 | 罗姆和哈斯公司 | 含有二氢哒嗪酮及其相关化合物的杀菌组合物 |
| IL115889A0 (en) * | 1994-11-14 | 1996-01-31 | Rohm & Haas | Pyridazinones and their use as fungicides |
| US5635494A (en) * | 1995-04-21 | 1997-06-03 | Rohm And Haas Company | Dihydropyridazinones and pyridazinones and their use as fungicides and insecticides |
| US6121251A (en) * | 1996-10-11 | 2000-09-19 | Rohm And Haas Company | Dihydropyridazinones and pyridazinones and their use as fungicides and insecticides |
| UA90360C2 (ru) * | 2005-12-07 | 2010-04-26 | Сумитомо Кемикал Компани, Лимитед | Пиридазинова соединение, его применение, агент и способ контролирования заболевания растений, а также промежуточное соединение |
| WO2008071714A1 (en) | 2006-12-15 | 2008-06-19 | Rohm And Haas Company | Mixtures comprising 1-methylcyclopropene |
| BRPI0809498A2 (pt) * | 2007-04-02 | 2014-09-23 | Inst Oneworld Health | Compostos inibidores de cftr e seus usos |
| KR20100015796A (ko) | 2007-04-23 | 2010-02-12 | 바스프 에스이 | 화학 작용제와 트랜스제닉 변형의 조합에 의한 식물 생산성의 증진 |
| ES2381320T3 (es) | 2007-09-26 | 2012-05-25 | Basf Se | Composiciones fungicidas ternarias que comprenden boscalida y clorotalonil |
| EP2278879B1 (en) * | 2008-04-21 | 2016-06-15 | PATH Drug Solutions | Compounds, compositions and methods comprising oxadiazole derivatives |
| US20090264433A1 (en) * | 2008-04-21 | 2009-10-22 | Institute For Oneworld Health | Compounds, Compositions and Methods Comprising Triazine Derivatives |
| US8236838B2 (en) * | 2008-04-21 | 2012-08-07 | Institute For Oneworld Health | Compounds, compositions and methods comprising isoxazole derivatives |
| US20090270398A1 (en) * | 2008-04-21 | 2009-10-29 | Institute For Oneworld Health | Compounds, Compositions and Methods Comprising Pyridazine Derivatives |
| JP2012503005A (ja) * | 2008-09-19 | 2012-02-02 | インスティテュート フォア ワンワールド ヘルス | イミダゾール誘導体およびトリアゾール誘導体を含む、化合物、組成物ならびに方法。 |
| US8511216B2 (en) * | 2009-03-30 | 2013-08-20 | Kanzaki Kokyukoki Mfg. Co., Ltd. | Hydraulic actuator unit |
| US8343976B2 (en) * | 2009-04-20 | 2013-01-01 | Institute For Oneworld Health | Compounds, compositions and methods comprising pyrazole derivatives |
| US20100330884A1 (en) * | 2009-06-29 | 2010-12-30 | Ferro Corporation | Diatomaceous Earth-Containing Slurry Composition And Method For Polishing Organic Polymer-Based Ophthalmic Substrates Using The Same |
| WO2011026796A1 (en) | 2009-09-01 | 2011-03-10 | Basf Se | Synergistic fungicidal mixtures comprising lactylates and method for combating phytopathogenic fungi |
| US20130267476A1 (en) | 2010-12-20 | 2013-10-10 | Basf Se | Pesticidal Active Mixtures Comprising Pyrazole Compounds |
| EP2481284A3 (en) | 2011-01-27 | 2012-10-17 | Basf Se | Pesticidal mixtures |
| ES2660555T3 (es) | 2011-03-23 | 2018-03-22 | Basf Se | Composiciones que contienen compuestos iónicos, poliméricos que comprenden grupos imidazolio |
| BR112014004568A2 (pt) | 2011-09-02 | 2017-04-04 | Basf Se | misturas agrícolas, método para proteger plantas de ataque, método para controlar insetos, método para a proteção de material de propagação de planta, semente, método para controlar fungos nocivos fitopagênicos, uso de uma mistura e composição agrícola |
| PT3300602T (pt) | 2012-06-20 | 2020-06-17 | Basf Se | Misturas pesticidas que compreendem um composto de pirazol |
| US20150257383A1 (en) | 2012-10-12 | 2015-09-17 | Basf Se | Method for combating phytopathogenic harmful microbes on cultivated plants or plant propagation material |
| CN105050406B (zh) | 2012-12-20 | 2017-09-15 | 巴斯夫农业公司 | 包含三唑化合物的组合物 |
| US9890127B2 (en) | 2013-03-11 | 2018-02-13 | The Broad Institute, Inc. | Compounds and compositions for the treatment of cancer |
| EP2783569A1 (en) | 2013-03-28 | 2014-10-01 | Basf Se | Compositions comprising a triazole compound |
| EP2835052A1 (en) | 2013-08-07 | 2015-02-11 | Basf Se | Fungicidal mixtures comprising pyrimidine fungicides |
| WO2015036059A1 (en) | 2013-09-16 | 2015-03-19 | Basf Se | Fungicidal pyrimidine compounds |
| CN105722833A (zh) | 2013-09-16 | 2016-06-29 | 巴斯夫欧洲公司 | 杀真菌的嘧啶化合物 |
| EP2979549A1 (en) | 2014-07-31 | 2016-02-03 | Basf Se | Method for improving the health of a plant |
| RU2707051C2 (ru) | 2014-10-24 | 2019-11-21 | Басф Се | Неамфолитные, кватернизируемые и водорастворимые полимеры для модифицирования поверхностного заряда твердых частиц |
| US11207320B2 (en) | 2015-08-13 | 2021-12-28 | The Broad Institute, Inc. | Compositions and methods for cancer expressing PDE3A or SLFN12 |
| EP3661917B1 (en) | 2017-08-04 | 2022-05-11 | Bayer Aktiengesellschaft | 6-((3-trifluoromethyl)phenyl)-4,5-dihydropyridazin-3(2h)-one derivatives as pde3a and pde3b inhibitors for treating cancer |
| JOP20200024A1 (ar) | 2017-08-04 | 2020-02-02 | Bayer Ag | مركبات ثنائي هيدروكساديازينون |
| TWI750573B (zh) | 2019-02-01 | 2021-12-21 | 德商拜耳廠股份有限公司 | 1,2,4-三-3(2h)-酮化合物 |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE1670043C3 (de) * | 1966-01-07 | 1975-05-22 | Basf Ag, 6700 Ludwigshafen | Verfahren zur Herstellung von 3-(Aminophenyl)-pyridazon-(6)-derivaten |
| GB1292443A (en) * | 1968-11-01 | 1972-10-11 | Ct D Etudes Experimentales Et | New pyridazine derivatives and process for their preparation |
| IL37788A0 (en) * | 1970-10-09 | 1971-12-29 | American Cyanamid Co | New pyridazinone compounds,their preparation and pharmaceutical compositions containing them |
| US3975388A (en) * | 1971-02-22 | 1976-08-17 | Bdh Pharmaceuticals Limited | Pyridazinones |
| GB1383906A (en) * | 1971-02-22 | 1974-02-12 | Bdh Pharmaceuticals Ltd | Pyridazinones |
| DE2214059A1 (de) * | 1972-03-23 | 1973-09-27 | Bayer Ag | Halogenphenyl-pyridazino-thionophosphor (phosphon)-saeureester, verfahren zu ihrer herstellung sowie ihre verwendung als insektizide |
| US3824271A (en) * | 1972-07-20 | 1974-07-16 | American Cyanamid Co | 3-alkyl-3-(benzoyl)propionitriles |
-
1976
- 1976-08-30 US US05/718,589 patent/US4052395A/en not_active Expired - Lifetime
- 1976-09-09 PH PH18905A patent/PH14059A/en unknown
- 1976-09-10 CH CH1157376A patent/CH621683A5/de not_active IP Right Cessation
- 1976-09-10 BR BR7605990A patent/BR7605990A/pt unknown
- 1976-09-10 GB GB37597/76A patent/GB1533010A/en not_active Expired
- 1976-09-10 DE DE19762640806 patent/DE2640806A1/de active Granted
- 1976-09-11 ES ES451480A patent/ES451480A1/es not_active Expired
- 1976-09-13 NL NL7610155A patent/NL7610155A/xx not_active Application Discontinuation
- 1976-09-13 IT IT69226/76A patent/IT1071604B/it active
- 1976-09-13 FR FR7627492A patent/FR2323327A1/fr active Granted
- 1976-09-13 CA CA261,039A patent/CA1082105A/en not_active Expired
-
1977
- 1977-10-13 ES ES463200A patent/ES463200A1/es not_active Expired
-
1980
- 1980-07-10 FR FR8015402A patent/FR2464255A1/fr active Granted
-
1981
- 1981-12-30 MY MY58/81A patent/MY8100058A/xx unknown
Also Published As
| Publication number | Publication date |
|---|---|
| DE2640806C2 (cg-RX-API-DMAC10.html) | 1989-09-14 |
| NL7610155A (nl) | 1977-03-15 |
| CH621683A5 (cg-RX-API-DMAC10.html) | 1981-02-27 |
| GB1533010A (en) | 1978-11-22 |
| MY8100058A (en) | 1981-12-31 |
| DE2640806A1 (de) | 1977-03-24 |
| IT1071604B (it) | 1985-04-10 |
| FR2464255B1 (cg-RX-API-DMAC10.html) | 1984-04-06 |
| BR7605990A (pt) | 1977-08-23 |
| CA1082105A (en) | 1980-07-22 |
| US4052395A (en) | 1977-10-04 |
| ES463200A1 (es) | 1978-11-16 |
| PH14059A (en) | 1980-12-29 |
| FR2464255A1 (fr) | 1981-03-06 |
| FR2323327A1 (fr) | 1977-04-08 |
| FR2323327B1 (cg-RX-API-DMAC10.html) | 1981-09-18 |
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