ES2915698T3 - Formulaciones farmacéuticas que comprenden derivados de nitrocatecol y métodos para preparar las mismas - Google Patents
Formulaciones farmacéuticas que comprenden derivados de nitrocatecol y métodos para preparar las mismas Download PDFInfo
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- ES2915698T3 ES2915698T3 ES10714386T ES10714386T ES2915698T3 ES 2915698 T3 ES2915698 T3 ES 2915698T3 ES 10714386 T ES10714386 T ES 10714386T ES 10714386 T ES10714386 T ES 10714386T ES 2915698 T3 ES2915698 T3 ES 2915698T3
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Landscapes
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- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US16579409P | 2009-04-01 | 2009-04-01 | |
| PCT/PT2010/000015 WO2010114405A2 (en) | 2009-04-01 | 2010-03-31 | Pharmaceutical formulations comprising nitrocatechol derivatives and methods of making the same |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ES2915698T3 true ES2915698T3 (es) | 2022-06-24 |
Family
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES10714386T Active ES2915698T3 (es) | 2009-04-01 | 2010-03-31 | Formulaciones farmacéuticas que comprenden derivados de nitrocatecol y métodos para preparar las mismas |
Country Status (15)
| Country | Link |
|---|---|
| US (3) | US20100256194A1 (enExample) |
| EP (1) | EP2413913B1 (enExample) |
| JP (2) | JP5864410B2 (enExample) |
| KR (1) | KR101824257B1 (enExample) |
| CN (2) | CN102438595B (enExample) |
| AU (1) | AU2010231962B2 (enExample) |
| BR (1) | BRPI1016132B8 (enExample) |
| CA (1) | CA2757418C (enExample) |
| DK (1) | DK2413913T3 (enExample) |
| ES (1) | ES2915698T3 (enExample) |
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| US8168793B2 (en) | 2005-07-26 | 2012-05-01 | Portela & Ca., S.A. | Nitrocatechol derivatives as COMT inhibitors |
| EP1845097A1 (en) | 2006-04-10 | 2007-10-17 | Portela & Ca., S.A. | Oxadiazole derivatives as COMT inhibitors |
| PL2481410T3 (pl) | 2007-01-31 | 2017-03-31 | Bial - Portela & Ca., S.A. | Pochodne nitrokatecholu jako inhibitory COMT podawane w określonym schemacie dawkowania |
| CL2009000628A1 (es) | 2008-03-17 | 2010-04-09 | Bial Portela & Companhia S A | Forma cristalina de 5-[3-(2,5-dicloro-4,6-dimetil-1-oxi-piridin-3-il)-[1,2,4]oxadiazol-5-il]-3-nitrobenceno-1,2-diol, composicion farmaceutica que la comprende, proceso para obtenerla y su uso para tratar trastornos del animo, enfermedad de parkinson y trastornos parkinsonianos, alteraciones gastrointestinales, entre otros. |
| US9132094B2 (en) | 2009-04-01 | 2015-09-15 | Bial—Portela & Ca, S.A. | Pharmaceutical formulations comprising nitrocatechol derivatives and methods of making thereof |
| US20140045900A1 (en) * | 2011-02-11 | 2014-02-13 | Bial-Portela & Ca, S.A. | Administration regime for nitrocatechols |
| PT2791134T (pt) | 2011-12-13 | 2019-12-18 | BIAL PORTELA & Cª S A | Composto químico útil como intermediário para a preparação de um inibidor de catecol-o-metiltransferase |
| NO2699580T3 (enExample) | 2014-01-24 | 2018-02-24 | ||
| RU2017120184A (ru) | 2014-11-28 | 2018-12-28 | БИАЛ - ПОРТЕЛА ЭНД Ка, С.А. | Лекарства для замедления течения болезни паркинсона |
| JP2021506762A (ja) * | 2017-12-18 | 2021-02-22 | ユニケム ラボラトリーズ リミテッド | オピカポンとその中間体の製造方法 |
| HRP20250115T1 (hr) | 2018-03-01 | 2025-05-23 | Astrazeneca Ab | Farmaceutski pripravci koji sadrže (2s)-{(1s)-1-cijano-2-[4-(3-metil-2-okso-2,3-dihidro-1,3-benzoksazol-5-il)fenil]etil} -1,4-oksazepan-2-karboksamid |
| CA3106269A1 (en) | 2018-07-17 | 2020-01-23 | Insmed Incorporated | Certain (2s)-n-[(1s)-1-cyano-2-phenylethyl]-1,4-oxazepane-2-carboxamides for treating lupus nephritis |
| EP3860602A1 (en) | 2018-10-05 | 2021-08-11 | Neurocrine Biosciences, Inc. | Methods for the administration of comt inhibitors |
| US12097193B2 (en) | 2018-10-05 | 2024-09-24 | Bial—Portela & Ca, S.A. | Methods for the administration of COMT inhibitors |
| EP4117637A1 (en) | 2020-03-13 | 2023-01-18 | Bial-Portela & CA, S.A. | Micronised opicapone |
| GB202011709D0 (en) | 2020-07-28 | 2020-09-09 | Bial Portela & Ca Sa | Solid dispersion of opicapone |
| GB202016425D0 (en) | 2020-10-16 | 2020-12-02 | Bial Portela & Ca Sa | Treatment regimens for parkinson's disease |
| KR20230118933A (ko) | 2020-12-17 | 2023-08-14 | 바이알 - 포르텔라 앤드 씨에이 에스에이 | 초기 특발성 파킨슨병에 대한 치료 요법 |
| US20240300930A1 (en) * | 2021-02-26 | 2024-09-12 | Msn Laboratories Private Limited, R&D Center | Novel process for the preparation of 2,5-dichloro-3-(5-(3,4-dihydroxy-5-nitrophenyl)-1,2,4-oxadiazol-3-yl)-4,6-dimethylpyridine-1-oxide |
| GB202212082D0 (en) | 2022-08-18 | 2022-10-05 | Bial Portela & Ca Sa | Treatment regimens for parkinson's disease |
| EP4646265A1 (en) | 2023-01-06 | 2025-11-12 | Insmed Incorporated | Novel, reversible dpp1 inhibitors and uses thereof |
| AU2023449890A1 (en) | 2023-05-25 | 2025-11-27 | Bial-Portela & Ca., S.A. | Treatment regimens for early idiopathic parkinson's disease |
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| US8168793B2 (en) * | 2005-07-26 | 2012-05-01 | Portela & Ca., S.A. | Nitrocatechol derivatives as COMT inhibitors |
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| EP1845097A1 (en) * | 2006-04-10 | 2007-10-17 | Portela & Ca., S.A. | Oxadiazole derivatives as COMT inhibitors |
| JP2008162955A (ja) * | 2006-12-28 | 2008-07-17 | Chugai Pharmaceut Co Ltd | バリン含有高密度顆粒剤 |
| PL2481410T3 (pl) * | 2007-01-31 | 2017-03-31 | Bial - Portela & Ca., S.A. | Pochodne nitrokatecholu jako inhibitory COMT podawane w określonym schemacie dawkowania |
| PE20081891A1 (es) * | 2007-03-22 | 2008-12-27 | Opko Health Inc | Formulaciones de comprimidos que contienen sales de 8-[{1-(3,5-bis-(trifluorometil)fenil)-etoxi}-metil]-8-fenil-1,7-diaza-spiro[4.5]decan-2-ona y comprimidos elaborados a partir de estas |
| CL2009000628A1 (es) * | 2008-03-17 | 2010-04-09 | Bial Portela & Companhia S A | Forma cristalina de 5-[3-(2,5-dicloro-4,6-dimetil-1-oxi-piridin-3-il)-[1,2,4]oxadiazol-5-il]-3-nitrobenceno-1,2-diol, composicion farmaceutica que la comprende, proceso para obtenerla y su uso para tratar trastornos del animo, enfermedad de parkinson y trastornos parkinsonianos, alteraciones gastrointestinales, entre otros. |
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2010
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2015
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2018
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2020
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| PL2413913T3 (pl) | 2022-09-26 |
| BRPI1016132B8 (pt) | 2021-05-25 |
| US20210315824A1 (en) | 2021-10-14 |
| WO2010114405A2 (en) | 2010-10-07 |
| CA2757418A1 (en) | 2010-10-07 |
| EP2413913A2 (en) | 2012-02-08 |
| JP2012522764A (ja) | 2012-09-27 |
| MX361618B (es) | 2018-12-13 |
| PT2413913T (pt) | 2022-06-09 |
| RU2550133C2 (ru) | 2015-05-10 |
| CN105816456A (zh) | 2016-08-03 |
| JP6336420B2 (ja) | 2018-06-06 |
| AU2010231962B2 (en) | 2015-05-21 |
| EP2413913B1 (en) | 2022-05-18 |
| MX2011010311A (es) | 2012-03-07 |
| KR20120008040A (ko) | 2012-01-25 |
| US20190008774A1 (en) | 2019-01-10 |
| CN102438595A (zh) | 2012-05-02 |
| AU2010231962A1 (en) | 2011-11-17 |
| KR101824257B1 (ko) | 2018-01-31 |
| BRPI1016132B1 (pt) | 2020-11-24 |
| CA2757418C (en) | 2021-06-15 |
| BRPI1016132A2 (pt) | 2016-04-19 |
| WO2010114405A3 (en) | 2011-01-06 |
| US20100256194A1 (en) | 2010-10-07 |
| CN102438595B (zh) | 2016-04-27 |
| DK2413913T3 (da) | 2022-06-13 |
| RU2011143619A (ru) | 2013-05-10 |
| JP5864410B2 (ja) | 2016-02-17 |
| JP2016020369A (ja) | 2016-02-04 |
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