ES2842208T3 - Composiciones farmacéuticas de donepezilo que tienen perfil de disolución in vitro o parámetros farmacocinéticos específicos - Google Patents
Composiciones farmacéuticas de donepezilo que tienen perfil de disolución in vitro o parámetros farmacocinéticos específicos Download PDFInfo
- Publication number
- ES2842208T3 ES2842208T3 ES14710647T ES14710647T ES2842208T3 ES 2842208 T3 ES2842208 T3 ES 2842208T3 ES 14710647 T ES14710647 T ES 14710647T ES 14710647 T ES14710647 T ES 14710647T ES 2842208 T3 ES2842208 T3 ES 2842208T3
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- donepezil
- release control
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- release
- sleep
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Classifications
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- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
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- A61K9/167—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction with an outer layer or coating comprising drug; with chemically bound drugs or non-active substances on their surface
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- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
- A61K9/5073—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings
- A61K9/5078—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings with drug-free core
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Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- General Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
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- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
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- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Biophysics (AREA)
- Molecular Biology (AREA)
- Hospice & Palliative Care (AREA)
- Anesthesiology (AREA)
- Psychiatry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IN991KO2012 | 2013-02-28 | ||
| PCT/IB2014/059302 WO2014132218A1 (en) | 2013-02-28 | 2014-02-27 | Pharmaceutical compositions of donepezil having specific in vitro dissolution profile or pharmacokinetics parameters |
Publications (1)
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| ES2842208T3 true ES2842208T3 (es) | 2021-07-13 |
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| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES14710647T Active ES2842208T3 (es) | 2013-02-28 | 2014-02-27 | Composiciones farmacéuticas de donepezilo que tienen perfil de disolución in vitro o parámetros farmacocinéticos específicos |
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| Country | Link |
|---|---|
| US (1) | US20160015698A1 (enExample) |
| EP (1) | EP2961393B1 (enExample) |
| JP (1) | JP6429808B2 (enExample) |
| KR (1) | KR102241113B1 (enExample) |
| CN (1) | CN105163723A (enExample) |
| BR (1) | BR112015020771A2 (enExample) |
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| WO (1) | WO2014132218A1 (enExample) |
| ZA (1) | ZA201506665B (enExample) |
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| EP1133230A4 (en) * | 1998-11-23 | 2004-05-26 | Bonnie M Davis | DOSAGE FORMULAS FOR ACETYLCHOLINESTERASE INHIBITORS |
| EP1368000A4 (en) * | 2001-03-13 | 2004-12-01 | Penwest Pharmaceuticals Co | CHRONOTHERAPEUTIC PHARMACEUTICAL FORMS CONTAINING A GLUCOCORTICOSTEROID |
| AR040680A1 (es) * | 2002-07-25 | 2005-04-13 | Pharmacia Corp | Composicion de tabletas de liberacion sostenida |
| US20050232990A1 (en) | 2003-12-31 | 2005-10-20 | Garth Boehm | Donepezil formulations |
| US20060280789A1 (en) | 2004-12-27 | 2006-12-14 | Eisai Research Institute | Sustained release formulations |
| US20090208579A1 (en) | 2004-12-27 | 2009-08-20 | Eisai R & D Management Co., Ltd. | Matrix Type Sustained-Release Preparation Containing Basic Drug or Salt Thereof, and Method for Manufacturing the Same |
| CN101090738A (zh) * | 2004-12-27 | 2007-12-19 | 卫材R&D管理有限公司 | 含有碱性药物或其盐的基质型缓释制剂及其制备方法 |
| US20060159753A1 (en) | 2004-12-27 | 2006-07-20 | Eisai Co. Ltd. | Matrix type sustained-release preparation containing basic drug or salt thereof |
| US20070129402A1 (en) | 2004-12-27 | 2007-06-07 | Eisai Research Institute | Sustained release formulations |
| KR100866720B1 (ko) | 2004-12-27 | 2008-11-05 | 에자이 알앤드디 매니지먼트 가부시키가이샤 | 항치매 약물의 안정화 방법 |
| NZ556630A (en) * | 2005-01-27 | 2010-12-24 | Alembic Ltd | Extended release formulation of levetiracetam including a hydrophilic rate controlling polymer |
| BRPI0607017B8 (pt) * | 2005-04-06 | 2021-05-25 | Adamas Pharmaceuticals Inc | composição farmacêutica compreendendo memantina e donezepil, e seu uso para o tratamento de condições relacionadas ao snc |
| US20130059003A1 (en) | 2009-12-04 | 2013-03-07 | Dr. Reddy's Laboratories, Inc. | Sustained release donepezil formulations |
| US20110218216A1 (en) | 2010-01-29 | 2011-09-08 | Kumaravel Vivek | Extended release pharmaceutical composition of donepezil |
| EP2366378A1 (en) * | 2010-03-01 | 2011-09-21 | Dexcel Pharma Technologies Ltd. | Sustained-release donepezil formulations |
| GB201003734D0 (en) * | 2010-03-05 | 2010-04-21 | Univ Strathclyde | Delayed prolonged drug delivery |
| CN102309465B (zh) * | 2010-06-30 | 2015-04-22 | 天津药物研究院 | 含盐酸多奈哌齐活性成分的缓释片及其制备方法和用途 |
| WO2012035409A1 (en) * | 2010-09-14 | 2012-03-22 | Rubicon Research Private Limited | Sustained release compositions of anti-alzheimer's agents |
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2014
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- 2014-02-27 WO PCT/IB2014/059302 patent/WO2014132218A1/en not_active Ceased
- 2014-02-27 EP EP14710647.0A patent/EP2961393B1/en not_active Not-in-force
- 2014-02-27 RU RU2015140567A patent/RU2015140567A/ru not_active Application Discontinuation
- 2014-02-27 JP JP2015559595A patent/JP6429808B2/ja not_active Expired - Fee Related
- 2014-02-27 BR BR112015020771A patent/BR112015020771A2/pt not_active Application Discontinuation
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- 2014-02-27 KR KR1020157026728A patent/KR102241113B1/ko not_active Expired - Fee Related
- 2014-02-27 MX MX2015011099A patent/MX378413B/es unknown
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2015
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Also Published As
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| RU2015140567A (ru) | 2017-03-31 |
| KR102241113B1 (ko) | 2021-04-15 |
| WO2014132218A1 (en) | 2014-09-04 |
| KR20150123302A (ko) | 2015-11-03 |
| MX2015011099A (es) | 2016-04-06 |
| CN105163723A (zh) | 2015-12-16 |
| MX378413B (es) | 2025-03-10 |
| JP6429808B2 (ja) | 2018-11-28 |
| EP2961393A1 (en) | 2016-01-06 |
| BR112015020771A2 (pt) | 2017-07-18 |
| EP2961393B1 (en) | 2020-10-28 |
| JP2016513133A (ja) | 2016-05-12 |
| US20160015698A1 (en) | 2016-01-21 |
| ZA201506665B (en) | 2017-02-22 |
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