CN105163723A - 具有特定体外溶解曲线或药动学参数的多奈哌齐的药物组合物 - Google Patents
具有特定体外溶解曲线或药动学参数的多奈哌齐的药物组合物 Download PDFInfo
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- CN105163723A CN105163723A CN201480024046.5A CN201480024046A CN105163723A CN 105163723 A CN105163723 A CN 105163723A CN 201480024046 A CN201480024046 A CN 201480024046A CN 105163723 A CN105163723 A CN 105163723A
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Classifications
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- A61K9/167—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction with an outer layer or coating comprising drug; with chemically bound drugs or non-active substances on their surface
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- A61K9/5073—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings
- A61K9/5078—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings with drug-free core
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- A—HUMAN NECESSITIES
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Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
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- Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
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- Chemical Kinetics & Catalysis (AREA)
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- Neurosurgery (AREA)
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- Psychiatry (AREA)
- Hospice & Palliative Care (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
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| IN991KO2012 | 2013-02-28 | ||
| IN991/KOL/2012 | 2013-02-28 | ||
| PCT/IB2014/059302 WO2014132218A1 (en) | 2013-02-28 | 2014-02-27 | Pharmaceutical compositions of donepezil having specific in vitro dissolution profile or pharmacokinetics parameters |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CN105163723A true CN105163723A (zh) | 2015-12-16 |
Family
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| Application Number | Title | Priority Date | Filing Date |
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| US (1) | US20160015698A1 (enExample) |
| EP (1) | EP2961393B1 (enExample) |
| JP (1) | JP6429808B2 (enExample) |
| KR (1) | KR102241113B1 (enExample) |
| CN (1) | CN105163723A (enExample) |
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| KR102142026B1 (ko) * | 2017-05-31 | 2020-08-06 | 주식회사 대웅제약 | 방출제어가 용이한 서방성 약물 미립자의 제조방법 |
Citations (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN101090738A (zh) * | 2004-12-27 | 2007-12-19 | 卫材R&D管理有限公司 | 含有碱性药物或其盐的基质型缓释制剂及其制备方法 |
| US20110237623A1 (en) * | 2010-03-01 | 2011-09-29 | Adel Penhasi | Sustained-release donepezil formulation |
| CN102309465A (zh) * | 2010-06-30 | 2012-01-11 | 天津药物研究院 | 含盐酸多奈哌齐活性成分的缓释片及其制备方法和用途 |
Family Cites Families (15)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA2351347A1 (en) * | 1998-11-23 | 2000-06-02 | Bonnie Davis | Dosage formulations for acetylcholinesterase inhibitors |
| US20030190360A1 (en) * | 2001-03-13 | 2003-10-09 | Baichwal Anand R. | Chronotherapeutic dosage forms containing glucocorticosteroid and methods of treatment |
| US20070196481A1 (en) * | 2002-07-25 | 2007-08-23 | Amidon Gregory E | Sustained-release tablet composition |
| CA2552221A1 (en) * | 2003-12-31 | 2005-07-21 | Actavis Group Hf | Donepezil formulations |
| US20070129402A1 (en) * | 2004-12-27 | 2007-06-07 | Eisai Research Institute | Sustained release formulations |
| US20090208579A1 (en) * | 2004-12-27 | 2009-08-20 | Eisai R & D Management Co., Ltd. | Matrix Type Sustained-Release Preparation Containing Basic Drug or Salt Thereof, and Method for Manufacturing the Same |
| NZ555693A (en) | 2004-12-27 | 2010-10-29 | Eisai R&D Man Co Ltd | Matrix type sustained-release preparation containing donepezil |
| US20060159753A1 (en) | 2004-12-27 | 2006-07-20 | Eisai Co. Ltd. | Matrix type sustained-release preparation containing basic drug or salt thereof |
| US20060280789A1 (en) | 2004-12-27 | 2006-12-14 | Eisai Research Institute | Sustained release formulations |
| EA014249B1 (ru) * | 2005-01-27 | 2010-10-29 | Алембик Лимитед | Формуляция леветирацетама длительного высвобождения |
| EP1874282B1 (en) * | 2005-04-06 | 2010-09-15 | Adamas Pharmaceuticals, Inc. | Methods and compositions for treatment of cns disorders |
| US20130059003A1 (en) | 2009-12-04 | 2013-03-07 | Dr. Reddy's Laboratories, Inc. | Sustained release donepezil formulations |
| US20110218216A1 (en) | 2010-01-29 | 2011-09-08 | Kumaravel Vivek | Extended release pharmaceutical composition of donepezil |
| GB201003734D0 (en) * | 2010-03-05 | 2010-04-21 | Univ Strathclyde | Delayed prolonged drug delivery |
| WO2012035409A1 (en) * | 2010-09-14 | 2012-03-22 | Rubicon Research Private Limited | Sustained release compositions of anti-alzheimer's agents |
-
2014
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- 2014-02-27 EP EP14710647.0A patent/EP2961393B1/en not_active Not-in-force
- 2014-02-27 MX MX2015011099A patent/MX378413B/es unknown
- 2014-02-27 RU RU2015140567A patent/RU2015140567A/ru not_active Application Discontinuation
- 2014-02-27 JP JP2015559595A patent/JP6429808B2/ja not_active Expired - Fee Related
- 2014-02-27 KR KR1020157026728A patent/KR102241113B1/ko not_active Expired - Fee Related
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- 2014-02-27 BR BR112015020771A patent/BR112015020771A2/pt not_active Application Discontinuation
- 2014-02-27 US US14/771,241 patent/US20160015698A1/en not_active Abandoned
- 2014-02-27 WO PCT/IB2014/059302 patent/WO2014132218A1/en not_active Ceased
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2015
- 2015-09-09 ZA ZA2015/06665A patent/ZA201506665B/en unknown
Patent Citations (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN101090738A (zh) * | 2004-12-27 | 2007-12-19 | 卫材R&D管理有限公司 | 含有碱性药物或其盐的基质型缓释制剂及其制备方法 |
| US20110237623A1 (en) * | 2010-03-01 | 2011-09-29 | Adel Penhasi | Sustained-release donepezil formulation |
| CN102309465A (zh) * | 2010-06-30 | 2012-01-11 | 天津药物研究院 | 含盐酸多奈哌齐活性成分的缓释片及其制备方法和用途 |
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| 喻东山: "胆碱酯酶抑制药治疗阿尔茨海默病", 《医药导报》 * |
| 黄流清、邵福源: "Alzheimer病相关的睡眠障碍", 《临床精神医学杂志》 * |
Also Published As
| Publication number | Publication date |
|---|---|
| US20160015698A1 (en) | 2016-01-21 |
| MX2015011099A (es) | 2016-04-06 |
| RU2015140567A (ru) | 2017-03-31 |
| JP6429808B2 (ja) | 2018-11-28 |
| EP2961393B1 (en) | 2020-10-28 |
| KR20150123302A (ko) | 2015-11-03 |
| KR102241113B1 (ko) | 2021-04-15 |
| JP2016513133A (ja) | 2016-05-12 |
| ZA201506665B (en) | 2017-02-22 |
| EP2961393A1 (en) | 2016-01-06 |
| MX378413B (es) | 2025-03-10 |
| ES2842208T3 (es) | 2021-07-13 |
| BR112015020771A2 (pt) | 2017-07-18 |
| WO2014132218A1 (en) | 2014-09-04 |
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