ES2694297T3 - Formas cristalinas de ácido {[1-ciano-5-(4-clorofenoxi)-4-hidroxi-isoquinolina-3-carbonilo]-amino}-acético - Google Patents
Formas cristalinas de ácido {[1-ciano-5-(4-clorofenoxi)-4-hidroxi-isoquinolina-3-carbonilo]-amino}-acético Download PDFInfo
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- ES2694297T3 ES2694297T3 ES14704030.7T ES14704030T ES2694297T3 ES 2694297 T3 ES2694297 T3 ES 2694297T3 ES 14704030 T ES14704030 T ES 14704030T ES 2694297 T3 ES2694297 T3 ES 2694297T3
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- C—CHEMISTRY; METALLURGY
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- C07D—HETEROCYCLIC COMPOUNDS
- C07D217/00—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems
- C07D217/22—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the nitrogen-containing ring
- C07D217/26—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/472—Non-condensed isoquinolines, e.g. papaverine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/06—Antianaemics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Hematology (AREA)
- Diabetes (AREA)
- Epidemiology (AREA)
- Urology & Nephrology (AREA)
- Vascular Medicine (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Other In-Based Heterocyclic Compounds (AREA)
- Medicinal Preparation (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201361756361P | 2013-01-24 | 2013-01-24 | |
| US201361756361P | 2013-01-24 | ||
| PCT/US2014/012780 WO2014116849A1 (en) | 2013-01-24 | 2014-01-23 | Crystalline forms of {[1-cyano-5-(4-chlorophenoxy)-4-hydroxy-isoquinoline-3-carbonyl]-amino}-acetic acid |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ES2694297T3 true ES2694297T3 (es) | 2018-12-19 |
Family
ID=50073508
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
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| ES14704030.7T Active ES2694297T3 (es) | 2013-01-24 | 2014-01-23 | Formas cristalinas de ácido {[1-ciano-5-(4-clorofenoxi)-4-hidroxi-isoquinolina-3-carbonilo]-amino}-acético |
Country Status (15)
| Country | Link |
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| US (1) | US9643928B2 (https=) |
| EP (1) | EP2951159B1 (https=) |
| JP (1) | JP6437456B2 (https=) |
| KR (1) | KR102233081B1 (https=) |
| CN (1) | CN105452227B (https=) |
| AU (1) | AU2014209319B2 (https=) |
| CA (1) | CA2899024C (https=) |
| DK (1) | DK2951159T3 (https=) |
| ES (1) | ES2694297T3 (https=) |
| IL (1) | IL240066B (https=) |
| MX (1) | MX360048B (https=) |
| RU (1) | RU2666144C2 (https=) |
| SG (2) | SG10202009266PA (https=) |
| TW (1) | TWI685487B (https=) |
| WO (1) | WO2014116849A1 (https=) |
Families Citing this family (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA2528232C (en) | 2003-06-06 | 2010-05-25 | Fibrogen, Inc. | Novel nitrogen-containing heteroaryl compounds and their use in increasing endogenous erythropoietin |
| WO2010056767A1 (en) | 2008-11-14 | 2010-05-20 | Fibrogen, Inc. | Thiochromene derivatives as hip hydroxylase inhibitors |
| KR20210130849A (ko) | 2012-07-16 | 2021-11-01 | 피브로겐, 인크. | 프롤릴 하이드록실라제 억제제 [(4-하이드록시-1-메틸-7-페녹시-아이소퀴놀린-3-카보닐)-아미노]-아세트산의 결정형 |
| EP2872487B1 (en) | 2012-07-16 | 2017-04-26 | Fibrogen, Inc. | Process for making isoquinoline compounds |
| US8883823B2 (en) | 2012-07-16 | 2014-11-11 | Fibrogen, Inc. | Crystalline forms of a prolyl hydroxylase inhibitor |
| CA2899024C (en) | 2013-01-24 | 2022-01-04 | Fibrogen, Inc. | Crystalline forms of {[1-cyano-5-(4-chlorophenoxy)-4-hydroxy-isoquinoline-3-carbonyl]-amino}-acetic acid |
| KR20210104173A (ko) | 2013-06-06 | 2021-08-24 | 피브로겐, 인크. | Hif 하이드록실라제 억제자의 약학적 제형 |
| JP6506390B2 (ja) | 2014-09-02 | 2019-04-24 | サンシャイン・レイク・ファーマ・カンパニー・リミテッドＳｕｎｓｈｉｎｅ Ｌａｋｅ Ｐｈａｒｍａ Ｃｏ．，Ｌｔｄ． | キノリノン系化合物及びその薬物への使用 |
| WO2021186356A1 (en) * | 2020-03-17 | 2021-09-23 | Cadila Healthcare Limited | Formulation comprising hif prolyl hydroxylase inhibitors |
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-
2014
- 2014-01-23 CA CA2899024A patent/CA2899024C/en active Active
- 2014-01-23 US US14/763,127 patent/US9643928B2/en not_active Expired - Fee Related
- 2014-01-23 KR KR1020157022614A patent/KR102233081B1/ko not_active Expired - Fee Related
- 2014-01-23 EP EP14704030.7A patent/EP2951159B1/en active Active
- 2014-01-23 DK DK14704030.7T patent/DK2951159T3/en active
- 2014-01-23 ES ES14704030.7T patent/ES2694297T3/es active Active
- 2014-01-23 SG SG10202009266PA patent/SG10202009266PA/en unknown
- 2014-01-23 JP JP2015555276A patent/JP6437456B2/ja not_active Expired - Fee Related
- 2014-01-23 SG SG11201505748UA patent/SG11201505748UA/en unknown
- 2014-01-23 CN CN201480016402.9A patent/CN105452227B/zh not_active Expired - Fee Related
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- 2014-01-23 TW TW103102462A patent/TWI685487B/zh not_active IP Right Cessation
- 2014-01-23 AU AU2014209319A patent/AU2014209319B2/en not_active Ceased
- 2014-01-23 RU RU2015134420A patent/RU2666144C2/ru active
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2015
- 2015-07-21 IL IL240066A patent/IL240066B/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| MX360048B (es) | 2018-10-19 |
| JP2016505071A (ja) | 2016-02-18 |
| EP2951159A1 (en) | 2015-12-09 |
| JP6437456B2 (ja) | 2018-12-12 |
| CN105452227B (zh) | 2018-05-29 |
| TWI685487B (zh) | 2020-02-21 |
| CA2899024C (en) | 2022-01-04 |
| IL240066A0 (en) | 2015-09-24 |
| DK2951159T3 (en) | 2018-11-19 |
| RU2015134420A (ru) | 2017-03-03 |
| CA2899024A1 (en) | 2014-07-31 |
| MX2015009617A (es) | 2016-04-20 |
| AU2014209319A1 (en) | 2015-08-27 |
| RU2666144C2 (ru) | 2018-09-06 |
| HK1217331A1 (en) | 2017-01-06 |
| US20160002170A1 (en) | 2016-01-07 |
| KR20150129679A (ko) | 2015-11-20 |
| KR102233081B1 (ko) | 2021-03-29 |
| SG11201505748UA (en) | 2015-08-28 |
| AU2014209319B2 (en) | 2018-04-19 |
| EP2951159B1 (en) | 2018-08-22 |
| TW201444800A (zh) | 2014-12-01 |
| SG10202009266PA (en) | 2020-10-29 |
| US9643928B2 (en) | 2017-05-09 |
| CN105452227A (zh) | 2016-03-30 |
| IL240066B (en) | 2019-08-29 |
| WO2014116849A1 (en) | 2014-07-31 |
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