ES2675720T3 - Inhibidores de quinasa no selectivos - Google Patents
Inhibidores de quinasa no selectivos Download PDFInfo
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- ES2675720T3 ES2675720T3 ES14737648.7T ES14737648T ES2675720T3 ES 2675720 T3 ES2675720 T3 ES 2675720T3 ES 14737648 T ES14737648 T ES 14737648T ES 2675720 T3 ES2675720 T3 ES 2675720T3
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- A61P7/06—Antianaemics
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D241/00—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings
- C07D241/02—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings
- C07D241/10—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members
- C07D241/14—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D241/20—Nitrogen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
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- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
- Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
- Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
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- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Epidemiology (AREA)
- Endocrinology (AREA)
- Neurology (AREA)
- Cardiology (AREA)
- Obesity (AREA)
- Heart & Thoracic Surgery (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Rheumatology (AREA)
- Urology & Nephrology (AREA)
- Pain & Pain Management (AREA)
- Tropical Medicine & Parasitology (AREA)
- Physical Education & Sports Medicine (AREA)
- Pulmonology (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
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- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
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Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
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| US201361751217P | 2013-01-10 | 2013-01-10 | |
| US201361751217P | 2013-01-10 | ||
| US201361889887P | 2013-10-11 | 2013-10-11 | |
| US201361889887P | 2013-10-11 | ||
| PCT/US2014/010778 WO2014110200A1 (en) | 2013-01-10 | 2014-01-09 | Non-selective kinase inhibitors |
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| ES2675720T3 true ES2675720T3 (es) | 2018-07-12 |
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| Country | Link |
|---|---|
| US (3) | US9815815B2 (enExample) |
| EP (1) | EP3007689B1 (enExample) |
| JP (2) | JP6387488B2 (enExample) |
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| DK (1) | DK3007689T3 (enExample) |
| ES (1) | ES2675720T3 (enExample) |
| WO (1) | WO2014110200A1 (enExample) |
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| JP2016506417A (ja) * | 2013-01-10 | 2016-03-03 | プルモキネ、インコーポレイテッド | キナーゼ阻害剤の治療指標 |
| DK3007689T3 (en) | 2013-01-10 | 2018-06-14 | Pulmokine Inc | NON-SELECTIVE KINASE INHIBITORS |
| WO2014141104A1 (en) | 2013-03-14 | 2014-09-18 | Novartis Ag | 3-pyrimidin-4-yl-oxazolidin-2-ones as inhibitors of mutant idh |
| US20150044288A1 (en) * | 2013-07-31 | 2015-02-12 | Windward Pharma, Inc. | Aerosol tyrosine kinase inhibitor compounds and uses thereof |
| ES2959419T3 (es) * | 2013-10-11 | 2024-02-26 | Pulmokine Inc | Formulaciones secas por aspersión |
| BR112019008622A2 (pt) * | 2016-10-27 | 2019-07-09 | Pulmokine Inc | método para tratar uma condição |
| JP2020514747A (ja) * | 2017-03-16 | 2020-05-21 | ザ ボード オブ トラスティーズ オブ ザ レランド スタンフォード ジュニア ユニバーシティー | Ｋｒａｓ陽性癌の診断法及び治療法 |
| WO2019157337A1 (en) * | 2018-02-08 | 2019-08-15 | Pulmokine, Inc. | Formulations of kinase inhibitors and prostanoids |
| CN109574296B (zh) * | 2018-11-27 | 2021-05-07 | 合肥工业大学 | 一种从含蟹肉蛋白废水中回收蛋白的方法 |
| US11464776B2 (en) | 2019-05-16 | 2022-10-11 | Aerovate Therapeutics, Inc. | Inhalable imatinib formulations, manufacture, and uses thereof |
| SG11202112719XA (en) | 2019-05-16 | 2021-12-30 | Aerovate Therapeutics Inc | Imatinib formulations, manufacture, and uses thereof |
| EP4334300A1 (en) * | 2021-05-07 | 2024-03-13 | GB005, Inc. | Crystalline forms of n-{3-[(1s)-1-{[6-(3,4-dimethoxyphenyl)pyrazin-2-yl]amino}ethyl]phenyl}-5-methylpyridine-3-carboxamide and related products and methods |
| CA3237696A1 (en) | 2021-11-08 | 2023-05-11 | Progentos Therapeutics, Inc. | Platelet-derived growth factor receptor (pdgfr) alpha inhibitors and uses thereof |
| KR20250044883A (ko) * | 2022-08-10 | 2025-04-01 | 지비002 인코포레이티드 | 티로신 키나아제 억제제 및 폐동맥 고혈압(pah) 치료를 위한 액티빈 유형 2 수용체 길항제 병용 요법 |
| CN119930631B (zh) * | 2025-04-07 | 2025-06-24 | 山东大学 | 一种靶向ddr1受体的化合物及其衍生的放射性示踪剂 |
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2014
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- 2014-01-09 EP EP14737648.7A patent/EP3007689B1/en active Active
- 2014-01-09 AU AU2014205483A patent/AU2014205483B2/en active Active
- 2014-01-09 CN CN201480010529.XA patent/CN105142624A/zh active Pending
- 2014-01-09 WO PCT/US2014/010778 patent/WO2014110200A1/en not_active Ceased
- 2014-01-09 ES ES14737648.7T patent/ES2675720T3/es active Active
- 2014-01-09 CN CN201811323814.3A patent/CN109568319A/zh active Pending
- 2014-01-09 CA CA2897651A patent/CA2897651C/en active Active
- 2014-01-09 US US14/760,139 patent/US9815815B2/en active Active
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2017
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2018
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2019
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2020
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2023
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2024
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| JP6547042B2 (ja) | 2019-07-17 |
| AU2014205483A1 (en) | 2015-08-27 |
| US10246438B2 (en) | 2019-04-02 |
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| AU2023201605B2 (en) | 2024-08-29 |
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| CA2897651C (en) | 2021-09-21 |
| DK3007689T3 (en) | 2018-06-14 |
| AU2023201605A1 (en) | 2023-04-13 |
| EP3007689A4 (en) | 2016-07-13 |
| WO2014110200A1 (en) | 2014-07-17 |
| US9815815B2 (en) | 2017-11-14 |
| CN105142624A (zh) | 2015-12-09 |
| AU2014205483B2 (en) | 2017-11-30 |
| AU2020289802A1 (en) | 2021-01-21 |
| US10532994B2 (en) | 2020-01-14 |
| US20190248761A1 (en) | 2019-08-15 |
| CN109568319A (zh) | 2019-04-05 |
| CA2897651A1 (en) | 2014-07-17 |
| US20180162837A1 (en) | 2018-06-14 |
| AU2018201406A1 (en) | 2018-03-15 |
| AU2024259702A1 (en) | 2024-11-21 |
| EP3007689B1 (en) | 2018-03-07 |
| US20150353527A1 (en) | 2015-12-10 |
| JP2018158931A (ja) | 2018-10-11 |
| EP3007689A1 (en) | 2016-04-20 |
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