ES2647526T3 - Combinación de canagliflozina y probenecid para el tratamiento de la hiperuricemia - Google Patents
Combinación de canagliflozina y probenecid para el tratamiento de la hiperuricemia Download PDFInfo
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- ES2647526T3 ES2647526T3 ES14717246.4T ES14717246T ES2647526T3 ES 2647526 T3 ES2647526 T3 ES 2647526T3 ES 14717246 T ES14717246 T ES 14717246T ES 2647526 T3 ES2647526 T3 ES 2647526T3
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- Prior art keywords
- probenecid
- canagliflozin
- hyperuricemia
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Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/38—Heterocyclic compounds having sulfur as a ring hetero atom
- A61K31/381—Heterocyclic compounds having sulfur as a ring hetero atom having five-membered rings
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
- A61K31/19—Carboxylic acids, e.g. valproic acid
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
- A61K31/19—Carboxylic acids, e.g. valproic acid
- A61K31/195—Carboxylic acids, e.g. valproic acid having an amino group
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
- A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/06—Antigout agents, e.g. antihyperuricemic or uricosuric agents
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
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- Pain & Pain Management (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Physical Education & Sports Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Rheumatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201361786738P | 2013-03-15 | 2013-03-15 | |
| US201361786738P | 2013-03-15 | ||
| PCT/US2014/020958 WO2014149789A1 (en) | 2013-03-15 | 2014-03-06 | Combination of canagliflozin and probenecid for the treament of hyperuricemia |
Publications (1)
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| ES2647526T3 true ES2647526T3 (es) | 2017-12-22 |
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| ES14717246.4T Active ES2647526T3 (es) | 2013-03-15 | 2014-03-06 | Combinación de canagliflozina y probenecid para el tratamiento de la hiperuricemia |
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| US (2) | US20160022632A1 (enExample) |
| EP (1) | EP2968235B1 (enExample) |
| JP (2) | JP2016512817A (enExample) |
| CA (1) | CA2907079C (enExample) |
| ES (1) | ES2647526T3 (enExample) |
| WO (1) | WO2014149789A1 (enExample) |
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| CN105548378B (zh) * | 2015-12-03 | 2017-12-26 | 上海应用技术学院 | 一种卡格列净α、β异构体的分离方法 |
| WO2019087239A1 (ja) * | 2017-10-30 | 2019-05-09 | 合同会社カルナヘルスサポート | 腎症治療剤 |
| US11547685B2 (en) * | 2017-12-11 | 2023-01-10 | Mayo Foundation For Medical Education And Research | Using probenecid to treat polycystic kidney disease |
| US11554112B2 (en) | 2018-06-07 | 2023-01-17 | Herum Therapeutics International Limited | Combinations of β-lactam compounds and probenecid and uses thereof |
| CN113164439A (zh) | 2018-12-06 | 2021-07-23 | 安索治疗公司 | 用于治疗或预防痛风或高尿酸血症的方法 |
| JP2022511800A (ja) | 2018-12-06 | 2022-02-01 | アースローシ セラピューティクス，インク． | 痛風または高尿酸血症を処置または予防するための化合物の結晶形態 |
| CN112739330A (zh) | 2019-02-13 | 2021-04-30 | 伊泰伦治疗国际有限公司 | β-内酰胺化合物和丙磺舒的组合及其用途 |
| CN111057049B (zh) * | 2019-11-18 | 2021-06-01 | 杭州华东医药集团新药研究院有限公司 | 一种卡格列净半水化合物的制备方法 |
| KR20230024354A (ko) * | 2020-06-10 | 2023-02-20 | 아쓰로시 테라퓨틱스, 인크. | 만성 신장 질환을 치료 또는 예방하는 방법 |
| CN112957318A (zh) * | 2021-02-02 | 2021-06-15 | 河北科星药业有限公司 | 丙磺舒溶液及其制备方法 |
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| CN104109155A (zh) | 2003-08-01 | 2014-10-22 | 田边三菱制药株式会社 | 新颖化合物 |
| UY30730A1 (es) | 2006-12-04 | 2008-07-03 | Mitsubishi Tanabe Pharma Corp | Forma cristalina del hemihidrato de 1-(b (beta)-d-glucopiranosil) -4-metil-3-[5-(4-fluorofenil) -2-tienilmetil]benceno |
| EP2291189B1 (en) * | 2008-05-22 | 2014-10-01 | AstraZeneca AB | Method for treating hyperuricemia employing an sglt2 inhibitor and composition containing same |
| JP2013523681A (ja) * | 2010-03-30 | 2013-06-17 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | Ｓｇｌｔ２インヒビター及びｐｐａｒ−ガンマアゴニストを含む医薬組成物並びにその使用 |
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2014
- 2014-03-06 WO PCT/US2014/020958 patent/WO2014149789A1/en not_active Ceased
- 2014-03-06 US US14/774,779 patent/US20160022632A1/en not_active Abandoned
- 2014-03-06 CA CA2907079A patent/CA2907079C/en active Active
- 2014-03-06 ES ES14717246.4T patent/ES2647526T3/es active Active
- 2014-03-06 JP JP2016500694A patent/JP2016512817A/ja not_active Withdrawn
- 2014-03-06 EP EP14717246.4A patent/EP2968235B1/en active Active
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2017
- 2017-09-07 US US15/698,062 patent/US20170368025A1/en not_active Abandoned
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2019
- 2019-02-12 JP JP2019022272A patent/JP2019089825A/ja active Pending
Also Published As
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|---|---|
| CA2907079C (en) | 2021-06-22 |
| WO2014149789A1 (en) | 2014-09-25 |
| US20160022632A1 (en) | 2016-01-28 |
| EP2968235A1 (en) | 2016-01-20 |
| EP2968235B1 (en) | 2017-09-13 |
| US20170368025A1 (en) | 2017-12-28 |
| JP2019089825A (ja) | 2019-06-13 |
| JP2016512817A (ja) | 2016-05-09 |
| CA2907079A1 (en) | 2014-09-25 |
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