ES2627338T3 - Derivados de triazol útiles como antagonistas de receptores nicotínicos - Google Patents
Derivados de triazol útiles como antagonistas de receptores nicotínicos Download PDFInfo
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- ES2627338T3 ES2627338T3 ES12802484.1T ES12802484T ES2627338T3 ES 2627338 T3 ES2627338 T3 ES 2627338T3 ES 12802484 T ES12802484 T ES 12802484T ES 2627338 T3 ES2627338 T3 ES 2627338T3
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Landscapes
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Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| PCT/US2011/041866 WO2012177263A1 (en) | 2011-06-24 | 2011-06-24 | Compounds and methods of prophylaxis and treatment regarding nictonic receptor antagonists |
| WOPCT/US2011/041866 | 2011-06-24 | ||
| US201161501207P | 2011-06-25 | 2011-06-25 | |
| US201161501207P | 2011-06-25 | ||
| PCT/US2012/043880 WO2012178112A1 (en) | 2011-06-24 | 2012-06-22 | Organic compounds |
Publications (1)
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| ES2627338T3 true ES2627338T3 (es) | 2017-07-27 |
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| ES12802484.1T Active ES2627338T3 (es) | 2011-06-24 | 2012-06-22 | Derivados de triazol útiles como antagonistas de receptores nicotínicos |
Country Status (13)
| Country | Link |
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| US (4) | US9108949B2 (https=) |
| EP (1) | EP2723173B1 (https=) |
| JP (1) | JP6087911B2 (https=) |
| KR (1) | KR20140036305A (https=) |
| CN (1) | CN103717069B (https=) |
| AU (2) | AU2012272646B2 (https=) |
| BR (1) | BR112013033306A2 (https=) |
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| ES (1) | ES2627338T3 (https=) |
| IL (1) | IL230036A (https=) |
| MX (1) | MX342322B (https=) |
| RU (1) | RU2610094C2 (https=) |
| WO (3) | WO2012177263A1 (https=) |
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| WO2012177263A1 (en) * | 2011-06-24 | 2012-12-27 | Intra-Cellular Therapies, Inc. | Compounds and methods of prophylaxis and treatment regarding nictonic receptor antagonists |
| US11491150B2 (en) | 2017-05-22 | 2022-11-08 | Intra-Cellular Therapies, Inc. | Organic compounds |
| WO2019152680A1 (en) * | 2018-01-31 | 2019-08-08 | Flagship Pioneering Innovations V, Inc. | Methods and compositions for treating cancer using chrna6 inhibitors |
| US12396992B2 (en) | 2019-01-07 | 2025-08-26 | Intra-Cellular Therapies, Inc. | Organic compounds |
| WO2021008565A1 (zh) * | 2019-07-16 | 2021-01-21 | 清华大学 | 乙酰胆碱通路调节剂在治疗癌症中的用途 |
| AU2020343329C1 (en) | 2019-09-03 | 2026-02-12 | Intra-Cellular Therapies, Inc. | Methods of treatment |
| EP4238970A1 (en) * | 2022-03-03 | 2023-09-06 | InterAx Biotech AG | Modulators of ackr3 and uses thereof |
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| PE20021019A1 (es) * | 2001-04-19 | 2002-11-13 | Upjohn Co | Grupos azabiciclicos sustituidos |
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| WO2004039815A2 (en) * | 2002-11-01 | 2004-05-13 | Pharmacia & Upjohn Company Llc | Compounds having both alpha7 nachr agonist and 5ht antagonist activity for treatment of cns diseases |
| WO2004064836A2 (en) | 2003-01-22 | 2004-08-05 | Pharmacia & Upjohn Company Llc | Treatment of diseases with alpha-7 nach receptor full agonists |
| US7135575B2 (en) * | 2003-03-03 | 2006-11-14 | Array Biopharma, Inc. | P38 inhibitors and methods of use thereof |
| US20040220170A1 (en) | 2003-05-01 | 2004-11-04 | Atkinson Robert N. | Pyrazole-amides and sulfonamides as sodium channel modulators |
| JP2006525355A (ja) * | 2003-05-01 | 2006-11-09 | アボット・ラボラトリーズ | ナトリウムチャンネルモジュレーターとしてのピラゾール−アミドおよびスルホンアミド |
| EP1638944A1 (en) * | 2003-06-12 | 2006-03-29 | Eli Lilly And Company | Tachykinin receptor antagonists |
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| WO2012177263A1 (en) | 2011-06-24 | 2012-12-27 | Intra-Cellular Therapies, Inc. | Compounds and methods of prophylaxis and treatment regarding nictonic receptor antagonists |
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| EP2723173B1 (en) | 2017-04-19 |
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