ES2405531B1 - Formulaciones sólidas y su uso en el mantenimiento de la salud gastrointestinal - Google Patents
Formulaciones sólidas y su uso en el mantenimiento de la salud gastrointestinal Download PDFInfo
- Publication number
- ES2405531B1 ES2405531B1 ES201131774A ES201131774A ES2405531B1 ES 2405531 B1 ES2405531 B1 ES 2405531B1 ES 201131774 A ES201131774 A ES 201131774A ES 201131774 A ES201131774 A ES 201131774A ES 2405531 B1 ES2405531 B1 ES 2405531B1
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- solid
- peg
- mannitol
- solid formulation
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Classifications
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- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/075—Ethers or acetals
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- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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- A61K31/74—Synthetic polymeric materials
- A61K31/765—Polymers containing oxygen
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- A—HUMAN NECESSITIES
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- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
- A61K47/10—Alcohols; Phenols; Salts thereof, e.g. glycerol; Polyethylene glycols [PEG]; Poloxamers; PEG/POE alkyl ethers
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- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
- A61K47/12—Carboxylic acids; Salts or anhydrides thereof
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- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/26—Carbohydrates, e.g. sugar alcohols, amino sugars, nucleic acids, mono-, di- or oligo-saccharides; Derivatives thereof, e.g. polysorbates, sorbitan fatty acid esters or glycyrrhizin
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- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
- A61K47/36—Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
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- A—HUMAN NECESSITIES
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- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
- A61K9/0056—Mouth soluble or dispersible forms; Suckable, eatable, chewable coherent forms; Forms rapidly disintegrating in the mouth; Lozenges; Lollipops; Bite capsules; Baked products; Baits or other oral forms for animals
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
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- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2013—Organic compounds, e.g. phospholipids, fats
- A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/2031—Organic macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyethylene glycol, polyethylene oxide, poloxamers
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/10—Laxatives
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- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
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- Molecular Biology (AREA)
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- Nutrition Science (AREA)
- Biochemistry (AREA)
- Zoology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Organic Chemistry (AREA)
- Biophysics (AREA)
- Inorganic Chemistry (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (8)
| Application Number | Priority Date | Filing Date | Title |
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| GB1018647 | 2010-11-04 | ||
| GBGB1018647.6A GB201018647D0 (en) | 2010-11-04 | 2010-11-04 | Formulations |
| US41210910P | 2010-11-10 | 2010-11-10 | |
| US61/412109 | 2010-11-10 | ||
| GBGB1104049.0A GB201104049D0 (en) | 2011-03-09 | 2011-03-09 | Formulations |
| GB1104049 | 2011-03-09 | ||
| GBGB1107626.2A GB201107626D0 (en) | 2011-05-06 | 2011-05-06 | Formulations |
| GB1107626 | 2011-05-06 |
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| ES2405531A2 ES2405531A2 (es) | 2013-05-31 |
| ES2405531R1 ES2405531R1 (es) | 2013-06-07 |
| ES2405531B1 true ES2405531B1 (es) | 2014-06-11 |
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| ES201131774A Active ES2405531B1 (es) | 2010-11-04 | 2011-11-04 | Formulaciones sólidas y su uso en el mantenimiento de la salud gastrointestinal |
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| TWI535461B (zh) | 2011-03-11 | 2016-06-01 | 諾金私人有限公司 | 結腸清潔溶液、用於製備該溶液之組成物、包含該組成物或溶液之套組、與製備該溶液之方法 |
| US20130209522A1 (en) * | 2012-02-06 | 2013-08-15 | University Of Utah Research Foundation | Drug Release from a Polymer-Controlled Local Antibiotic Delivery System Using a Degradable Bone Graft |
| BR112015005270B1 (pt) | 2012-09-11 | 2022-11-01 | Norgine Bv | Composição para mistura com água, solução de limpeza de cólon, seus usos e seu kit |
| WO2014123978A2 (en) | 2013-02-05 | 2014-08-14 | University Of Utah Research Foundation | Implantable devices for bone or joint defects |
| EA034234B1 (ru) | 2013-03-15 | 2020-01-20 | Брейнтри Лабораторис, Инк. | Пероральные фармацевтические таблетированные композиции двойного применения, содержащие сульфат натрия или его комбинацию с другими сульфатными солями, и способы их получения и применения |
| EP3137167A4 (en) * | 2014-04-29 | 2017-12-20 | Colonaryconcepts LLC | Foods, systems, methods, and kits for providing electrolyte replacement |
| EP3344238A4 (en) * | 2015-09-01 | 2019-04-24 | Colonaryconcepts LLC | DEFLECTIVE FORMULATIONS AND MANUFACTURE |
| US10859512B2 (en) | 2016-06-15 | 2020-12-08 | Shimadzu Corporation | X-ray phase contrast imaging apparatus |
| FR3056109B1 (fr) | 2016-09-21 | 2019-10-11 | Pierre Fabre Medicament | Utilisation de formulations solides de polyethylene glycol dans le traitement de la constipation |
| CN112386577B (zh) * | 2019-08-16 | 2024-01-23 | 北京天衡药物研究院有限公司 | 一种治疗便秘的组合物 |
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| US5710183A (en) * | 1995-07-14 | 1998-01-20 | Halow; George M. | Laxative/antidiarrheal composition comprising polyethylene glycol and fiber bulking agent |
| CA2516291C (en) * | 2003-02-28 | 2012-02-14 | Alk-Abello A/S | Dosage form having a saccharide matrix |
| GB0409104D0 (en) * | 2004-04-23 | 2004-05-26 | Norgine Europe Bv | Compressed pharmaceutical compositions |
| AU2006244112B2 (en) * | 2005-05-06 | 2011-02-17 | Salix Pharmaceuticals, Inc. | Polyethylene glycol colonic purgative composition |
| CO5790164A1 (es) * | 2006-08-10 | 2007-08-31 | Procaps S A | Composicion farmaceutica solida que incluye en combinacion un agente regulador de la motilidad intestinal y un agente antiflatulento |
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Also Published As
| Publication number | Publication date |
|---|---|
| EA024566B1 (ru) | 2016-09-30 |
| WO2012059724A1 (en) | 2012-05-10 |
| US20160193245A1 (en) | 2016-07-07 |
| MX2013004972A (es) | 2013-08-27 |
| JP2014500246A (ja) | 2014-01-09 |
| BE1019493A3 (fr) | 2012-07-03 |
| AR083769A1 (es) | 2013-03-20 |
| EP2635264B1 (en) | 2018-05-30 |
| EP2635264A1 (en) | 2013-09-11 |
| TWI520730B (zh) | 2016-02-11 |
| NL2007716A (en) | 2012-05-07 |
| JP5872573B2 (ja) | 2016-03-01 |
| KR20130101102A (ko) | 2013-09-12 |
| MY164204A (en) | 2017-11-30 |
| EP2635264B8 (en) | 2018-07-18 |
| CN103384516A (zh) | 2013-11-06 |
| WO2012059724A8 (en) | 2013-06-06 |
| US20170296575A1 (en) | 2017-10-19 |
| EA201300539A1 (ru) | 2013-09-30 |
| NZ611148A (en) | 2015-09-25 |
| AU2011324995A1 (en) | 2013-05-02 |
| CN103384516B (zh) | 2017-02-15 |
| SG190018A1 (en) | 2013-06-28 |
| MX342181B (es) | 2016-09-20 |
| ES2405531A2 (es) | 2013-05-31 |
| NL2007716C2 (en) | 2012-11-13 |
| CA2816835A1 (en) | 2012-05-10 |
| IL225892A0 (en) | 2013-06-27 |
| TW201223522A (en) | 2012-06-16 |
| US20130225692A1 (en) | 2013-08-29 |
| BR112013010884A2 (pt) | 2016-08-02 |
| ES2405531R1 (es) | 2013-06-07 |
| AU2011324995B2 (en) | 2015-12-24 |
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